List of Scientific Articals of Allaсhem's Scientists
1.
Morozova M.A., Lepikina T. A., Rupchev G. E., Beniashvily A. G., Burminskiy D. S., Potanin S. S.,
Bondsrenko E. V., Kazey V. I., Lavrovsky Y., Ivachtchenko A.V. Add-on clinical effects of selective antagonist of 5HT6 receptors AVN-211 (CD-008-0173) in patients with schizophrenia stabilized on antipsychotic treatment: pilot study . CNS Spectrums , FirstView Article, 1-
8 (3013). http://journals.cambridge.org/abstract_S1092852913000394.
2.
Ivachtchenko, A. V.; Golovina, E. S.; Kadieva, M. G.; Mitkin, O. D.; Tkachenke S.E.; Okun, I.M.
Synthesis of Substituted Diphenyl Sulfones and Their Structure-Activity Relationship with the
Antagonism of 5-НТ6 Receptors.
Bioorg. Med. Chem.
, 21б 4614-4627 (2013).
3.
Ivachtchenko, A. V.; Golovina, E. S.; Kadieva, M. G.; Kysil, V. M.; Mitkin, O. D.; Vorobiov, A. A.;
Okun, I. M. Antagonists of 5-HT6 receptors. Substituted 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[3,4-
1
e]pyrimidines and 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[4,3-d]pyrimidines — synthesis and
«structure – activity» relationship.
Bioorg. Med. Chem. Lett.
, 22 , 4273-4280 (2012).
4.
Ivachtchenko, A. V.; Golovina, E. S.; Kadieva, M. G.; Kysil, V. M.; Mitkin, O. D.; Tkachenko, S. E.;
Okun, I. M. Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists . Bioorg. Med. Chem . 19, 1482–1491(2011).
5.
Ivachtchenko, A. V.; Golovina, E. S.; Kadieva, M. G.; Koryakova, A. G.; Mitkin, O. D.; Tkachenko, S.
E.; Kysil, V. M.; Okun, I. M. 2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines:
New series of highly potent and specific serotonin 5-HT6 receptor antagonists . Eur. J. Med. Chem ., 46
1189-1197(2011).
6.
Ivachtchenko, A. V.; Golovina, E. S.; Kadieva, M. G.; Kysil, V. M.; Mitkin, O. D.; Tkachenko, S. E.;
Okun, I. M. Synthesis and Structure Activity Relationship (SAR) of (5,7-disubstituted 3phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT
6
Receptor (5-
HT
6
R) Antagonists. J. Med. Chem ., 54, 8161-8173 (2011).
7.
Ivachtchenko, A. V.; Frolov, E. B.; Mitkin, O. D.; Tkachenko, S. E.; Okun, I. M.; Khvat, A. V. Synthesis and biological activity of 5-styryl and 5-phenethyl-substituted 2,3,4,5-tetrahydro-1H-pyrido[4,3b]indoles.
Bioorg. Med. Chem. Lett ., 20 (1), 78–82 (2010).
8.
Ivachtchenko, A. V.; Dmitriev, D. E.; Golovina, E. S.; Dubrovskaya, E. S.; Kadieva, M. G.; Koryakova,
A. G.; Kysil, V. M.; Mitkin, O. D.; Tkachenko, S. E.; Okun, I. M.; Vorobiov, A. A. Synthesis of cycloalkane-annelated 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines and their evaluation as 5-HT6
receptor antagonists. Bioorg. Med. Chem. Lett. , 20 (7), 2133–2136 (2010).
9.
Tsirulnikov, S.; Kysil, V.; Ivachtchenko, A.; Krasavin, M. Trimethylsilyl Chloride as a Promoter for the Groebke-Blackburn Reaction: Preparation of Imidazo[2,1-b][1,3]Benzothiazoles .
Synth. Comm .,
40(1), 111–119 (2010).
10.
Ivachtchenko, A. V.; Mitkin, O. D.; Tkachenko, S. E.; Okun, I. M.; Kysil, V. M. 8-Sulfonyl-substituted tetrahydro-1H-pyrido[4,3-b]indoles as 5-HT6 receptor antagonists.
Eur. J. Med. Chem ., 45(2), 782–789
(2010).
11.
Ivachtchenko, A. V.; Golovina, E. S.; Kadieva, M. G.; Koryakova, A. G.; Kovalenko, S. M.; Mitkin, O.
D.; Okun, I. M.; Ravnyeyko, I. M.; Tkachenko S. E.; Zaremba, O. V. Synthesis and biological study of 3-
(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines as potent and selective serotonin 5-HT6 receptor antagonists.
Bioorg. Med. Chem., 18 , 5282–5290 (2010).
12.
Ivachtchenko, A. V.; Golovina, E. S.; Kadieva, M. G.; Koryakova, A. G.; Kysil, V. M.; Mitkin, O. D.;
Okun, Ravnyeyko, I. M.; I. M.; Tkachenko, S. E.; Zaremba O. V . Solution Phase Parallel Synthesis of
Substituted 3-Phenylsulfonyl-[1,2,3]triazolo[1,5-a]quinazolines: Selective Serotonin 5-HT(6) Receptor
Antagonists.
J. Comb. Chem.
, 12 , 445–452 (2010).
13.
Ivachtchenko, A. V.; Dmitriev, D. E.; Golovina, E. S.; Kadieva, M. G.; Koryakova, A. G.; Kysil, V. M.;
Mitkin, O. D.; Okun, I. M.; Tkachenko, S. E.; Vorobiov, A. A. (3-Phenylsulfonylcycloalkano[e and

d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT(6)
Receptor. J. Med. Chem,. 53 , 5186–5196 (2010).
14.
A.V. Ivachtchenko, E.B. Frolov, O.D. Mitkin, S.E. Tkachenko, A.V. Khvat.
Synthesis of hydrogenated
2,7-dimethylpyrrolo[3,4-b]indoles – analogs of Dimebon. Heterocyclic Comp., 46 (2), 170-178 (2010).
15.
A.V. Ivaschenko, E.B. Frolov, O.D. Mitkin, S.E. Tkachenko, A.V. Khvat. Synthesis and Biological
Evaluation of Novel Bioisosteric Analogues of Dimebon
TM
. Letters in Drug Design & Discovery , 7(6), 446-
2
451 (2010).
16.
Ivachtchenko A.V., Yamanushkin P.M., Mitkin O.D., Kiselev O.I. Bromination of indomethacin .
Mendeleev Comm ., 20, 111-112 (2010).
17.
Ivachtchenko, A.; Kysil, V.; Mitkin, O.; Kadieva, M.; Tkachenko, S.; Khvat, A.; Okun, I.;
Lavrovsky Y. Pre-clinical and Erly Clinical Studies of AVN-322, a novel 5-HT6 Receptor Small
Molecule Antagonist for the Treatment of Alzheimer’s Disease.
Alzheimer’s Disease Keystone Symposia
Meeting.
January 10 – 15, USA, PA221, 81 (2010).
18.
Lavrovsky,Y.; Ivachtchenko, A.; Morozova, M.; Salimov, R. M.; Kazey, V. Preclinical and early clinical stadies of AVN-101, a novel balanced molecule for the treatment of Alzheimers's disease.
Alzheimer's Dementia, 6(4), Suppl 1, S583 (2010), Alzheimers's Association International Conference on
Alzheimers's Disease, July 10–15, 2010, Honolulu, Hawaii, USA, P3-442 (2010).
19.
Potapov, V. V.; Fetisova, N. A.; Nikitin, A. V.; Ivachtchenko, A. V. One-step assembly of novel carbamoyl substituted 6-oxo-4,5,6,11-tetrahydropyrrolo[1,2-b][2,5]benzodiazo-cine . Tetrah. Lett.
,
50(23), 2790–2792 (2009).
20.
Kysil, V.; Khvat, A.; Tsirulnikov, S.; Tkachenko, S.; Ivachtchenko, A. Multicomponent approach to unique 1,4-diazepine-2-amines.
Tetrah. Lett.
, 50(24), 2854–2856 (2009).
21.
Tsirulnikov, S.; Nikulnikov, M.; Kysil, V.; Ivachtchenko, A.; Krasavin, M. Streamlined access to 2,3dihydropyrazino[1,2-a]indole-1,4-diones via Ugi reaction followed by microwave-assisted cyclization.
Tetrah. Lett.
, 50(39), 5529–5531 (2009).
22.
Ivachtchenko, A. V.; Frolov, E. B.; Mitkin, O. D.; Kysil, V. M.; Khvat, A. V.; Tkachenko, S. E.
Synthesis and Biological Evaluation of Novel 5,8-Disubstituted-2-methyl-2,3,4,5-tetrahydro-1Hpyrido[4,3-b]indoles as 5-HT6 and H1 Receptors Antagonists . Arch. Pharm.
, 342(12), 740–747 (2009).
23.
Alyab'ev, S. B.; Kravchenko, D. V.; Ivashchenko, A. V. Synthesis and functionalization of the 3-
(1,3,4-oxadiazol-2-yl)-1h-indoles.
Chem. Heterocycl. Comp ., 45(10), 1270–1275 (2009).
24.
Potapov, V. V.; Fetisova, N. A.; Nikitin, A. V.; Ivachtchenko, A. V. A convenient synthesis of heterocyclic compounds containing 11-oxo-6,11,12,13-tetrahydrodiben-zo[b,g][1,5]oxazonine fragment . Mend. Commun ., 19(5), 287–289 (2009).
25.
Lakner, F. J.; Parker, M. A.; Rogovoy, B.; Khvat, A.; Ivachtchenko, A. Synthesis of novel trisubstituted imidazolines . Synthesis , 1987–1990 (2009).
26.
Ivachtchenko, A. V.; Frolov, E. B.; Mitkin, O. D.; Kysil, V. M.; Khvat, A. V.; Okun, I. M.; Tkachenko,
S. E.
Synthesis and biological evaluation of novel γ-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists . Bioorg. Med. Chem. Lett.
, 19(12), 3183–3187 (2009).
27.
Nikulnikov, M.; Tsirulnikov, S.; Kysil, V.; Ivachtchenko, A.; Krasavin, M. tert-Butyl isocyanide as a convertible reagent in Ugi reaction: microwave-assisted preparation of 5,6-dihydropyrazolo[1,5a]pyrazine-4,7-diones.
Synlett , 260–262 (2009).
28.
Ryzhova, E. A.; Koryakova, A. G.; Bulanova, E. A.; Mikitas, O. V.; Karapetyan, R. N.; Lavrovskii, Ya.
V.; Ivashchenko, A. V. Synthesis, molecular docking, and biological testing of new selective inhibitors of glycogen synthase kinase 3β . Pharm. Chem. J ., 43(3), 148–153 (2009).
29.
Alyabiev, S. B.; Kravchenko, D. V.; Ivachtchenko, A. V. Regioselective synthesis of substituted isoxazolo[5,4-d]pyrimidines.
Mend. Commun ., 18 (3), 144–146 (2008).
30.
Alyabiev, S. B.; Kravchenko, D. V.; Ivachtchenko, A. V. Synthesis of ethyl 4-oxo-3,4dihydro[1]benzofuro[3,2-d]pyrimidine-2-carboxylate and its derivatives.
Mend. Commun ., 18 (4), 217–
219. (2008).

3
31.
Sapegin, A. V.; Sakharov, V. N.; Kalandadze, L. S.; Smirnov, A. V.; Khristolyubova, T. A.; Plakhtinskii,
V. V.; Ivashchenko, A. V. Synthesis of dibenzo[b,f][1,4]oxazepin-11(10H)-one and pyrido[2,3b][1,4]benzoxazepin-10(11H)-one compounds based on o-nitrochloro derivatives of benzene and pyridine . Mend. Commun.
, 18(5), 281–283 (2008).
32.
Sandulenko, Yu. B.; Ivashchenko, A. V.; Kravchenko, D. V.; Tkachenko, S. E.; Vvedensky, V. Yu.
Parallel solid-phase synthesis of novel 3,7-diazabicyclo[3.3.1]nonane derivatives starting from natural alkaloid cytisine.
Russ. Chem. Bull ., 57 (9), 1999–2004 (2008).
33.
Krasavin, M.; Tsirulnikov, S.; Nikulnikov, M.; Kysil, V.; Ivachtchenko, A. Poorly reactive 5-piperazin-
1-yl-1,3,4-thiadiazol-2-amines rendered as valid substrates for Groebke-Blackburn type multicomponent reaction with aldehydes and isocyanides using TMSCl as a promoter.
Tetrah. Lett.
,
49 (36), 5241–5243(2008).
34.
Koryakova, A. G.; Ivanenkov, Y. A.; Ryzhova, E. A.; Bulanova, E. A.; Karapetian, R. N.; Mikitas, O. V.;
Katrukha, E. A.; Kazey, V. I.; Okun, I. М.; Kravchenko, D. V.; Lavrovsky, Y. V.; Korzinov, O. M.;
Ivachtchenko, A. V. Novel aryl and heteroaryl substituted N-[3-(4-phenylpiperazin-1-yl)propyl]-1,2,4oxadiazole-5-carboxamides as selective GSK-3 inhibitors.
Bioorg. Med. Chem. Lett.
, 18 (12), 3661–3666
(2008).
35.
Ivachtchenko, A. V.; Tkachenko, S. E.; Okun, I. M.; Savchuk, N. F.; Miroshnichenko, I. I.; Lelishentsev,
A. A.; Kalmykov, Yu. M.; Fedotov, Yu. A.; Ivashchenko, A. A. Determining amlodipine in blood plasma by liquid chromatography coupled to tandem mass spectrometry.
Pharm. Chem. J ., 42 (8), 493–495
(2008).
36.
Aliabiev, S. B.; Ivanov, I. S.; Ilyin, A. P.; Kravchenko, D. V.; Ivachtchenko, A. V. Synthesis of novel
5,6,7-substituted 3-phenyl-6,7-dihydroisoxazolo[4,5-d]pyrimidines Lett. Org. Chem ., 4 (3), 203–211
(2007).
37.
Smirnov, A. V.; Kalandadze, L. S.; Sakharov, V. N.; Dorogov, M. V.; Ivachtchenko, A. V.
Denitrocyclization in synthesis of dibenzo[b,f][1,4]thiazepin-11(10H)-ones and their derivatives.
J. Heterocycl. Chem.
, 44(6), 1247–1251 (2007).
38.
Aliabiev, S. B.; Bykova, R. V.; Kravchenko, D. V.; Ivachtchenko, A. V. A convenient of novel substituted isoxazolo[5,4-d]pyrimidines.
Lett. Org. Chem ., 4(4), synthesis
273–280 (2007).
39.
Kysil, V.; Tkachenko, S.; Khvat, A.; Williams, C.; Tsirulnikov, S.; Churakova, M.; Ivachtchenko, A.
TMSCl-promoted isocyanide-based MCR of ethylenediamines: An efficient assembling of 2aminopyrazine core . Tetrah. Lett ., 48(36), 6239–6244 (2007).
40.
Ivanovsky, S. A.; Dorogov, M. V.; Kravchenko, D. V.; Ivachtchenko, A. V. Synthesis of the
Substituted 3-Cyclobutene-1,2-diones.
Synth. Commun ., 37 (15), 2527–2542 (2007).
41.
Savchenko, T. I.; Silin, O. V.; Kovalenko, S. M.; Musatov, V. I.; Nikitchenko, V. M.; Ivachtchenko, A.
V. Alkylation of 3-phenyl-1H-pyrazolo[4,3-c] quinoline: theoretical analysis of regioselectivity.
Synth. Commun ., 37 (8), 1321–1330 (2007).
42.
Trifilenkov, A. S.; Ilyin, A. P.; Kysil, V. M.; Sandulenko, Y. B.; Ivachtchenko, A. V. One- pot tandem complexity-generating reaction based on Ugi four component condensation and intramolecular cyclization.
Tetrah. Lett ., 48 (14), 2563–2567 (2007).
43.
Kiselyov, A.; Balakin, K. V.; Tkachenko, S. E.; Savchuk, N.; Ivachtchenko, A. V. Recent progress in discovery and development of antimitotic agents.
Anti-Cancer Agents Medicin. Chem.
, 7 (2), 189–208
(2007).
44.
Ilyin, A. P.; Dmitrieva, I. G.; Kustova, V. A.; Manaev, A. V.; Ivachtchenko, A. V. Synthesis of
Heterocyclic Compounds Possessing the 4H-Thieno[3,2-b]Pyrrole Moiety.
J. Combin. Chem., 9 (1),
96–106 (2007).
45.
Яманушкин, П. М.; Митькин, О. Д.; Кравченко, Д. В.; Введенский, В. И.; Иващенко, А.В.
Новый метод синтеза циклических гуанидинов
. XVIII Менделеевский съезд по общей и прикладной химии , 23 – 28 сентября, Москва, Т. 1, 525 (2007).
46.
Lakner, F. J.; Parker, M. A.; Rogovoy, B.; Khvat, A.; Ivachtchenko, A.
Synthesis of Novel

Trisubstituted Imidazolines. 41 st Western Regional Meeting of the American Chemical Society ,
October 9–13, San Diego, CA, (2007).
47.
Khvat, A.; Kysil, V.; Ilyin, A.; Rogovoy, В.; Lakner, F.; Hammaker, J.; Ivachtchenko, A. Targeting
Diversity: One-Pot Syntheses of Compounds for Target-Biased Screening Libraries.
41 s t Western
Regional Meeting of the American Chemical Society , October 9– 13, San Diego, CA, (2007).
48.
Dorogov, M. V.; Ivanovsky, S. A.; Khakhina, M. Y.; Kravchenko, D. V.; Tkachenko, S. E.;
4
Ivachtchenko, A. V. Synthesis of 7-sulfamoyl-substituted 2-oxo-2,3,4,5-tetrahydro-1Hbenzo[b]azepines . Synth. Commun.
, 36(23), 3525–3535 (2006).
49.
Ilyin, A. P.; Loseva, M. V.; Vvedensky, V. Y.; Putsykina, E. B.; Tkachenko, S. E.; Kravchenko, D.
V.; Khvat, A. V.; Krasavin, M. Y.; Ivachtchenko, A. V. One-Step Assembly of Carbamoyl-Substituted
Heteroannelated [1,4]Thiazepines.
J. Org. Chem ., 71 (7), 2811–2819 (2006).
50.
Ilyin, A.; Kysil, V.; Krasavin, M.; Kurashvili, I.; Ivachtchenko, A. V. Complexity- Enhancing Acid-
Promoted Rearrangement of Tricyclic Products of Tandem Ugi
Alder Reaction . J. Org. Chem., 71(25), 9544–9547(2006).
4CC/Intramolecular Diels-
51.
Shevyakov, S. V.; Davydova, O. I.; Pershin, D. G.; Krasavin, M.; Kravchenko, D. V.; Kiselyov,
A.; Tkachenko, S. E.; Ivachtchenko, A. V. Natural products as templates for bioactive compound libraries: synthesis of biaryl derivatives of (±)vasicine .
Nat. Prod. Res.
, 20 (8), 735–741 (2006).
52.
Shevyakov, S. V.; Davydova, O. I.; Kiselyov, A. S.; Kravchenko, D. V.; Ivachtchenko, A. V.;
Krasavin, M. Natural products as templates for bioactive compound libraries: part 2. Novel modifications of vasicine (peganine) core via efficient and regioselective generation of 3lithiodeoxyvasicine and its stereoselective addition to aliphatic ketones.
Nat. Prod. Res.
, 20 (9), 871–881
(2006).
53.
Okun, I.; Malarchuk, S.; Dubrovskaya, E.; Khvat, A.; Tkachenko, S.; Kysil, V.; Ilyin, A.;
Kravchenko, D.; Prossnitz, E. R.; Sklar, L.; Ivachtchenko, A. Screening for caspase-3 inhibitors: a new class of potent small-molecule inhibitors of caspase-3.
J. Biomol. Scr.
, 11 (3), 277–285 (2006).
54.
Okun, I.; Malarchuk, S.; Dubrovskaya, E.; Khvat, A.; Tkachenko, S.; Kysil, V.; Kravchenko, D.;
Ivachtchenko, A. Screening for caspase-3 inhibitors: effect of a chemotypes.
J. Biomol. Scr.
, 11 (6), 694–703 (2006). reducing agent on identified hit
55.
Ilyin, A.; Kobak, V.; Dmitrieva, I.; Peregudova, Y.; Kustova, V.; Mishunina, Y.; Tkachenko, S.;
Ivachtchenko, A. Synthesis of 7,8-dihydrothieno[3',2':4,5]pyrrolo[1,2- a]pyrazin-5(6H)-ones using a modification of four-component Ugi reaction.
Synth. Commun.
, 36 (7), 903–910 (2006).
56.
Kravchenko, D.; Kysil, V.; Ilyn, A.; Tkachenko, S.; Maliarchouk, S.; Okun, I.; Ivachtchenko, A.
Synthesis and chemical transformations of 6-(morpholine-4- sulfonyl)quinoline-2,3,4-tricarboxylic acid.
Synth. Commun., 36 (7), 911–917 (2006).
57.
Kravchenko, D. V.; Kysil, V. M.; Tkachenko, S. E.; Maliarchouk, S.; Okun, I. M.; Ivachtchenko, A.
V. New variant of the Pfizinger reaction. Synthesis and chemical transformations of substituted
2-aminomethyl-quinoline-3,4-dicarboxylic acids.
Heterocycl. Comm ., 12 (1), 15–18 (2006).
58.
Ilyn, A. P.; Trifilenkov, A. S.; Kovrigin, D. I.; Yudin, M. V.; Ivachtchenko, A. V. New fourcomponent Ugi-type reaction. Synthesis of 3-methyl-1-oxo-1,3,4,6,11,11a- hexahydro-2Hpyrazino[1,2-b]isoquinoline-3-carboxamides.
Heterocycl. Comm ., 12 (2), 107–110 (2006).
59.
Trifilenkov, A. S.; Kobak, V. V.; Salina, M. A.; Kusovkova, J. A.; Ilyin, A. P.; Khvat, A. V.;
Tkachenko, S. E.; Ivachtchenko, A. V. Liquid-Phase Parallel Synthesis of
Combinatorial Libraries of Substituted 6-Carbamoyl-3,4-dihydro-2H-
benzo[1,4]thiazines.
J. Combin. Chem ., 8 (4), 469–479 (2006).
60.
Filimonov, S. I.; Korsakov, M. K.; Kravchenko, D. V.; Dorogov, M. V.; Tkachenko, S. E.;
Ivachtchenko, A. V. Convenient synthesis of novel 5-substituted 3-methylisoxazole-4sulfonamides.
J. Heterocycl. Chem ., 43 (3), 663–671 (2006).
61.
Ilyin, A. P.; Parchinski, V. Z.; Peregudova, J. N.; Trifilenkov, A. S.; Poutsykina, E. B.; Tkachenko,
S. E.; Kravchenko, D. V.; Ivachtchenko, A. V. One-step assembly of carbamoyl substituted

5 annulated 1,4-oxazepines.
Tetrah. Lett ., 47 (15), 2649–2653 (2006).
62.
Kravchenko, D. V.; Kuzovkova, J. A.; Kysil, V. M.; Tkachenko, S. E.; Malarchuk, S.; Okun, I.
M.; Ivachtchenko, A. V. Pyrrolo[3,4-c]quinoline-1,3-diones as potent caspase-3 inhibitors: synthesis and SAR of 8-sulfamoyl-1,3-dioxo-2,3-dihydro-1H-pyrrolo[3,4- c]quinolines.
Lett. Drug
Des. Discov.
, 3 (1), 61–70 (2006).
63.
Kravchenko, D. V.; Ivanenkov, Ya. A.; Balakin, K. V.; Kisil, V. M.; Tkachenko, S. E.; Okun, I.
M.; Ivashchenko, A. V. Design and synthesis of new nonpeptide caspase-3 inhibitors.
Pharm. Chem.
J ., 40 (3), 127–131(2006).
64.
Ivachtchenko, A. V.; Kobak, V. V.; Ilyn, A. P.; Khvat, A. V.; Kysil, V. M.; Williams, C. T.;
Kuzovkova, J. A.; Kravchenko, D. V. Parallel Liquid-Phase Synthesis of N-Substituted 6-
Aminosulfonyl-2-oxo-1,2-dihydroquinoline-4-carboxamide and 6-Aminosulfonyl-quinoline-4-
carboxamide Derivatives. J. Combin. Chem. , 7 (2), 227–235 (2005).
65.
Dalinger, I. L.; Vatsadse, I. A.; Shevelev, S. A.; Ivachtchenko, A. V. Liquid-phase synthesis of
combinatorial libraries based on 7-trifluoromethyl-substituted pyrazolo[1,5-a]pyrimidine scaffold. J.
Combin. Chem ., 7 (2), 236–245 (2005).
66.
Ilyin, A. P.; Trifilenkov, A. S.; Kurashvili, I. D.; Krasavin, M.; Ivachtchenko, A. V. One- Step construction of peptidomimetic 5-carbamoyl-4-sulfonyl-2-piperazinones.
J. Combin. Chem ., 7 (3),
360–363 (2005).
67.
Ilyn, A. P.; Trifilenkov, A. S.; Tsirulnikov, S. A.; Kurashvily, I. D.; Ivachtchenko, A. V. Synthesis of 4-Oxo-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-6-carboxamides Using a Modification of Ugi
Condensation.
J. Combin. Chem.
, 7 (6), 806–808 (2005).
68.
Ilyn, A. P.; Kuzovkova, A. A.; Potapov, V. V.; Shkirando, A. M.; Kovrigin, D. I.; Tkachenko, S. E.;
Ivachtchenko, A. V. An efficient synthesis of novel heterocycle-fused derivatives of 1-oxo-1,2,3,4tetrahydropyrazine using Ugi condensation.
Tetrah. Lett.
, 46 (5), 881–884 (2005).
69.
Vvedensky, V. Y.; Ivanov, Yu. V.; Kysil, V.; Williams, C.; Tkachenko, S.; Kiselyov, A.; Khvat, Al.
V.; Ivachtchenko, A. V. Microwave-mediated reactions of 3- aminomethylpyridines with acetylenedicarboxylates. A novel synthetic route to dihydronaphthyridines and naphthyridin-1ones.
Tetrah. Lett.
, 46 (23), 3953–3956 (2005).
70.
Lakner, F. J.; Xia, H.; Pervin, A.; Hammaker, J. R.; Jahangiri, K G.; Dalton, M. K.; Khvat, A.;
Kiselyov, A.; Ivachtchenko, A. V. A novel mesoionic ring system: unusual cyclization of thio- and amino-acid derivatives of 6-azauracil.
Tetrah. Lett.
, 46 (32), 5325–5328 (2005).
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