Mini-Tox: Liberia Management of common and commonly problematic toxicological emergencies Andrew Shannon, MD MPH Jacobi Medical Center Emergency Medicine Residency Albert Einstein College of Medicine, Yeshiva University Objectives and Outline Brief overview of important initial steps in managing intoxications History Toxicological physical exam and adjuncts Toxidromes Gastric decontamination Approach to coma Specific poisonings Acetaminophen (APAP) Salicylates CO / CN Caustics / Iron Alcohols Drugs of abuse Special psychiatric overdoses Toxic bradycardia Pesticides Heavy Metals Helpful Resources Poison Centers in the US: 1-800-222-1222 Vaults of Erowid: www.erowid.org Lycaeum: www.lycaeum.org MMWR: www.cdc.gov/mmwr Medwatch: www.fda.gov/medwatch Emergency Preparedness and Response: www.bt.cdc.gov Household Products Database: http://housholdproducts.nlm.nkh.gov Cornell Univ. Poisonous Plants Informational Database: www.ansci.cornell.edu/plants Dartmouth Toxic Metals Research Program: www.darmouth.edu/~toxmetal History Pts p/w ingestions may not be reliable AMPLE Hx SI/HI who called EMS? why? altered mental status (AMS) Family EMS (check ACR!) MiSys- prior visit/med hx allergies, medications (recent changes), procedures, last po intake, what led up to incident Ingestion Hx chemicals/meds available to pt? (ie Soc Hx) how much, when, why? SI/HI, accidental med OD, abuse/Munchausen by proxy paraphernalia/bottles at scene last time Pt noted to be at baseline? Physical Exam HEENT ABC’s GCS - not prognostic Dry if wet, warm if cold, cool if hot Re-address decon and staff safety/contamination Vital Signs (VS) do not rely on a “Nurses’ 20” for RR If you can’t get a BP, there probably isn’t one FSBG is 6th VS! Skin rales Abd diaphoresis; piloerection cyanosis track marks CV Chest Count/repeat yourself “E” – Exposure/(EKG) “D”- Disability/(Dextrose) signs of trauma MMM; burns nystagmus, pupils bowel sounds Neuro MS (O x ?); gag gait tremor, fasciculation, DTRs Adjuncts to Physical Exam FSBG Lab tests Arrhythmias Intervals End-organ effects (ischemia) CXR/AXR Aspiration Free-air / perforation Radio-opaque ingestants Order: EKG by now you’ve realized this is important body packers/stuffers halogenated hydrocarbons Fe, K, I or heavy metal compounds enteric coated preparations APAP / ASA level bHCG Consider: anion gap anti-convulsant level CO level EtOH level CPK ABG / VBG / lactate NH4 osmolality “Toxidromes” Sympathomimetic Hyperthermia Tachycardia Hypertension Mydriasis Diaphoresis AMS – agitated/combative, hallucinations, seizure Narcotic Pinpoint pupils (variable) AMS – obtundation Decrsd RR Sedative/Hypnotic AMS – obtundation Normal VS! CAUTION: toxidromes are generalities, and intoxications may not present classically, especially in mixed ingestions “Toxidromes” Cholinergic Muscarinc – “leaky” Anti-cholingergic SLUDGE: salivation, lacrimation, urination, diarrhea, GI cramps, emesis “Terrible B’s”: bradycardia, bronchorrhea, bronchospasm Nicotinic Autonomic: diaphoresis, mydriasis, tachycardia, HTN Neuromuscular: fasciculation, weakness, paralysis hyperthermia tachycardia/HTN dry/flushed skin; dry MM mydriasis decrsd bowel sounds urinary retention AMS – agitation, hallucination, seizure “Red as a beet, dry as a bone, hot as hell, blind as a bat, mad as a hatter” Classically, cholinergic toxidrome includes constricted pupils (miosis), but this is variable (agent; predominating effect) Gastric Decontamination Ipecac ~20 min to V onset No role in ED setting Gastric lavage Consider if <1 hr, critical toxin, protected airway Contraindicated: caustics, large or sharp FBs L lat decub/Trendelenberg, suction, intact gag or ETT Measure nose to xiphoid, confirm position, lavage until clear 36-40 Fr in adults; 22-24 Fr min in children “critical toxin” = a small decrease in toxin burden may have large impact on clinical status; i.e. TCAs, CCBs, colchicine, Li… Activated Charcoal Adsorbs many toxins MDAC (multi-dose) optimal charcoal: toxin ratio 10:1 Initial dose in unkn ingst 1 g/kg Must mix slurry well! (actual charcoal is in bottom of bottle) NOT USEFUL in… small molecules (Li, Fe, Pb) hydrocarbons, alcohols when endoscopy indicated (caustics) phenobarb, dapsone, theophylline, digitoxin, phyentoin, carbamazepine ensure cathartic only w/ 1st dose! Cathartics sorbitol (0.5g/kg), Mg citrate or sulfate AC contraindicated: gut perforation or ileus sig aspiration risk Whole Bowel Irrigation Rarely indicated metaclopramide; NGT; dose of AC minimum 1.5-2 L/hr (adult) or 25 mL/kg/hr (child) PEG large burdens poorly adsorbed (AC) agents (Li, Pb, Fe, Zn) or SR/ER preps In consultation w/ GI for body-packers (“mules”) Golytely, Nulytely, Colyte until rectal effluent is clear (? rectal tube) re-dose AC Contraindications No bowel sounds; obstruction or perf; unstable pt; unprotected compromised airway Coma Care of the undifferentiated coma patient is EM distilled ‘As a rule,’ said Holmes, ‘the more bizarre a thing is the less mysterious it proves to be. It is your commonplace, featureless crimes which are really puzzling, just as a commonplace face is the most difficult to identify.’ ATLS / ACLS / PALS protocols are key C-spine stabilization? HCT to r/o chronic subdurals? Roll the patient so you don’t miss the bullet hole… Infxn, SAH, CVAs, MIs, Ao dissections leading to CVAs can all affect a Pt’s “responsiveness” Coma due to toxins should be treated in the same way, with emphasis placed on above measures and observations Coma “Cocktail” Thiamine 100 mg iv prior to dextrose Dextrose 0.5-1.0 g/kg D50 – “1 amp” (50cc of 5% dextrose = 25 g) D10 in children Narcan 0.05-0.1 mg IVP initially; textbook dose (0.01 mg/kg) Indicated when RR < 11 & AMS ½ life 60-90 min 4 kcal/g = ~100kcal (less than ½ a candy bar! Food is next!) duration of action 20-90 min; less than most opiates Flumazenil (?) Risk of precipitating seizure severely limits routine use Acetaminophen (APAP) N-acetyl-para-aminophenol; aka paracetamol peak serum lvls 30-60 min; hepatic metabolism #1 cause acute liver failure in US; #1 cause tox fatalities in OD, NAPQI metabolite becomes toxic as glutathione is depleted APAP lvls are sent on unknown ingestions/SAs toxic, treatable, time dependent, commonly co-ingested, ASYMPTOMATIC ½-24 hrs: N/V, no sxs, (? APAP OD interferes w/ FSBG) 24-48 hrs: RUQ pain, elevated LFTs, PT/INR, bilirubin 48-96 hrs: hepatic dysfxn, acidosis, coagulopathy, LFTs peak, hypoglycemia, jaundice, cerebral edema death 4-14 days: resolution APAP Hx- time of ingestion & amnt 150 mg/kg : potentially toxic dose (~ 7.5 g adults) within 24 hr Rumack-Matthew nomogram: acute ingestions only obtain 4-hr level (or as soon after as possible) in unknown time frame, if initial lvl is zero, the 4hr lvl will not rise to toxic AST sens for hepatic injury prognostic markers in acute injury PT/INR, CO2/pH, lactate, renal function, phosphate “extended relief” APAP: sequential release in same pill if 4 hr lvl above nomogram, treat; if not, repeat in another 4 hrs APAP N-acetylcysteine (NAC) “mucomyst” multiple mechanisms charcoal (AC) binds po NAC, but likely not significant po load 140mg/kg maint dose 70mg/kg q 4hrs x 17doses; 1330mg/kg/72hrs antiemetics, sweetners, etc.; ? po in asthmatics/anaphylactoid rxn risk iv load 150mg/kg in 200cc D5W ovr 1hr greatest benefit if started < 8 hrs; benefit for late start then 50mg/kg in 500cc x 4hrs; 100mg/kg in 1L x 16hrs separate protocol for children <40kg 2/2 fluid concerns; or give po Indicated in h/o ingestion presenting >8hrs out while awaiting lvl chronic large ingestions (>4g/day; >120mg/kg/day) high APAP lvl (nomogram) late (>24hrs) presentations w/ detectable APAP or high LFTs Salicylates ASA (acetylsalicylic acid) Methyl salicylate - “oil of wintergreen” max serum lvls ~ 1hr; in OD, ~ 4-6 hrs Michaelis-Menten (“saturation”) kinetics: from 1st to 0 order elimination initial resp alkalosis 2/2 direct stim of medulla 1 mL 98% m.s. = 1.4 g salicylate; 5 mL potentially fatal in 2 yo not present in young children, so present later w/ severe acidosis AG met acidosis 2/2 dcrsd renal excret of acids & uncoupling of oxidative phosphorylation, et al. resp acidosis superimposed on 10 mixed resp alk/met acidosis when ventilation fails-- from fatigue or ASA induced ALI Pre-terminal event “Salicylism” N/V, ALI, tachy, tinnitus, vertigo, cerebral edema, hepatitis, dehydration, hypoglycemia, hypokalemia ASA lvl MDAC 2-4 doses; IVF for dehydration RSI & subsequent impairment of hyperventilation may worsen acidosis Urine alkalinization: goal urine pH 7.5-9.0, ABG 7.45-7.55 >30mg/dL = s/sxs present : >100mg/dL requires HD repeat lvl hourly during Rx for symp salicylism, lvl > 40 mg/dL Hemoperfusion removes salicylate most efficiently HD can also correct lytes, H+ status ALI, AMS, coagulopathy, ARF, unable to tol IVF, acute lvl > 100 mg/dL Carbon Monoxide (CO) colorless, odorless tasteless gas mild exposure– HA, N, malaise sig exposure– chest pain, focal neuro signs, dysrhythmias, syncope venous carboxyhemoglobin (CO-Hb) lvl, beta-hcg ?EKG, ?CPK, ?UA, ?chem-7 nml CO-Hb 1-2%; smokers 5-10% poor correlation w/ sx’s ME uses >50% lvl is min lvl for lethality – “CO poisoning death” CO-Hb dcrs’s O2 carrying capacity shifts curve to the left (dcrsd O2 offloading to tissues) binds myoglobin inducing cardiac/skeletal muscle hypoxia binds cytochrome oxidase, blocking (not uncoupling!) mitochondrial oxidative phosphorylation induces CNS lipid peroxidation CO Rx O2 therapy at highest conc possible Hyperbaric O2 (HBO2): best effect if within 6 hrs primarily to prevent delayed neurological sequelae absolute indications for HBO2 pregnant w/ lvl >10% or fetal distress (3rd trimstr) CO-Hb > 25% unconscious/syncope on scene or ER, AMS, cerebellar signs, seizure or confusion end-organ ischemia (EKG chngs, chest pain, pH < 7.1) Asymp Pts or those asymp in 4-6 hrs w/ (-) lab/EKG findings d/c home Ongoing study to correlate CO finger sensor and blood levels! Cyanide (CN) suicide, homocide, nitroprusside, jewelry production, fumigants, combustion of inorganic materials, artificial nail remover blockade of electron transport chain anaerobic metabolism lactic acidosis high AG, lactate, & central venous O2 sat CN antidote kit suspect in acidotic CO poisonings w/ high lactate (ie >10mmol/L) 1) induce methemoglobinemia to bind CN: 20-30% metHb tolerable amyl nitrite pearls – inhaled while awaiting iv access sodium nitrite (3%) - 0.33 mL/kg to max 10mL ovr 2-4min 2) sodium thiosulfate (25%) – 1.65 mL/kg to max 50mL (adults); may repeat dose Cyanokit – hydroxycobalamin 5g (70mg/kg) ovr 15 min cyanocobalamin (B12) formed, chelating CN initial hypotn possible; subsequent dosing uses longer infusion (6-8hrs) CO & CN poisoning avoid metHb in setting of CO-Hb; use only the sodium thiosulfate and HBO2 Caustics Acid – H+ donator – pH < 3; coagulation necrosis Base – H+ acceptor – pH >11; liquefactive necrosis Pts w/ sx’s require w/u incld bloods & CXR (r/o perf) endoscopy intentional ingestions, stridor, pain, vomiting, drooling within 12 hrs, no later than 24 Grade I – hyperema/edema, w/o ulceration Grade IIa/IIb – submucosal lesions, exudates not/near-circumferential Grade III - deep ulcers/necrosis into peri-esophageal tissues med clear if can eat/drink; no incrsd risk for stricture/CA IIa; soft diet as tol; NGT under direct visualization prn IIb/III; risk for perf/infxn (days to wks); all form strictures; ?Surg consult airway inspection (direct/fiberoptic laryngoscopy); ?ETT, ? dexamethasone Caustics Gastric decon contraindicated except large acid ingestions, ZnCl2, HgCl2 ? gastric emptying w/ narrow NGT if < 30 min bleach (sodium hypochlorite, NaOCl) ammonia (ammonium hydroxide, NH4OH); 3-10% household, 28% industrial str severity of systemic absorption may outweigh risks lrg industrial str exposures or those w/ sx’s require w/u otherwise clear if tol po Ophthalmic exposures immediate high vol irrigation for at least 15 min check pH (UA, litums paper, nitrazine paper), goal pH 7.4 ?ant chamber irrigation; d/w Ophtho Iron Direct GI irritant, vasodilator, neg ionotrope, disrupts electron transport chain & aerobic metabolism Min/no sxs- observe 6 hrs; if no sxs, d/c Mild/mod tox- emesis, mild tachy, mild acidosis local effects N/V/D onset < 6 hrs from ingestion Rx if: Fe on KUB, persistent clin toxicity (>4 episodes emesis), acidosis, serum Fe > 350 mcg/dL, estimate of elemental Fe >2060mg/kg sulfate 20% eFe; gluconate 12%, fumarate 33% Severe tox – GIB, acidosis, AMS, hypotn, coagulopathy IVF, RBCs, lavage/WBI if feasible; ICU admission iv deferoxamine: start 5mg/kg/hr, titrate up to 15mg/kg/hr as BP allows obtain pre-Rx and 4-6hr post-Rx UA when urine color returns to baseline, no more free Fe is being chelated DFO Rx should stop @ 24hrs; safe in pregnancy Alcohol Intoxication “Intoxicated” is a clinical diagnosis 1 g/kg EtOH = serum lvl 100mg/dL ~ 1 hr later 12 oz beer (5%EtOH) x (30 mL/oz) x 0.8 g/mL = 14.4 g EtOH 5 oz wine (12%EtOH) = 14.4 g EtOH 1.5 oz liquor (40%EtOH) = 14.4 g EtOH “proof” ~ 2 x %EtOH unhabituated patients eliminate EtOH 1520mg/dL/hr alcoholics avg 25-35 mg/dL/hr Alcohol Intoxication Withdrawal from EtOH 6-24 hrs after last drink - "the shakes“ 4-24 hrs – hallucinosis persecutory auditory, visual, tactile hallucinations w/o delirium 6-72 hrs – “rum fits” tremor, tachycardia, diaphoresis, anorexia, insomnia generalized seizures 3-10 days - delirium tremens (DT) disorientation, fever, visual hallucinations Managing Alcohol High incidence of infection/trauma ?HCT, ?c-collar & c-spineCT, ?LP, ?CXR Dehydration w/ osmolar gap VS, FSBG, ?chem-7, ?CPK, ?EtOH lvl (prognostic), ?osms “Banana bag”/“Osler bag”/“Rally pack” – expensive D5NS or ½NS, 2g MgSO4, 10mL MVI, 1mg folate, 100mg thiamine thiamine only vitamin affecting outcome (dcrsd incidence DTs) Alcohol Withdrawal diazepam 10mg ivp lorazepam 2mg ivp no active metabolites (liver pts) phenobarbital 130 mg iv (up to 390mg) shorter time to peak onset of action failure to respond to benzos (200mg / 40mg) in first 3-5 hrs prepare for intubation; arrange ICU admission IVF, MgSO4 phenytoin – no role in w/d sz’s unless a proven focus chlordiazepoxide – mild/early w/d 50-100 mg/d single or divided dose Elderly/debilitated: Initial 10 mg PO/IV/IM Detox: 25 mg PO q6h for 1 d, q8h for 1 d, q12h for 1 d, qhs for 1 d Toxic Alcohols Ethylene glycol – antifreeze, coolants; “sweet” tasting LD 1-1.5 mL/kg cardiac depression, ATN (Ca oxalate crystals in UA), AG acidosis, hypo-Ca UA can fluoresce under UV (Wood’s lamp) light; poor Sens/Spec Glycolic acid (metabolite) may cross-react with some lactate assays! Detox cofactors - pyridoxine (B6) 50mg q6hr; thiamine (B1) 100mg q6hr HD indications – serum lvl >25mg/dL, acidosis, pulm edema, renal failure, VS instability Methanol – “wood alcohol” solvents, windshield washer fluid, paints/removers, varnishes, “canned heat” LD 15-30mL; metabolized into formaldehyde/formic acid Ocular toxicity “snowstorm” vision, ARF/myoglobinuria, CNS dep & seizures, N/V Optic disc hyperemia Detox cofactors – folic or folinic (leucovorin) acid 1 mg/kg up to 50 q 4-6 hrs iv HD – serum 20-50mg/dL, acidosis, visual impairment, renal failure, VS instability Toxic Alcohols NaHCO3 to alkalinize urine may enhance metabolite excretion Fomepizole – ADH competitive inhibitor witnessed ingestion/strong history; lvl >25mg/dL; lrg osmol gap w/ suspicion; significant unexplained AG acidosis load 15mg/kg over 30 min; 10mg/kg q 12 for 48hrs; then 15mg/kg q 12 reload post-HD Isopropyl alcohol – “rubbing alcohol” solvent, disinfectant, window cleaners, skin/hair products LD (70% soln) 1 mL/kg metabolized to acetone significant ketosis w/ minimal acidosis CNS dep, unstable VS, N/V, ATN, hemolytic anemia, myoglobinuria HD indications- uncorrectable hypotn, deep coma, VS instability, serum lvl > 400-500mg/dL supportive care Drugs of Abuse Opiates (natural); Opioids (semi-/synthetic) CNS,CV & respiratory depression, histamine release Lomotil (diphenoxylate) and Imodium (loperamide) poorly absorbed, may give acute toxicity Narcan (naloxone)- typically needed if RR < 11 miosis common, not universal (esp. w/ coingestant) hypoventilation, rhabdomyolysis, hypothermia, concomitant APAP toxicity, lung injury (talc pneumonitis, ALI ?2/2 naloxone) 0.05mg test dose, escalate prn, lowest effective dose q 2-3min If infusion needed, use 2/3 of dose giving a response / hr Clonidine overdose may appear identical 50% pediatric clonidine ODs may respond to naloxone Opiates Withdrawal – if iatrogenic, do not give opioid! unpleasant, not dangerous Methadone- 10mg IM; 20mg po (dissolved) piloerection, mydriassis, incrsd BS, yawning, diaphoresis, larcimation, N/V effective regardless of abuse pattern use antiemetics prn DO NOT give full methadone maint dose, esp if unverified if diverting, “prescribed” dose potentially an acute OD Clonidine 0.1mg-0.3mg po q1hr until sx’s improve ? maint dose 0.3mg bid/tid watch for hypotn Sympathomimetics Cocaine, amphetamines CVA, szs, MI, hypo-/hypertn, hyperthermia, bronchospasm, pneumothorax/mediastinum, rhabdomyolysis, quinidine effect (dysrhythmias, interval prolongation), placental abruption (2nd/3rd trimester) Chest pain AMI risk in 1st hr after cocaine use 24x normal 6% pts w/ cocaine CP have CE elevations EKGs less sens/spec for MI in recent cocaine users cocaine prothombotic “Crack lung” 1-48hrs s/p smoking - hypersensitivity pneumonitis acute pulm infiltrates, pain, eosinophilia benzos (diazepam 2.5mg), external cooling nitroglycerin, ASA, ?CCBs in pts w/ concern for ACS withdrawal – lethargy, dysphoria Benzodiazepines “Coma with normal vital signs” RR should be normal DDx: head trauma, stroke, hypoglycemia, CO poisoning, multisubstance ingestion ABCs: ?ETT EKG, FSBG, bHCG, EtOH lvl “Anyone who can tolerate a nasopharyngeal airway probably deserves one” if awake, activated charcoal most pts are arousable within 12-36 hrs w/ supportive care Flumazenil: use only to avoid an intubation! 0.5mg slow IVP 1-2 hrs to max 5.0 mg w/d similar to EtOH predictable based on pharmacokinetics chronic use of long-acting agents (diazepam) may delay w/d 4-10 days Psychiatric Overdoses TCAs: NE/DA/5-HT reuptake blockade anti-cholinergic effects, antihistamine effect, Na channel blockade ABCs; orogastric lavage if < 1 hr; AC 1-2 doses (q4hrs) EKG as screen: QRS <100ms = no toxicity >100ms = 1/3 pts w/ szs: ADMIT, think about ICU >160ms = ½ pts w/ ventricular dysrhythmia: ADMIT to ICU NaHCO3 2 amps (1-2mEq/kg) bolus – observe response on rhythm strip 3 amps in 1 L D5W @ 2-3x maint; goal narrow QRS or max pH 7.55 replete Mg, K consider 24 hr tele admission for pts w/ persistent HR > 120, or QTc > 480 No Sz, nml EKG (exept tachy that resolves) observe 6 hrs to clear terminal 40 ms R axis deviation: aVR R wave > 3mm (~ 81% PPV for poisoning) w/ R/S ratio in aVR > 0.7 ; deep slurred S wave in I & aVL long QT, sinus tach Mood Stabilizers Lithium precipitants- dehydration, renal dysfunction, preeclampsia, Na depletion, thermal stress, drug interactions NSAIDs, carbamazepine, ACE-Is/ARBs, metronidazole, antipsychotics, diuretics tremor, slurred speech, ataxia, hyperreflexia/clonus, sz, CV collapse, EPS acute- dilute urine, prolonged QT, hypothyroid, inc WBCs chronic- nephro DI, interstitial nephritis, aplastic anemia, dermatitis IVF; WBI if SR preparations ingested repeat Li lvl 2 hrs after initial draw in acute (6 hrs in chronic) OD HD: call nephrologist w/ 2nd lvl value S/Sxs neurotoxicity (AMS); unable to eliminate Li (ARF); unable to tol IVF load (CHF); Li lvl > 4.0mEq/L (acute) or > 2.5mEq/L (chronic) “re-bound”- tissue redistribution requires post-HD lvl and again 6 hrs later Mood Stabilizers Valproic acid (VPA) carnitine depletion leads to hyperammonemia 11% pts w/ asymp chemical hepatitis risk for (rare) fulminant hepatic failure, hypoglycemia OD usually benign, self-limited drowsiness > 30mg/kg coma, respiratory depression poor correlation w/ serum lvls; repeat in 2-3 hrs for downward trend consider NH4 lvl, lytes, lactate if AMS MDAC in lrg acute OD w/ rising lvls HD: deterioration, hepatic dysnfxn, rising lvls, VPA > 1000mg/L carnitine supplement: VPA-induced hepatotoxicity, NH4 > 35 micromol/L, peds <2 yo or on ketogenic diets 100mg/kg (max 6g) ovr 30 min iv 100mg/kg/day (max 3g) divided q6hrs po Toxic Bradycardia CCBs rapid onset 1-2 hrs IR, SR 12-18 hrs BBs CHF, low HR, bronchospasm, hyper K, hypoglycemia (children) early onset of effect (<6hrs); peak 1-4 hrs verapamil – nodal (HR, CO) nifedipine – peripheral (SVR) (sotalol may delay >24hrs) Clonidine onset 30-60 min; peak 2-3 hrs naloxone, IVF, atropine, pressors Toxic Bradycardia atropine 0.5-1.0mg (0.02mg/kg) q2-3min, max 3mg CaCl2 10-20 cc 10% soln (1-2 amps); slow IVP ovr 3-5min 3-6 amps Ca gluc q 15-20min; up to 5 gms w/o serial Ca, PO4 peds 10-20 mg/kg Ca gluc (10% soln ~ 0.1cc/kg) glucagon 2-5mg slow IVP, q5-10min; 10mg max; BB>CCBs hypotn 2/2 myocard dep, not incr vagal tone slows gut in pts receiving WBI gtt to follow; mg/hr = effective initial dose mg peds 50-150 mcg/kg; gtt 50mcg/kg/hr pressors (NE) pacing – often ineffective Pesticides 200,000 deaths/yr leading cause of suicide/unintentional poisonings Vomiting, diarrhea resp distress LOC Cholinesterase inhibitors cholinergic toxidrome (miosis, SLUDGE, “killer ‘B’s”) organophosphates bradycardia is muscarinic, but bronchorrhea/constriction induced hypoxia may cause tachycardia penetrate latex/vinyl; leather is reservoir; 0.5% hypochlorite bleach or alcohol based soap for dermal decon “age” – irreversible inactivation of AChE carbamates reversible binding- no aging muscarinic > nicotinic effects Pesticides atropine 0.5-1.0 mg (0.02 mg/kg) initial; double dose q2-3min pralidoxime (2-PAM) titrate to drying of bronchial secretions 0.5mg min adult dose (0.1mg peds) 2/2 paradoxical brady no effect on nicotinic neuromuscular junction (paralysis) frees un-”aged” AChE 1-2 g in 100 cc NS (25mg/kg, max 1 g) ovr 15-30min; then q6-12hr WHO regimen: 30 mg/kg iv bolus; then > 8mg/kg/hr gtt glycopyrrolate/ipratropium periph-acting/inhaled anti-muscarinics may be considered as adjuncts to atropine for clearing lung secretions Pesticides Sxs usually unlikely if not developed in 6-12 hrs exceptions: fenthion, VX gas (nerve agent) ~ 24 hrs Sequelae of organophosphate/carbamates “Intermediate Syndrome” acute prox/resp muscle wkns; cranial neuropathy 24-96 hrs following poisoning; up to 1st few wks unpredictable occurrence supportive care; pralidoxime/atropine as indicated persistent sensory/motor neuropathy occasionally Pesticides Organochlorines DDT, benzene hexachloride (Lindane), aldrin, etc. Pyrethrins and Pyrethroids permethrin, deltamethrin, fenvalerate supportive Rx for agitation, szs; decon supportive Rx; paresthesias self-limited (top vit E) Nicotine/neonicotinoids nithizaine, dinotefuran, thiacloprid irritant, szs, resp dep decon (skin), supportive care Marine toxins Ciguatera tropics/subtropics; reef dwelling tropical fish barracuda, moray eel, amberjack, grouper, mackerel, parrot fish, red snapper GI (N/V), CNS (palsies, paresthesias, hot/cold reversal), CV (heart block, brady), fatigue/malaise Scombroid tuna, mackerel, skip-jack, bonito, mahi mahi, bluefish, amberjack flushing, rash, palpitations, tachycardia anti-H1,2, epinephrine, beta-agonists Heavy Metals Multi-system toxicity Acute GI: N/V/diarrhea – most metal salt ingestions Renal: proteinuria, aminoaciduria, ATN CV: response to volume loss, dysrhythmia, congestive CM CNS: dMS; periph neuropathies in hours to days Hair/skin/nail changes: lag days -wks behind acute exposure Chronic CNS/PNS: predominate Heme: anemias, cytopenias Renal: CRI/CRF CA: various Skin: rashes, colored lines on nails/gums Heavy Metals Arsenic ABCs, gastric emptying/AC KUB to r/o residual GI content inhaled dusts; copper/lead/zinc ore smelting; pesticides/herbicides; naturally occurring well water IM Dimercaprol (BAL) if can’t take po; ?add DMSA (meso-2,3dimercaptosuccinic acid) when GI tract clear Mercury Elemental- medical, Ore processing, mining, jewelry/battery making Inorganic salts- batteries, calomel, dyes, fireworks Organic- antiseptics, fungicides, by-products supportive/ABCs; AC for HgCl Milk, NAC, egg whites- may bind salts in gut BAL: acute (esp GI) tox- not in organic Hg DMSA: organic Hg, chronic or mild tox, when tol po Heavy Metals Lead wrist-drop (PNS effects); Fanconi-like nephropathy; plumbism-gout crystal, solder, glaze, batteries, traditional meds ABCs/supportive care R/o GI burden; DMSA for sxs or elevated levels; BAL followed by Ca EDTA if encephalopathy present Thalium: semi-conductors, insecticide/rodenticide, jewelry salts; elemental/organic v. rare GI absorp; ~ 1 g lethal dose in adults MDAC likely helpful Prussian Blue enhances gut elimination via K exchange BAL, EDTA, etc. not effective References New York City Poison Control Center. An intensive review course in clinical toxicology; March 13-14, 2008. All Rights Reserved. Toxicology and Pharamacology. In Emergency Medicine: A comprehensive study guide, 6th ed. Tintinalli JE, Kelen GD, Stapczynski JS Eds. McGraw-Hill Companies, Inc. 2004