Roumanian Biotechnological Letters Copyright © 2006 Bucharest University Roumanian Society of Biological Sciences Vol. 11, No. 5, 2006, pp. 2915-2921 Printed in Romania. All rights reserved ORIGINAL PAPER Extraction and transport of neutral amino acids through liquid membranes Received for publication, July 15, 2006 Accepted, September 15, 2006 ALEXANDRA CRISTINA BLAGA1), ANCA-IRINA GALACTION2), DAN CAŞCAVAL1)*, ELENA FOLESCU1) 1) Technical University "Gh. Asachi" of Iasi, Faculty of Chemical Engineering, Dept. of Biochemical Engineering, 71 D. Mangeron Avenue, 700050 Iasi, Romania, email: dancasca@ch.tuiasi.ro 2) University of Medicine and Pharmacy, Faculty of Medical Bioengineering, Dept. of Biotechnology, 16 University Street, 700115 Iasi, Romania, email: galact@from.ro * the corresponding author Abstract This study is focused on facilitated pertraction of some neutral amino acids (L-cysteine, Ltryptophan, L-glycine, L-alanine) with D2EHPA dissolved in dichloromethane. The results indicated the significant influences of the pH-gradient between the aqueous phases, carrier concentration and mixing intensity. The maximum mass flows of the amino acids through liquid membrane can be reached at the pH-value of the feed phase of 3, pH-value of the stripping solution of 1, D2EHPA concentration in solvent layer of 60 g l-1, using an intense mixing of the two aqueous phases. In function of the pH-gradient between the aqueous phases, it is possible to separate selectively the considered amino acids. Keywords: amino acids, L-cysteine, L-tryptophan, L-glycine, L-alanine, D2EHPA, pertraction, liquid membrane, carrier, mass flow, permeability factor. Introduction Biotechnology has much progressed and represents the principal way for obtaining of some very important products for human activity. In this context, the production of amino acids, which are the main structural components of proteins and enzymes, has been significantly increased. The amino acids can be obtained by biosynthesis or from protein hydrolysis, but their separation from fermentation broths or protein hydrolysates is rather difficult. Generally, the techniques used for separation or purification of amino acids include chromatography, adsorption, ion-exchange, and crystallization at the isoelectric point [1]. But these techniques are difficult to scale-up, consequently the production of amino acid is limited and the technology is rather expensive. Recently the separation of amino acids by liquid-liquid extraction has been analyzed. Because amino acids dissociate in aqueous solutions, forming characteristic ionic species as a function of the solution pH value, their solubility in organic solvents, especially in low-polar ones, is very low. The extraction of amino acids is only possible by adding into the organic phase extractants such as phosphoric acid derivatives [1-5], high molecular weight quaternary aliphatic amines [6,7] or crown-ethers [1,8,9]. 2915 ALEXANDRA CRISTINA BLAGA, ANCA-IRINA GALACTION, DAN CAŞCAVAL, ELENA FOLESCU Extraction and transport through liquid membrane, also called pertraction, represents a development of the extraction processes. This technique can be applied for amino acids separation and mainly uses emulsion liquid membranes [10-12] and supported liquid membranes [13-15]. Because the main limitations of these processes are the swelling of emulsion liquid membrane and the low stability of supported liquid membrane, the extraction and transport of amino acids can be carried out through the free liquid membranes, which do not need to stabilize the membrane by adding surfactants or by including into porous membranes or hollow fibers [1,16]. The previous studies have been focused on the separation the acidic amino acids (Laspartic and L-glutamic acids) by facilitated pertraction with di-(2-ethylhexyl) phosphoric acid (D2EHPA) [16]. In this paper, the studies are continued by analyzing the possibility to separate some neutral amino acids (L-cysteine, L-tryptophan, L-glycine, L-alanine) using the same technique, in the purpose to establish the optimum conditions required for selective separation of amino acids from fermentation broths or protein hydrolysates. Materials and methods The experiments have been carried out using a patented pertraction equipment of U-type cell, which allows obtaining and easily maintaining the free liquid membrane and was described in the previous paper [16,17]. The liquid membrane phase consists of a solution of 20 - 100 g/l D2EHPA as carrier dissolved in dichloromethane. The feed phase contains initial solutions of 3 g l-1 L-cysteine/ L-tryptophan/L-glycine/L-alanine. The pH of the feed phase varied from 2 to 6, being adjusted at the prescribed values with solutions of 4% H2SO4 or 4% NaOH. The pH of stripping solution has been adjusted with 4% HCl solution in the pH-domain of 1 to 5. The pH values were determined using a digital pHmeter of Consort C831 type. The aqueous solutions are independently mixed by means of double blades stirrers with 6 mm diameter and 3 mm height, having a rotation speed between 0 and 600 rpm. In order to reach high diffusion rates through the solvent layer, the organic phase has been mixed with one stirrer of the same design, at a constant rotation speed of 500 rpm. The area of mass transfer surface, both for extraction and for re-extraction, was of 1.59x10-3 m2. At this mixing intensity level, the interfaces between the phases remained flat, and, consequently, the interfacial area constant. The experiments have been carried out in a continuous system, at the steady state conditions for aqueous solutions, these solutions being separately fed with a volumetric flow of 1.92 l h-1. The evolution of pertraction was followed by means of the amino acid mass flows and permeability factors through liquid membrane. The initial mass flows, ni, represents the flux of amino acid transferred from the feed phase to the solver layer, and the final mass flow, nf, also called overall mass flow, represents the flux of amino acid transferred from the organic solvent to the striping phase. The permeability factor, P, is a measure of the capacity to transport the solute through the liquid membrane, being defined as the ratio between the final mass flow and the initial mass flow of amino acid. For calculating these parameters, the amino acids concentration in the feed and stripping solutions have been measured by high performance liquid chromatography technique (HPLC) with a HP 1090 liquid chromatography, then the mass balance being used. 2916 Roum. Biotechnol. Lett., Vol. 11, No. 5, 2915-2921 (2006) Extraction and transport of neutral amino acids through liquid membranes Results and discussion Extraction and transport through liquid membranes is strongly influenced by the pHgradient between the feed and stripping phases, carrier concentration in liquid membrane, and mixing intensity of the three phases. In the case of amino acids pertraction, the influence of the pH-gradient between is enhanced by the formation of the ionized forms of amino acids in the aqueous phases and controls the efficiency both of extraction/re-extraction and the transport rate through the solvent layer. Thus, from Figure 1 it can be observed that for all studied neutral amino acids the initial mass flows increase with the increase of feed phase pH, reach a maximum value at pH = 3, followed by their strong decrease. L-Cysteine L-Tryptophan 1.0 -1 1.0 -2 n, moles m h P -2 n, moles m h -1 1.0 0.8 0.8 0.6 0.6 0.4 P 0.8 0.8 0.6 0.6 0.4 ni nf P 0.2 0.4 0.4 ni nf P 0.2 0.2 0.0 0.0 0.2 2 3 4 5 2 6 3 4 pH of feed phase L-Glycine L-Alanine 1.0 1.0 1.0 -2 0.8 0.6 0.6 0.4 -2 -1 P n, moles m h -1 0.8 n, moles m h 5 6 pH of feed phase P 0.8 0.8 0.6 0.6 0.4 ni nf P 0.2 0.4 0.2 0.0 2 3 4 5 6 0.4 ni nf P 0.2 0.2 0.0 2 pH of feed phase 3 4 5 6 pH of feed phase Figure 1. Variation of the amino acids mass flows and permeability factor in function of the pH-value of the feed phase (pH of stripping phase = 2, D2EHPA concentration = 40 g l -1, rotation speed = 500 rpm). This evolution is the result of the reactive extraction mechanism of amino acids with D2EHPA, which occurs by means of an interfacial chemical reaction of ionic exchange type controlled by the pH of aqueous phase. The carrier, D2EHPA, reacts only if the amino acids exist in aqueous solution in their cationic form (pH of aqueous phase has to be below pKi), the general expression of the chemical reaction being as follows: R-CH(NH3+)-COOH(aq) + HP(o) R-CH(NH3+)-COOH.P-(o) + H+(aq) where HP is the carrier [4]. The maximum of mass flows is the result of two opposite phenomena: the increase of the concentration of extractant active form, which is able to react with the amino acid, and the Roum. Biotechnol. Lett., Vol. 11, No. 5, 2915-2921 (2006) 2917 ALEXANDRA CRISTINA BLAGA, ANCA-IRINA GALACTION, DAN CAŞCAVAL, ELENA FOLESCU decrease of the total amount of amino acid existing in cationic form. The supplementary increase of pH-value of feed phase to the isoelectric point determines the increase of zwitterions concentration, that significantly reducing the initial mass flows of the amino acids (at the isoelectric point the reactive extraction of amino acids becomes impossible [4]). Due to its lower isoelectric point, this effect is more pronounced for L-cysteine (pKi = 5.1) comparatively with the other considered amino acids (at pH = 6 the pertraction efficiency for L-tryptophan, L-glycine, L-alanine is very low, but becomes 0 for L-cysteine). The highest values of initial mass flows were recorded for L-tryptophan, owing to its aromatic radical R which induces superior hydrophobicity. Similar to the acidic amino acids, the final mass flows of neutral amino acids initially increase with pH of feed solution, due to their accumulation in the liquid membrane. But, unlike the aspartic and glutamic acids [16], the final mass flows of all neutral amino acids reach a maximum value at pH = 4. The further increase of pH leads to the decrease of the final mass flows, owing to the change of the sense of pH-gradient which controls the direction of solute transfer through liquid membrane. The permeability factor strongly increases with the pH increase, becoming higher than 1 for pH 3-3.5. This variation indicates that the final mass flows become superior to the initial ones, phenomena that are possibly due to the re-extraction of the supplementary amount of amino acids accumulated into the organic layer. The increase of the pH-value of the stripping phase determines the reducing of both initial and final mass flows, the same evolution being registered for the permeability factor, as it can be seen from Figure 2. For all studied neutral amino acids, the maximum values of the permeability factors are over 0.9, being reached for the pH-value of stripping phase of 1 and pH for the feed phase of 3. L-Cysteine L-Tryptophan -2 0.8 0.8 0.6 0.6 1.0 -1 1.2 P -2 n, moles m h P n, moles m h 1.0 -1 1.0 1.0 0.8 0.8 0.6 0.6 0.4 0.4 0.4 0.4 ni nf P 0.2 0.2 0.0 0.2 2 3 4 0.2 0.0 0.0 1 ni nf P 0.0 1 5 2 3 4 5 pH of stripping phase pH of stripping phase L-Glycine L-Alanine 1.2 1.0 0.8 0.8 0.6 0.6 -2 n, moles m h P -2 n, moles m h -1 -1 1.0 1.0 P 1.0 0.8 0.8 0.6 0.6 0.4 0.4 0.4 0.4 ni nf P 0.2 0.0 1 2 3 4 5 pH of stripping phase 0.2 0.2 0.0 0.0 ni nf P 0.2 0.0 1 2 3 4 5 pH of stripping phase Figure 2. Variation of the amino acids mass flows and permeability factor in function of the pH-value of the stripping phase (pH of feed phase = 3, D2EHPA concentration = 40 g l-1, rotation speed = 500 rpm). 2918 Roum. Biotechnol. Lett., Vol. 11, No. 5, 2915-2921 (2006) Extraction and transport of neutral amino acids through liquid membranes The carrier concentration inside the liquid membrane is another important factor that controls the amino acids pertraction efficiency. From Figure 3 it can be observed that the initial and final mass flows of amino acids are continuously intensified with the increase of D2EHPA concentration to 60 g l-1, due to the increase of the concentration of one of the reactants and, consequently, to the accumulation of the interfacial compound into the organic layer. Over this level, the increase of mass flows becomes slower, this variation being more accentuated for the final mass flows. Contrary to the above mentioned variations, the permeability factors initially increase with D2EHPA concentration to a maximum value, followed by its decreasing. For all neutral amino acids, the maximum level of permeability factor corresponds to a carrier concentration of 60 g l-1. Therefore, similar to the acidic amino acids, the pertraction system reaches its maximum capacity of solute transfer at 60 g l-1 carrier concentration, for the given experimental conditions. L-Cysteine L-Tryptophan 2.0 -2 n, moles m h P 1.4 1.2 0.9 1.0 0.8 P 1.6 0.9 1.2 0.8 ni nf P 0.6 1.0 -1 1.0 -2 n, moles m h -1 1.6 ni nf P 0.8 0.4 0.7 20 40 60 80 0.8 0.4 100 20 40 -1 Carrier concentration, gl L-Glycine 60 80 100 Carrier concentration, g/l L-Alanine 1.6 1.0 1.0 -1 P -2 n, moles m h P 1.4 -2 n, moles m h -1 1.6 1.2 0.9 1.0 1.2 0.9 0.8 0.8 0.8 ni nf P 0.6 ni nf P 0.4 0.4 0.8 0.7 20 40 60 80 100 20 -1 Carrier concentration, gl 40 60 80 100 Carrier concentration, g/l Figure 3. Variation of the amino acids mass flows and permeability factor in function of the carrier concentration (pH of feed phase = 3, pH of stripping phase = 2, rotation speed = 500 rpm). The dependences of amino acids mass flows on rotation speed, plotted in Figure 4, suggest that the overall separation process could be controlled by the diffusional processes or interfacial chemical reactions. The mixing intensification of the two aqueous phases induces the enhancement both of the initial and final mass flows for all neutral amino acids, owing to the diminution of resistance to the diffusion through the interfacial boundary layers, evolution Roum. Biotechnol. Lett., Vol. 11, No. 5, 2915-2921 (2006) 2919 ALEXANDRA CRISTINA BLAGA, ANCA-IRINA GALACTION, DAN CAŞCAVAL, ELENA FOLESCU that is recorded also for the permeability factor. The recorded influence is more important for rotation speed values below 500 rpm, over this level the kinetic resistance becoming the limiting step. The increase of permeability factors with the rotation speed intensification indicates a stronger influence of mixing on final mass flows, due to the more accentuated resistance to the diffusion through the boundary layer on the stripping phase side. L-Cysteine L-Tryptophan 0.8 0.6 -1 1.0 P -2 P 1.0 n, moles m h 0.8 -2 n, moles m h -1 1.0 0.8 0.8 0.6 0.6 0.6 0.4 0.4 ni nf P 0.2 200 300 0.4 ni nf P 200 400 500 600 Rotation speed, rpm 300 400 500 600 Rotation speed, rpm L-Glycine L-Alanine -1 P -2 0.8 0.6 -1 1.0 P -2 0.8 1.0 n, moles m h 1.0 n, moles m h 0.4 0.2 0.8 0.8 0.6 0.6 0.6 0.4 0.4 ni nf P 0.2 200 300 0.4 400 500 600 Rotation speed, rpm ni nf P 0.4 0.2 200 300 400 500 600 Rotation speed, rpm Figure 4. Variation of the amino acids mass flows and permeability factor in function of the rotation speed (pH of feed phase = 3, pH of stripping phase = 2, D2EHPA concentration = 40 g l-1). Conclusions The studies on facilitated pertraction of some neutral amino acids (L-cysteine, Ltryptophan, L-glycine, L-alanine) through a liquid membrane of dichloromethane and D2EHPA as a carrier underlined the major influence of pH-gradient between the feed and striping phases, carrier concentration in organic layer and mixing intensity of aqueous phases. In the purpose to reach the maximum values of amino acids mass flows, the facilitated pertraction has to be carried out at the pH of feed phase of 3, pH of stripping phase of 1, 2920 Roum. Biotechnol. Lett., Vol. 11, No. 5, 2915-2921 (2006) Extraction and transport of neutral amino acids through liquid membranes D2EHPA concentrations in the liquid membrane of 60 g l-1, and the aqueous phases must be intensively mixed. By modifying the pH of the feed phase it is possible to separate selectively the studied amino acids. 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