Research Tracers A clear path for the future EXPAND ACCELERATE INNOVATE www.ibamolecular.com Molecular Imaging: A Clear Path The future of molecular imaging is on the minds of many in the imaging community. Today’s research is crucial to the future of molecular imaging, diagnostics and therapeutics. In this exciting time of exploring new frontiers, the deployment of more targeted and impactful compounds is key to winning the fight against disease. IBA Molecular has made a strong commitment to supporting the research and development of these new products. With many years of collective experience in producing F-18-labelled and other radiopharmaceutical compounds, we are continuing to expand our research tracer offerings to support programs at leading institutions. Creating a clear path for research and development is crucial and the choices made today can lead to an active commitment to the future of molecular imaging. IBA Molecular is uniquely positioned to: EXPAND Maximize worldwide access to a wide range of novel radioisotopes and compounds ACCELERATE Utilize our expertise, innovation and experience to focus and accelerate research efforts INNOVATE Align with key biopharma entities to develop new compounds and access to clinical trials The Next Generation of Molecular Imaging Ga-68 DOTATOC CASE STUDY Whole body “one-stop shop” diagnosis with receptor-PET/CT (A - MIP; B, C and D - PET, CT and fused images) using Ga-68 DOTATOC showing primary neuroendocrine tumor in the ileum (B) with lymph node (C) & bone metastases (D). Study and images source: Theranostics 2012; 2(5):437-447. doi:10.7150/thno.3645 IBA Molecular is providing the next generation of molecular imaging products and services to research programs worldwide. We provide radiolabeling and development services, as well as manufacturing of clinical trial and commercial doses for promising diagnostic and therapeutic isotopes. By aligning with academic institutions, biotechnology and pharmaceutical companies, we will work with our partners to validate the ongoing unmet medical needs as well as the potential impact of these products on disease management. Our objective is to facilitate research, development and commercialization of the next generation of molecular imaging and therapeutic products, which is expected to provide targeted improvements in patient care and outcomes 181,000 The number of registered studies has grown 1500% in 10 yrs* $100 B Capital investment spent on research in the last 10 yrs* 1 Goal. To deliver the next generation of targeted agents Research Tracers Ga-68 DOTATOC/TATE (DOTATOC Under DMF) Radiolabeled somatostatin analogs being investigated for the diagnosis and treatment of neuroendocrine tumors (NETs). Ga-68 Chloride and Citrate For use in labeling peptides and antibodies such as PSMA. F-18 Bulk For use in synthesis of multiple F-18 based tracers. F-18 FLT Fluorothymidine Thymidine analog which targets cell proliferation, currently being studied for response to therapy in lymphoma, breast, head and neck, brain, cervical, pancreatic, esophageal, kidney, lung, colorectal and neuroendocrine cancers. F-18 FLT IN RESPONSE TO THERAPY Highest purity I-124 (sole DMF in U.S.) Being used in a variety of PET applications, including protein and antibody iodinations, and in the design of new PET tracers. Also being used to develop novel therapies using large biomolecules and nanoparticles. Zr-89 Zirconium Zr-89 Zirconium is used in PET imaging with radiolabeled monoclonal antibodies. Zr-89-based PET imaging has been investigated for a wide variety of cancer-related targets. Ac-225 Actimab-A** Monoclonal antibody-directed alpha emitter drug candidate under development for the front line treatment of newly diagnosed elderly acute myeloid leukemia patients. I-131- Iomab-B** Monoclonal antibody under development that targets CD45, an antigen associated with acute myeloid leukemia. Also shows utility in other indications, including myelodysplasia syndrome, acute lymphoblastic leukemia, Hodgkin’s disease and Non-Hodgkin Lymphoma. Zr-89 PSMA** An immunoPET tracer for imaging prostate cancer, IAB2m is a monoclonal antibody fragment targeting prostate-specific membrane antigen (PSMA). Breast FLT PET-CT SUVmax reduction >39% pretreatment (lower row) compared with 10 days after start of the first cycle of chemotherapy (upper row). Drawn circles indicate lesion position on respective PET slices containing SUVmax. FLT = 3-Deoxy-318F-fluorothymidine, PET = positron emission tomography, CT = computed tomography, SUV = standardized uptake value, max = maximum Study and images source: Indian J Nucl Med. 2014 Apr-Jun; 29(2): 65–73. F-18 Tau** Imaging agent under development to identify tau neurofibrillary tangles in the characterization of cognitive impairment, including Alzheimer’s disease. * Source: http://clinicaltrials.gov ** Proprietary compound Clinical Trial Use - Clinical trial use of certain products should include the appropriate filing of an investigator-sponsored Investigational New Drug (IND) application to the FDA. Where applicable, IBA Molecular may supply a Letter of Authorization to permit cross-reference to its Drug Master File for the specific product. Access to Clinical Trials IBA Molecular has partnered with key biopharma companies to develop new compounds for clinical trials. Your qualification and selection in clinical trials may optimize the use of your imaging equipment and staff expertise as well as potentially being included in published outcomes. IBA Molecular IBA Molecular is a global developer, manufacturer and distributor of radiopharmaceutical products and supporting services used in molecular imaging. We have engineered a strong and unique product portfolio of diagnostic and therapeutic tracers. We also provide educational content, technical, research and marketing support to medical specialists worldwide to help better respond to patient needs. Contact Us IBA Molecular North America, Inc. 21000 Atlantic Blvd., Suite 730 Dulles, VA 20166 Toll Free: 1 877 334 3673 Tel.: + 1 703 787 7900 Fax.: + 1 571 434 0330 IBA Molecular North America | January 2015 | Research Tracers © IBA 2015/All Rights Reserved. For additional information regarding technical specifications, availability, pricing and ordering of these and other products please contact us at marketingus@ibamolecular.com www.ibamolecular.com