多肽合成相关文献
Reviews and mini-reviews
1. “Instrumentation for automated solid-phase peptide synthesis.” Cammish，L.E.，Kates，S.A. In
Fmoc Solid Phase Peptide Synthesis: A Practical Approach (Chan，W.，White，P.) Oxford
University Press，Oxford，1998，in press.
2. “Peptide technologies: Nuts & bolts intelligence on practical industry solutions for peptede
design，purification and production.” Kates，S.A. Current Drugs Ltd，1998，in press.
3. “Functionalized resins and linkers for solid-phase synthesis of small molecules.” Blackburn，
C.，Albericio，F.，Kates，S.A. Drugs of the Future，1997，22，1007.
4. “Polyethylene glycol-containing supports for solid-phase synthesis of peptides and
combinatorial organic libraries.” Barany，G.，Albericio，F.，Kates，S.A.，Kempe，M. In Chemistry
and Biological Application of Polyethylene Glycol，ACS Symposium Series (Harris，J.M.，
Zalipsky，S.，Eds.) American Chemical Society Books，Washington，DC，1997，239.
5. “Solid-phase peptide and small molecule synthesis.” Blackburn，C.，Albericio，F.，Kates，
S.A. In Recent Research Developments in Organic Chemistry (Pandalai，S.G.，Ed.) Transworld
Research Network，India 1997，1，477.
6. “Solid-phase synthesis of cyclic homodetic peptides.” Blackburn，C.，Kates，S.A. In Methods
of Enzymology (Fields，G.B.，Ed.) Academic Press，New York，1997，289，175.
7. “N-[(dimethylamino)-1H-1,2,3-triazolo[4,5-b]pyridin-1-ylmethylene]-N-methylmethanaminium hexafluorophosphate N-oxide.” Albericio，F.，Kates，S.A.，Carpino，L.A. In Encyclopedia
of Reagents for Organic Synthesis (Paquette，L.A.，Ed.) Wiley， New York，1996，3，2026.
8. “3-Hydroxy-3H-1,2,3- triazolo[4,5-b]pyridin.” Kates，S.A.，Albericio，F，Carpino，L.A. In
Encyclopedia of Reagents for Organic Synthesis (Paquette，L.A.，Ed.) Wiley， New York，1996，
4，2784.
9. “Azidotris(dimethylamino)phosphonium hexafluorophosphaste.” Albericio，F.，Kates，S.A. In
Encyclopedia of Reagents for Organic Synthesis (Paquette，L.A.，Ed.) Wiley， New York，1996，
1，224.
10. “1,1’-Axobis-1-cyclohexanenitrile(ACN).” Kates，S.A.，Albericio，F. In Encyclopedia of
Reagents for Organic Synthesis (Paquette，L.A.，Ed.) Wiley， New York，1996，1，228.
11. “1-Phenylsulfonyl-1H-tetrazole.” Eritja，R.，Kates，S.A.，Albericio，F. In Encyclopedia of
Reagents for Organic Synthesis (Paquette，L.A.，Ed.) Wiley， New York，1996，6，4058.
12. “1-benzotriazolyl diethyl phosphate.” Albericio，F. Kates，S.A. In Encyclopedia of Reagents
for Organic Synthesis (Paquette，L.A.，Ed.) Wiley， New York，1996，1，300.
13.
“O-Benzoriazol-1-yl-N,N,N’,N’-tetramethyluronium
hexafluorophosphate
(HBTU)”.
Albericio，F.，Kates，S.A. In Encyclopedia of Reagents for Organic Synthesis (Paquette，L.A.，
Ed.) Wiley， New York，1996，1，304.
14. “4,4’-Bis(2-amino-6-methylpyrimidyl) disulfide.” Albericio，F.，Kates，S.A.，Eritja，R. In
Encyclopedia of Reagents for Organic Synthesis (Paquette，L.A.，Ed.) Wiley， New York，1996，
1，421.
15. “Solid-phase synthesis of cyclic peptides.” Kates，S.A.，Solé，N.A.，Albericio，F.A.，Barany，
G. In Peptides: design，synthesis and biological activity (Basava，C.，Anantharamaiah，G.M.Eds.)
Birkhauser，Boston(Massachusetts)，1994，39.
16. “Synthetic Peptides Come of Age.” Fishman，J.B.，Kates，S.A. Biomedical Products Review，
1995，20，52.
Article in refereed journals
1. “Continuous-flow solid-phase peptide sysnthesis using polystryrene resins.” Kates，S.A.，
Cammish，L.E.，Albericio，F.J. Peptide Science，1998，in press.
2. “On the uniformity of product quality for peptides generated in service laboratories: Peptides
containing phosphorylated tyrosone residues.” Bonewald，L.F.，Bibbs，L.，Kates，S.A.，Khatri，
A.，McMurray，J.S.，Medzihradszky，K.F.，Weintraub，S.T. J. Peptide Science，1998，in press.
3. “Improved synthesis and purification of Alzeimer’s Ab 1-42 and analogs.” Milton，S.C.F.，de
Lisle Milton，R.C.，Kates，S.A.，Glabe，C. Letters in peptide Science，1998，in press.
4. “High load” Polyethylene glycol-polystryrene (PEG-PS) graft supports for solid-phase
synthesis.” Kates，S.A.，Blackburn，C.，McGuinness，B.F.，Griffin，G.W.，Solé，N.A.，
Barany，G.，Albericio，F. Biopolymers: Peptide Science，1998，in press.
5. “On the Use of Onium Salt-Based Coupling Reagents in Peptide Synthesis” Albericio，F.，
Bofill，J.M.，Carpino，L.A.，El-Faham，A.，Kates，S.A. J.Org. Chem. 1998，in press.
6. “Automated，high productivity purification and analysis of synthetic peptides.” Londo，T.R.，
Kehoe，T.，Kates，S.A.，Hantman，S.，Gordon，N.F. Letters in Peptide Science，1998，in press.
7. “On the use of PyAOP，a phosphonium salt derived from HOAt，in solid-phase peptide
synthesis.” Albericio，F.，Cases，M.，Alsina，J,.，Triolo，S.A.，Carpino，L.A.，Kates，S.A.
Tetrahedron Lett.，1997，38，4853.
8. “N-Dependent transcriptional antitermination in phage λis mediated by an inducible RNA
bridge.” Su，L.，Radek，J.T.，Labeots，L.A.，Hermanto，P.，Chem，H.，Nakagawa，S.，
Zhao，M.，Kates，S.A.，Weiss，M.A. Genes & Development，1997，11，2214.
9. “Optimization of the synthesis of peptide combinatorial libraries (SPCLs) using a one-pot
method.” Herman，L.W.，Tarr，G.，Kates，S.A. Molecular Diveristy，1996，1，147.
10. “Solid-phase synthesis of angiotensin converting enzyme (ACE) inhibtor libraries derived
from N-alkylated dipeptide.” Blackburn，C.，Pingali，A.，Kehoe，T.，Herman，L.W.，Wang，
H.，Kates，S.A. Bioorg. Chem. Med. Lett. 1997，7，823.
11. “N-Piperidylalanine formation during the preparation of C-terminal Cys peptides with an
Fmoc/tBu strategy.” Lukszo，J.，Patterson，D.，Albericio，F.，Kates，S.A. Lett. Peptide Science，
1996，3，157.
12. “Labeling of synthetic biomolecules with biotin and fluorescein by active esters of
1-phenylpyarzolin-5-ones.” Kremsky，J.N.，Pluskal，M.，Casey，S.，Perry-O’Keefe，H.，Sinha，
N.D.，Kates，S.A. Tetrahedron Lett. 1996，37，4313.
13. “Preparation and applications of xanthenylamide (XAL) handles for solid-phase synthesis of
C-terminal peptide amides under particularly mild conditions.” Han，Y,.，Bontems，S.L.，Hegyes，
P.，Munson，M.C.，Minor，C.A.，Kates，S.A.，Albericio，F.，Barany，G. J. Org. Chem.，
1996，61，6326.
14. “Optimized preparation of deca(L-alanyl)-L-valinamide by 9-fluorenylmethyloxycarbonyl
(Fmoc) Solid-phase synthesis on polyethylene glycol-polystyrene (PEG-PS) graft supports，with
1,8-diazobicyclo[5.4.0]-undec-7-ene (DBU) deprotection.” Kates，S.A.，Solé，N.A.，beyermann，
M.，Barany，G.，Albericio，F. Peptide Res.，1996，9，106.
15. “Novel carbozylic acid and carboxamide protective groups based on the exceptional
stablization of the cyclopropylmethyl cation.” Carpino，L.A.，Chao，H.-G.，Ghassemi，S.，
Mansour，E.M.E.，Riemer，C.，Warrass，R.，Sadat-Aalaee，D.，Truran，G.A.，Imazumi，
H.，El-Faham，A.，Ionescu，D.，Ismail，M.，Kowaleski，T.L.，Han，C.H.，Wenschuh，
H.，Beyermann，M.，Bienert，M.，Shroff，H.，Alericio，F.，Triolo，S.A.，Solé，N.A.，
Kates，S.A，J. Org. Chem.，1995，60，7718.
16. “Rearrangement of Glu(OtBu) and Asp(OtBu)-containing peptides upon fluoride treatment in
solid-phase synthesis.” Kates，S.A.，Albericio，F. Lett.Pep.Sci.，1995，1，213.
17. “Structural studies of reagents for peptide bond formation: Crystal and molecular structures of
HBTU and HATU.” Abdelmoty，I.，Albericio，F.，Carpino，L.A，Foxman，B.M.，Kates，
S.A. Lett. Peptide Science 1994，1，57.
18. “Solid-phase N-glycopeptide synthesis using allyl side-chain protected Fmoc-amino acids.”
Kates，S.A.，De la Torre，B.G.，Erijua，R.，Albericio，F. Tetrahedron Lett. 1994，35，1033.
19. “Automate allyl deprotection for continuous-flow synthesis of cyclic and branch peptide.”
Kates，S.A.，Daniels，S.B.，Albericio，F. Anal. Biochem. 1993，212，303.
20. “A novel，
convenient，
three-dimensional orthogonal strategy for solid-phase synthesis of cyclic
peptides.” Kates，S.A.，Solé，N.A.，Johnson，C.R.，Hudson，D.，Barany，G.，Albericio，
F. Tetrahedron Lett. 1993，34，1549.
21. “The development of high-performance liquid chromatographic analysis of allyl and
allyloxycarbonyl side-chain-protected phenylthiohydanoin amino acids.” Fields，C.G.，Loffet，
A.，Kates，S.A.，Fields，G.B. Anal. Biochem. 1992，203，245.
22. “Manganese (Ⅲ) based oxidative free-radical cyclization of unsaturated β-keto esters，
1,3-diketones and malonate diesters.” Kates ， S.A. ， Dombroski ， M.A. ， Snider ， B.B.
J.Org.Chem.1990，55，2427.
23. “Manganese (Ⅲ) based oxidative free-radical tandem and triple cyclizations.” Dombroski，
M.A.，Kates，S.A.，Snider，B.B. J.Am.Chem.Soc. 1990，112，2759.
24. “Formation of seven- and eight-membered rings by manganese (Ⅲ) based oxidative free
radical cyclizations.” Merritt，J.E.，Sasson，M.，Kates，S.A.，Snider，B.B. Tetrahedron Lett.
1988，29，5209.
25. “Mechanism of manganese (Ⅲ) based oxidative ofβ-ketoesters.” Snider，B.B.，Patricia，J.J.，
Kates，S.A. J.Org.Chem. 1988，53，2137.
26. “Manganese ( Ⅲ ) based oxidative free-radical cyclization. 3.Polycyclization reactions
proceeding through secondary radicals.” Mohan，R.，Kates，S.A.，Dombroski，M.A.，Snider，
B.B. Tetrahedron Lett. 1987，28，845.
27. “Manganese ( Ⅲ ) based oxidative free-radical cyclization. 2.Polycyclization reactions
proceeding through tertiary cations.” Snider，B.B.，Mohan，R.，Kates，S.A. Tetrahedron Lett.
1987，28，841.
28. “Manganese (Ⅲ) based oxidative free-radical cyclization. Synthesis of (±)-podocarpic acid.”
Snider，B.B.，Mohan，R.，Kates，S.A. J.Org.Chem. 1985，50，3659.
Other articles
1. “A comparison of solid-phase techniques for the construction of chemokines.” McNamara，J.F.，
Lombardo，H.，Pillai，S.K.，Jensen，I.，Kates，S.A. In Peptides 1998 Proceedings of the
Twenty-Fifth European Peptide Symposium (Bajusz，S.，Judecz，F.，Eds.) Mayflower Worldwide
Limited， Birmingham，England，1999，in press.
2. “Design and synthesis of cyclic peptides for iron-sulfur cluster assembly and encapsulation.”
Segal，B.M.，McNamara，J.F.，Jensen，I.，Kates，S.A.，Holm，R.H. In Peptides 1998 Proceedings
of the Twenty-Fifth European Peptide Symposium (Bajusz，S.，Judecz，F.，Eds.) Mayflower
Worldwide Limited， Birmingham，England，1999，in press.
3. De novo peptide design as an approach for the synthesis of a sturctural representation of the
center A active site of carbon monoxide dehydrogenase/acetyl-CoA synthase.” Laplaza，C.E.，
McNamara，J.F.，Jensen，I.，Kates，S.A.，Holm，R.H. In Peptides 1998 Proceedings of the
Twenty-Fifth European Peptide Symposium (Bajusz，S.，Judecz，F.，Eds.) Mayflower Worldwide
Limited， Birmingham，England，1999，in press.
4. “Design and synthesis of cyclic cysteine-containing peptides for transition metal incorporation.”
Nivorozhkin，A.L.，Kates，S.A.，Holm，R.H. In Peptides 1998 proceedings of the Twenty-Fifth
European Peptide Symposium (Bajusz，S.，Judecz，F.，Eds.) Mayflower Worldwide Limited，
Birmingham，England，1998，in press.
5. “Solid-phase synthesis of “head-to-tail” cyclic and C-terminal modified peptides.” Albericio，
F.，Frieden，A.，Del Fresno，M.，Royo，M.，Alsina，J.，Jensen，K.J.，Kates，S.A.，Barany，
G. In Innovation and Perspectives in Solid Phase Synthesis and Combinatorial Chemical Libraries
(Epton，R.，ed.) Mayflower Worldwide Limited， Birmingham，England，1998，in press.
6. “Homodetic cyclic peptides via solid-phase synthesis.” Blackburn，
C.，
Kates，S.A. In Innovation
and Perspectives in Solid Phase Synthesis and Combinatorial Chemical Libraries (Epton，R.，ed.)
Mayflower Worldwide Limited， Birmingham，England，1998，in press.
7. “Handles for solid-phase chemistry: Progress from peptide to small molecule synthesis.”
Blackburn，C.，Barany，G.，Albericio，F.，Kates，S.A. In Innovation and Perspectives in Solid
Phase Synthesis and Combinatorial Chemical Libraries (Epton，R.，ed.) Mayflower Worldwide
Limited， Birmingham，England，1998，in press.
8. “A comparison of solid supports for PNA synthesis.” Casale，R.A.，Paul，C.H.，Jensen，I.S.，
Moyer，M.L.，Kates，S.A.，Egholm，M. In Innovation and Perspectives in Solid Phase Synthesis
and Combinatorial Chemical Libraries (Epton，R.，ed.) Mayflower Worldwide Limited，
Birmingham，England，1998，in press.
9. “Backbone amide Linker (BAL) for solid-phase synthesis of 2,5-piperazinediones (DKP)，
useful scaffolds for combinatorial chemistry.” Albericio，F.，del Fresnl，M.，Alsina，J.，Frieden，
A.，Royo，M.，Jensen，K.J.，Kates，S.A.，Barany，G. In Peptides-Chemistry and Biology:
Proceedings of the Fourteenth American Peptide Symposium (Tam，J.) 1998，Escom，in press.
10. “Encoding schemes for application with polyethylene glycol-polystyrene graft (PEG-PS)
supports in solid-phase peptide and small molecule synthesis.” Kates，S.A.，Hines，W.H.，Kelley，
M.A.，Lynch，P.，Albericio，F.，Barany，G. In Peptides-Chemistry and Biology: Proceedings of
the Fourteenth American Peptide Symposium (Tam，J.) 1998，Escom，in press.
11. “1997 ABRF peptide synthesis research committee study on a peptide containing a
phosphorylated tyrosine.” Bonewald，L.F.，Bibbs，L.，Kates，S.A.，Khatri，A.，Medzihradxzky，
K.F.，McMurray，J.S.，Weintraub，S. In Peptides-Chemistry and Biology: Proceedings of the
Fourteenth American Peptide Symposium (Tam，J.) 1998，Escom，in press.
12. “Polyethylene glycol-containing supports for solid-phase synthesis of peptides and
combinatorial organic libraries.” Barany，G.，Albericio，F.，Kates，S.A.，Kempe，M. Polymer
Preprints Am. Chem. Soc. Div. Polym. Chem.，1997，38，587.
13. “Synthesis of Alzheimer’s (1-42) Aβ-amyloid peptide with preformed Fmoc-aminoacyl
fluorides.” Milton，S.C.F.，Milton，R.C.d.L.，Kates，S.A.，Glabe，C. In Techniques in Protein
Chemistry Ⅷ (Marshak，D.R.，Ed.) 1997，Academic Press，San Diego，CA，865.
14. “Recent aspects of the use of tetramethylfluorofomamidinium hexafluorophosphate (TFFH) as
a convenient peptide coupling reagent.” Triolo, S.A., Ionescu, D., Wenschuh, H., Solé, N.A.,
El-Faham, A., Carpino, L.A., Kates, S.A. In Peptides 1996 Proceedings of the Twenty-Fourth
European Peptide Symposium (Ramage, R., Ed.) 1997, Mayflower Worldwide Limited,
Birmingham, England, 839.
15. “PioneerTM: A continuous-flow peptide synthesis system.” Daniels, S.B., Solé, N.A., Hantman,
S.F., Gibney, B.R., Rabanal, F., Kates, S.A., In Peptides 1996 Proceedings of the Twenty-Fourth
European Peptide Symposium (Ramage, R., Ed.) 1997, Mayflower Worldwide Limited,
Birmingham, England, 323.
16. “Crystal and solution structures of HBPyU and HAPyU.” Henklein, P., Costisella, B., Wray, V.,
Domke, T., Carpino, L.A., El-Faham, A. Kates, S.A., Abdelmoty, I., Foxman, B.M. In Peptides
1996 Proceedings of the Twenty-Fourth European Peptide Symposium (Ramage, R., Ed.) 1997,
Mayflower Worldwide Limited, Birmingham, England, 465.
17. “New coupling techniques for solid-phase peptide synthesis.” Kates, S.A., Carpino, L.A.,
Albercio, F. In Peptides-Chemistry and Biology: Proceedings of the Fourteenth American Peptide
Symposium (Kaumaya, P.T.P., Hodges, R.S., Eds.) 1996, Mayflowers Worldwide Limited,
Birmingham, England, 893.
18. “Recent developments in azabenzotriazole-based coupling reagents for use in solid-phase
peptide synthesis: PyAOP and HAPyU.” Kates, S.A., Triolo, S.A., Diekmann, E., Carpino, L.A.,
El-Faham, A., Ionescu, D., Albericio, F. In Peptides-Chemistry and Biology: Proceedings of the
Fourteenth American Peptide Symposium (Kaumaya, P.T.P., Hodges, R.S., Eds.) 1996,
Mayflowers Worldwide Limited, Birmingham, England, 115.
19. “High load polyethylene glycol-polystyrene graft supports for solid-phase peptide synthesis.”
McGuinness, B.F., Kates, S.A., Grifin, G.W., Herman, L.W., Solé, N.A., Vágner, J., Albercio, F.,
Barany, G. In Peptides-Chemistry and Biology: Proceedings of the Fourteenth American Peptide
Symposium (Kaumaya, P.T.P., Hodges, R.S., Eds.) 1996, Mayflowers Worldwide Limited,
Birmingham, England, 125.
20. “On the use of novel coupling reagents for solid-phasepeptide synthesis.” Kates, S.A.,
Diekmann, E., El-Faham, A., Herman, L.W., Ionescu, D., McGuinness, B.F., Triolo, S.A.,
Albericio, F., Carpino, L.A., In Techniques in Protein Chemistry Ⅶ (Marshak, D.R., Ed.) 1996,
Academic Press, San Diego, CA, 515.
21. “Advances in the use of onium-based coupling reagents: application for solid-phase peptide
synthesis and combinatorial libraries.” Kates, S.A., Triolo, S.A., Griffin, G.W., Herman, L.W., Tarr,
G., Solé, N.A., Diekmann, E., El-Faham, A., Ionescu, I., Albericio, F., Carpino, L.A. In Innovation
and Perspectives in Solid Phase Synthesis and Combinatorial Chemical Librariers (Epton, R., Ed.)
1997 Mayflower Worldwide Limited, Birmingham, England, 41.
22. “Use of XAL handles for solid-phase synthesis of peptide amides.” Kates, S.A., Minor, C.A.,
Han, Y., Albericio, F., Barany, G. In Peptides 1994: Proceedings of the Twenty-third European
Peptide Symposium (Maia, H.L.S., Ed.) 1995, Escom, Science Publishers, Leiden, The
Netherlands, 262.
23. Practival
Protocols
for
efficient
solid-phasepeptide
synthesis.
Minimization
of
side-reactions.” Kates, S.A., Minor, C.A., Shroff, H., Haaseth, R.C., Triolo, S., El-Faham, A.,
Carpino, L.A., Albericio, F. In Peptides 1994: Proceedings of the Twenty-third European Peptide
Symposium (Maia, H.L.S., Ed.) 1995, Escom, Science Publishers, Leiden, The Netherlands, 248.
24. “Polyethylene glycol-polystryrene (PEG_PS) supports for Boc solid-phase peptide and PNA
synthesis strategies.” Albericio, F,. Bacardit, J., Barany, G., Coull, J.M., Egholm, M., Giralt, E.,
Griffin, G.W., Kates, S.A., Nicolás, E., Solé, N.A. In Peptides 1994: Proceedings of the
Twenty-third European Peptide Symposium (Maia, H.L.S., Ed.) 1995, Escom, Science Publishers,
Leiden, The Netherlands, 271.
25. “Azabenzotriazole (HOAt) derivatives as superior coupling reagents for peptide synthesis.”
Albericio, f., Abdelmoty, I., Bofill, J.M., Carpine, L.A., El-Faham,A., Foxman, B.M., Gairí, M.
Giralt, E., Griffin, G.W., Kates, S.A., Lloyd-Williams, P., Minor, C.A., Scarmoutzos, L.W., Shroff,
H., Triolo, S., henschuh, H. In Peptides 1994: Proceedings of the Twenty-third European Peptide
Symposium (Maia, H.L.S., Ed.) 1995, Escom, Science Publishers, Leiden, The Netherlands, 23.
26. “New approaches for extending the scope of solid-phase peptide synthesis.” Carpino, L.A.,
El-Faham. A., Truran, G.A., Minor, C.A., Kates, S.A., Griffin, G.W., Shroff, H., Triolo, S.A.,
Albericio,F. In Innovation and perspectives in Solid Phase Synthesis-Peptides, Proteins and
Nucleic Acids (Epton, R., Ed.) 1994 Mayflower Worldwide Limited, Birmingham, England, 95.
27. “Orthogonal Solid-phase synthesis of bicyclic peptides.” Solé, N.A., Kates, S.A., Albericio, F.,
Barany, G. In Innovation and perspectives in Solid Phase Synthesis-Peptides, Proteins and Nucleic
Acids (Epton, R., Ed.) 1994 Mayflower Worldwide Limited, Birmingham, England, 105.
28. “Orthogonal Solid-phase synthesis of bicyclic analogues of αconotoxin SI.” Solé, N.A.,
Kates, S.A., Albericio, F., Barany, G. In Innovation and perspectives in Solid Phase
Synthesis-Peptides, Proteins and Nucleic Acids (Epton, R., Ed.) 1994 Mayflower Worldwide
Limited, Birmingham, England, 93.
29. “Automated allyl chemistry forsolid-phase peptide synthesis: Applications to cyclic and
Branched peptides.” Kates, S.A., Daniels, B.B., Solé, N.A., Barany, G., Albericio, F. In
Peptides-Chemistry and Biology: proceedings of the Thirteenth American Peptide symposium
(Hodges, R., S., Smith J.A., Eds.) 1994 Escom, Science Publishers, Leiden, The Netherlands, 113.
30. “Azabenzotriazole-based coupling reagents in solid-phase peptide sythesis.” Carpino, L.A.,
El-Faham, A., Truran, G.A., Triolo, S.A., Shroff, H., Griffin, G.W., Minor, C.A., Kates, S.A.,
Albericio, F. In Peptides-Chemistry and Biology: proceedings of the Thirteenth American Peptide
symposium (Hodges, R., S., Smith J.A., Eds.) 1994 Escom, Science Publishers, Leiden, The
Netherlands,124.
31. “Allyl-based orthogonal solid-phase peptide synthesis.” Albericio, F., Barany, G., Fields, G.B.,
Hudson, D., Kates, S.K., Lyttle, M.H., Sole N.A. In Peptides 1992: Proceedings of the
Twenty-second European Peptide Symposium (Schneider, C.H., Eberle, Eds.) 1993, Escom ,
Science Publishers, Leiden, The Netherlands, 191.
32. “Novel polyethylene glycol-polystyrene (PEG-PS) graft supports for solid-phase peptide
synthesis.” Barany, G., Albericio, F., Sole, N.A., Griffin, G.W., Kates, A.A., Hudson, D. In
Peptides 1992: Proceedings of the Twenty-second European Peptide Symposium (Schneider, C.H.,
Eberle, Eds.) 1993, Escom , Science Publishers, Leiden, The Netherlands, 267.
33. “New approaches in solid-phase peptide synthesis.” Albericio, F., Carpino, L.A., Daniels, S.B.,
El-Faham, A., Fukuda, H., Griffin, G.W., Kates, S.A., Minor, C.A., Shroff, H.N., Triolo, S.A.,
Truran, G.T., Yamabe, K., In “Peptide Chemistry 1993: Proceedings of the 31th Symposium on
Peptide Chemistry (Okada, Y, Ed.) 1994, Protein Research Foundation, 121.
Patents:
“Automated allyl deprotection in solid-phase synthesis.” Albericio, F., Kates, S.A. submitted
1993, awarded 1998.
Abstracts:
1. Susumu Funakoshi, G. William Griffin, Derek Hudson, Steven A. Kates, Mattew H. Lyttle,
Hitesh Shroff, Nuria A. Solé, and Salvatore A. Triolo. Effective strategies for chemical
synthesis of peptides. Twenty-second European Peptide Symposium-Millipore Forum.
September, 1992, Interlaked (Switzerland).
2. Fernando Albericio, George Barany, Gregg. B. Fields, Hiroyuki Fukuda, Susumu Funakoshi,
Hiroyuki Fukuda, Nobutaka Fjjii, Fernando Albericio, Steven A, Kates, Vishnu C. Solan, and
Salvatore A. Triolo. Biolinker: An affinity purification procedure for synthetic peptides.
Thirteenth American Peptide Symposium. June, 1993. Edmonton (Canada).
3. Steven A. Kates, G. William Griffin, Charles A. Minor, Nuria A. Solé, George Barany, and
Fernando Albericio. New methods for the solid-phase synthesis of cyclic, branched, and
multiple antigenic (MAP) peptides. Seven Symposium of the Protein Society. July, 1993, San
Diego (California).
4. Fernando Albericio, Louis A. Carpino, Ayman El-Faham, G. William Griffin ,Steve A. Kates,
Charles A. Minor, Hitesh N. Shroff, Salvatore A Triolo, George A. Truran. Science
Innovation ’93 of the American Association for the Advancement of Science. August, 1993.
Boston (Massachusetts.)
5. Steven A. Kates, G. William Griffin, Yonxin Han, Brian F. McGuinness, Joan McNeil, Charles
A. Minor, Nuriá A. Solé, Michael F. Songster, Josef Vágner, Fernando Albericio, and George
Barany. Improved handles and supports for solid-phase peptide synthesis. Ninth symposium of
the Protein Society. July, 1995. Boston (Massachusetts).
6. Michael F. Songster, Steven A. Kates, Fernando Albericio, and George Barany. Use of HAL
(hypersensitive acid-labile) handle for solid-phase synthesis of peptide acids. Fourteenth
American Peptide Symposium June 1995, Columbus (Ohio).
7. Iman Abdelmoty, Fernando Albericio, Josep M. Bofill, Burce M.Foxman, and Steven A. Kates.
The solid state structures of HATU and HBTU: A reexamination. Fourteenth American Peptide
Symposium June 1995, Columbus (Ohio).
8. Steven A. Kates, Solid-phase synthesis of cyclic peptides. Peptide Synthesis Workshop Tenth
Annual Meeting of the Association of Biomolecular Resource Facilities, July 1995, Boston
(Massachusetts).
9. Aruna Pingali, Christopher Blackburn, Lee W. Herman, Hongqi Wang, Steven A. Kates.
Solid-phase synthesis and affinity selection of ACE inhibitor libraries derived from N-alkylated
dipeptides. First Annual Solid-Phase Synthesis. Developing Small Molecule Libraries,
Cambridge HealthTech Institute, February 1996, San Diego (California).
10. Christopher Blackburn, Lee W. Herman, Nuriá A. Solé, Salvatore A. Triolo, Steven A. Kates.
Reagents for solid-phase peptide and small molecule combinatorial synthesis. First Annual
Solid-Phase Synthesis, Developing Small Molecule Libraries, Cambridge HealthTech Institute,
February 1996, San Diego (California).
11. Steven A. Kate, Christopher Blackburn, Lee W. Herman, Elizbeth A. Luchow, Savatore A.
Triolo. Onium-based coupling reagent and high-load polyethylene glycol-polystyrene (PEG-PG)
supports: Tools for solid-phase peptide and small molecule combinatorial synthesis.
Associaiton of Biomolecular Resource Facilities, April 1996, San Francisco, (California).
12. Christopher Blackburn, Lee W. Herman, Nuriá A. Solé, Salvatore A. Triolo, Steven A. Kates.
Reagents for solution and solid-phase peptide and small molecule combinatorial synthesis.
Tenth Symposium of the Protein Society, August,1996, San Jose (California).
13. Steven A. Kates. Solid-phase Organic Chemistry: A Peptide Chemist’s Perspective. Second
Annual Solid-Phase Synthesis, Developing Small Molecule Libraries, Cambridge Healthtech
Institute, February 1997, San Diego (California).
14. Steven A. Kates. Applications on onium-based coupling reagent for peptide and organic
solution/solid-phase method. Peptide Technologies, Nuts & Bolts Intelligence on Practical
Industry Solutions for Peptide Design, Purification and production, International Business
Communications, March 1998, Las Vegas (Nevada).
15. Sasi K. Pillai, Steven A. Kates, Subhasish Purkayastha. TFFH, A versatile reagent for organic
transformations in solid- and solution-phase. 215th American National Meeting March