1. RCM as a Tool to Freeze Conformation of Monosaccharides : Synthesis of a β-Mannopyranoside
Mimic Adopting a Conformation Close to the Biologically Relevant B2,5 Boat
L. Amorim, D. Díaz, J.Jiménez-Barbero, P. Sinaÿ, Y. Blériot
Tetrahedron Letters 2006, 47, 8887-8891
2. Synthesis of a Close Mimic of L-Iduronic Acid Adopting the Biologically Active 2S0 Conformation
A.Herrera, M.Beneitez, L. Amorim, J Esnault, J Cañada, J Jimenez-Barbero, J.M. Mallet, P. Sinaÿ, Y.
Blériot
2006, submitted
3. 2-C-Hydroxymethyl-2,3-O-isopropylidene-D-ribono-1,5-lactam
C.R. Newton, M. Iezzi Simone, G. W. J. Fleet, Y. Blériot, D. J. Watkin
Acta. Cryst. 2004, E60, o909-o910
4. (2S, 3R, 4R, 5S)-3,4-O-isopropylidene-2-methyl-6,9-diazo-1-oxaspiro[4.5]-decane-7,10-dione
D.J. Watkin, M. Müller, Y. Blériot, M.I. Simone, G.W.J. Fleet,
Acta Cryst. 2004, E60, o1820-o1822.
5. Sugar amino acids at the anomeric position of carbohydrates: synthesis of spirocyclic amino acids of 6deoxy-L-lyxofuranose
Y. Blériot, M. I. Simone, M. R. Wormald, R.A. Dwek, D. J. Watkin and G. W. J. Fleet..
Tetrahedron: Asymmetry 2006, 17, 2276-2286
6. Looking glass inhibitors: efficient synthesis and biological evaluation of D-deoxyfuconojirimycin
Y. Blériot, D. Gretzke, T. M. Krulle, T. D. Butters, R. A. Dwek, R. J. Nash, N. Asano and G. W. J. Fleet
Carbohydrate Research 2005, 340, 2713–2718
7. Synthesis and conformational analysis of novel N(OCH3)-disaccharide analogues
F. Peri, J. Jiménez-Barbero,V. García-Aparicio, I. Tvaroška, F. Nicotra
Chem. Eur. J. 2004, 10, 1433-1444
8. Mimics of ganglioside GM1 as Cholera Toxin ligands: The importance of carbohydrate-aromatic
interactions in molecular recognition processes.
A. Bernardi, D. Arosio, D. Potenza, I. Sanchez-Medina, S. Mari, F. J. Cañada, J. Jimenez-Barbero
Chem. Eur. J. 2004, 10, 4395-4405
9. Mimics of ganglioside GM1 as Cholera Toxin ligands: replacement of the GalNAc residue.
D. Arosio, A. Bernardi, L. Manzoni, D. Monti, H. Posteri, D. Potenza, S. Mari, J. Jimenez-Barbero
Org. Biomol. Chem. 2003, 1, 785-792
10. GM1 glycomimetics and bacterial endotoxins
A. Bernardi, C. Podlipnik, J. Jiménez-Barbero,
In Carbohydrates and Infectious Diseases, C. Bewley (Ed) 2006, RSC
11. Synthesis and conformational analysis of galactose-derived simple bicyclic scaffolds.
I. Velter, F. Nicotra, B. Laferla, A. Bernardi, G. Marcou, I. Motto, S. Mari, F. J. Cañada, J. JimenezBarbero
Eur. J. Org. Chem 2006, 2925-2933
12. Natural and Synthetic Cholera Toxin Antagonists
Velter A.I., Politi, M., Podlipnik C., Nicotra, F.
Minirev. Med. Chem, 2006, in press
13. First round of focused library for cholera toxin inhibitor search
C. Podlipnik, I. Velter, G. Marcou, B. La Ferla, L. Belvisi, A. Bernardi, F. Nicotra
2006, submitted
14. A simple model system for the study of carbohydrate-aromatic interactions.
G. Terraneo, D. Potenza, A. Canales, J. Jiménez-Barbero, K. Baldridge, A. Bernardi
2006, submitted
15. The first synthesis of substituted azepanes mimicking monosaccharides: a new class of potent
glycosidase inhibitors
H. Li, Y. Blériot, C. Chantereau, J.-M. Mallet, M. Sollogoub, Y. Zhang, E. Rodríguez-García, P. Vogel, J.
Jiménez-Barbero, P. Sinaÿ
Org. Biomol Chem. 2004, 2, 1492-1499.
16. The conformational behavior of novel glycosidase inhibitors with substituted azepan structures. A
NMR and modeling study
Martínez, J. L. Medina, S. Mari, F. Cañada, P. Vogel, H. Li, Y. Bleriot, P. Sinäy, J. Jiménez-Barbero
Eur. J. Org. Chem. 2004, 20, 4119-4129
17. PolyAzepanes mimicking monosaccharides: synthesis of an D-galacto-like iminoheptitol
H. Li, Y. Blériot, J-M. Mallet, Y. Zhang, E. R.-Garcia, P. Vogel, S. Mari, J. Jiménez-Barbero, P.
Sinaÿ
Heterocycles, 2004, 64, 65-74
18. Synthesis, Conformational Studies and Mannosidase stability of a Mimic of 1,2-Mannobioside.
S. Mari, H. Posteri, G. Marcou, D. Potenza, F. Micheli, F. J. Cañada, J. Jimenez-Barbero, A. Bernardi
Eur. J. Org. Chem. 2004, 5119-5125
19.
Synthesis and Conformational analysis of α-Man-(1→2)-α-Man-(1→6)-α-Man mimic.
S. Mari, I. Sánchez-Medina, P. Mereghetti, L. Belvisi, J. Jimenez-Barbero, A. Bernardi
2006, submitted
20. Design, Synthesis, and Biological Evaluation of Sugar-Derived Ras Inhibitors.
Peri, F., Airoldi, C., Colombo, S., Martegani, E., Stein, M., van Neuren, A.S., and Nicotra, F
ChemBioChem 2005, 6, 1839 – 1848 .
21. Sugar-derived Ras-inhibitors: group epitope mapping by NMR spectroscopy and biological
evaluation
F. Peri,. C. Airoldi,. S. Colombo,. S. Mari,.J. Jiménez-Barbero,.E. Martegani,.F. Nicotra..
Eur. J. Org. Chem., 2006, 3707-3720