International Center for Chemical and Biological Sciences
University of Karachi, Karachi-75270
Pakistan
List of US Patents Filed
1.
"Immunosuppressive Compounds" M. Ahmed Mesaik, Khalid M. Khan,
Omer M. Abdalla, Fazal Rahim, A. Shukralla, Khalid, Zaheer-ul-Haq,
Shahnaz Perveen, Samreen Soomro, Sobia A. Halim, Patent Ref. 2012.1219,
Application No. 13 / 921 / 705, 6/9/2013.
2.
Schiff Bases of Thiazoles: A New Class Of Ureases Inhibitors, M. Iqbal
Choudhary, Khalid M. Khan, Ajmal Khan, Nida Ambreen, Atia-tul Wahab,
Atta-ur-Rahman, Application Ref. 2013.0424.
3.
Anti-Glycation Properties of Oxindole Derivatives, M. Iqbal Choudhary,
Saima Rasheed, Nessar Ahmed, Khalid M. Khan, Momin Khan, Atta-urRahman , Atia-tul Wahab, Application reference 2013.0330.
4.
Anthranilic Acid Derivatives Nopvel Inhibitors of Advanced Glycation End
Products (AGEs) Formation, Atta-ur-Rahman, M.Iqbal. Choudhary, H. Jahan,
K. M. Khan, A. Atta, Serial No.13/968,071, 15/08/2013.
5.
Small molecule activators of HSIV protease for development of novel
antimicrobials, M. Kamran Azim, Yasmeen Rashid, Khalid M. Khan,
Application ref. 2013.0412.
6.
Patulitin a potent anti-TNF-and antiarthritic compound from Tagetes patula,
M. Ahmed Mesaik, Almas Jabeen, Shaheen Faizi, Shabana U. Simjee, Samina
Bano, Lubna, Application ref. 2013.0520.
7.
Artonin I to Treat Resistant Infectious Staphylococcus Aureus, M. Iqbal
Choudhary, Saba Farooq, Atia-tul-Wahab, Christian D.A. Fozing, Atta-urRahman, U.S. Patent Application Serial No. 13/740,919, 14/1/2013.
8.
Quinazolines as -glucuronidase novel inhibitors, M. Iqbal Choudhary,
Khalid M. Khan, Syed Muhammad Saad, Nimra Naveed Sheikh, Sammer
Yousuf, Atta-ur-Rahman, U. S. Patent Application Serial No. 13/789,021,
03/07/2013.
9.
Synthesis and Biological Studies of an Isomeric Mixture of (E/Z) Isoxylitones
and Its Analogues, Atta-ur-Rahman, M. Iqbal Choudhary, Farzana Shaheen,
Shabana Usman Simjee, Noureen Khan, Saima Mahmood Malhi, Syed Uzair
Ali Shah, Muhammad Nadeem Ashraf, Application No. 13/758/027, 2/4/2013.
10.
Bioactive antioxidants from plant foods, potential candidates for nutraceutical
products development, M. Iqbal Choudhary, Juveria Siddiqui, Ahmed
Abbaskhan, Suad Naheed, Achyut Adhikari, Jalauddine A. Jalal Awalia,
Application No. 13/759/820, 2012.
11.
Heterocyclic Schiff’s Bases as Novel and New Antiglcation Agents, S. Ibrahim, I.
Warad, M. A. Al-Nuri, M. I. Choudhary, Atia-tul-Wahab, S. Rasheed, Application
Number: 13/757, 956, 02/04/2013.
12.
Overcoming Antibiotic Resistance in Staphlococcus Aureus by new Thiruea
Dervatives, M.I. Choudhary, S. Farooq, K.M. Khan, F. Naz, Atia-tul-Wahab, Atta-urRahman, 2013. (Submitted).
13.
Thiourea Derivatives as -Chymotrypsin Inhibitors, Atta-ur-Rahman, M.Iqbal.
Choudhary, B. P. Marasini, K. M. Khan, F. Sheikh, Atia-tul-Wahab, 2013.
(Submitted).
14.
Abdullah Mohammed Al-Majid, Mohammad Shahidul Islam, Assem Barakat,
Sammer Yousuf, and M. Iqbal Choudhary, Catalytic Asymmetric Synthesis of Novel
Pharmacophores as -Glucosidase Inhibitors Incorporating Indole Moiety Ref. 2013.0902,
07/03/2013.
LIST OF US PATENTS GRANTED
15.
Anticancer compound, Saif Ullah, Saifullah Khan, Azzizuddin Muhammed
Kashif, Ahsana Dar, Muhammad Iqbal Choudhary, United States Patent
Publication # 2013/0018025, Application Number: 13/184548, publication
Date, 17/01/2013.
16.
Method of producing tibolone metabolites by fermentation with Gibberella
fujikuroi, Atta-ur-Rahman, Muhammad Iqbal Choudhary, Syed Adnan Ali
Shah, Shamsun Nahar Khan, United States Patent 8148557, Application
Number: 13/015559, Publication Date: 04/03/2012.
17.
Method of producing tibolone metabolites by fermentation with Fusarium lini,
Atta-ur-Rahman,
Muhammad Iqbal Choudhary, Syed Adnan Ali Shah,
Shamsun Nahar Khan, United States Patent 8148558 , Application Number:
13/015554, publication Date, 04/03/2012.
18.
Anti-inflammatory compound, Saif Ullah, Saifullah Khan, Muhammed
Ahmed Mesaik, Zaheer-ul Haq, Almas Jabeen, Sobia Ahsan Halim,
Muhammad Iqbal Choudhary, United States Patent 8329678, Application
Number: 13/184551, publication Date, 12/11/2012.
19.
Formulations against cutaneous leishmaniasis, Atta-ur-Rahman, Muhammad
Iqbal Choudhary, Sammer Yousuf,, Samreen Khan, Farooq Rahman Soomro,
Shahida Perveen, United States Patent 8287921, Application Number:
13/189509, Publication Date, 10/16/2012.
20.
Method of producing tibolone metabolites by fermentation with Rhizopus
stolonifer Atta-ur-Rahman, Muhammad Iqbal Choudhary, Syed Adnan Ali
Shah, Shamsun Nahar Khan, United States Patent 8148556, Application
Number: 13/015551, Publication Date, 04/03/2012.
21.
Method
of
producing
tibolone
metabolites
Cunninghamella elegans, Atta-ur-Rahman,
by
fermentation
with
Muhammad Iqbal Choudhary,
Syed Adnan Ali Shah, Shamsun Nahar Khan, United States Patent 8198041,
Application Number: 13/015553, Publication Date, 06/12/2012.
22.
7-Nitro-2-(3-nitro phenyl)-4H-3,1-benzoxazin-4-one or derivatives thereof for
treating or preventing antiviral infections, Shaikh Riazuddin, Atta-ur Rahman,
Usman Zafar, Muhammad Iqbal Choudhary, Usman Ali Ashfaq, Khalid M
Khan, Tayyab Husnain, Zulfiqar Ali Khan, Javed Akram, United States Patent
8148368, Application Number: 2/876999, Publication Date,04/03/2012.
23.
Novel
hydroxylated
enantiomers
of
(-)
3a,6,6,9a-
tetramethylperhydronaphtho[2,1-b]furan as perfuming agents derived from a
fungal fermentation process, Atta-ur-Rahman, Muhammad Iqbal Choudhary,
Syed Ghulam Musharraf, Amtul Sami, United States Patent Application
Number: 13/115991, Publication Date, 11/29/2012.
24.
Antitubercular alkaloid, Sabra Begum, Syed Nawazish Ali, Bina Shaheen
Siddiqui, United States Patent Application Number: 13/035756, Publication
Date: 08/30/2012.
25.
Steroidal antitubercular compounds, Bina Shaheen Siddiqui, Nasima Khatoon,
Sabira Begum, United States Patent Application Number: 13/037494,
Publication Date: 09/06/2012.
26.
α-Glucosidase inhibitors from lichens, Vinitha Moolchand Thadani, Shamsun
Nahar Khan, Veranja Karunratne, Muhammad Iqbal Choudhary, United States
Patent 7867989, Application Number: 11/767465, Publication Date,
01/11/2011.
27.
Tyrosinase enzyme inhibitors from fungal hydroxylation of tibolone, Atta-urRahman, Muhammad Iqbal Choudhary, Syed Adnan Ali Shah, Mahmud
Tareq Hassan Khan, Application Number: 11/944476, Publication date,
05/28/2009.
28.
Natural Novel Antioxidants, Muhammad Iqbal Choudhary, Sajjad Ali, Vinitha
M. Thadani, Veranja Karunaratne, United States Application Number:
11/838567, Publication Date, 02/19/2009.
29.
α-Glucosidase inhibitors from fungal hydroxylation of tibolone and
hydroxytibolones Atta-ur Rahman,
Muhammad Iqbal Choudhary, Syed
Adnan Ali Shah, Shamsun Nahar Khan, Application Number: 11/944475,
Publication Date, 05/28/2009.
30.
Anticonvulsant compounds, Atta-ur-Rahman, Muhammad Iqbal Choudhary,
Farzana Shaheen, Shabana Simjee, A. Ganesan, Mohsin Raza, United States
Patent U.S. 7399888 B-2; Application Number: 11/307251, Publication Date:
01/03/2008.
31.
New α-glucosidase inhibitors and antibacterial compounds from Myrtus
communis L. Atta-ur-Rahman,
Muhammad Iqbal Choudhary, Farzana
Shaheen, Manzoor Ahmad, Shamsun Nahar Khan, Shazia Anjum, Application
Number: 11/306345, Publication Date,10/30/2008.
32.
Novel α-glucosidase inhibitor from Tabernaemontana dichotoma, Mirihanage
Don Jayantha Wijayabandara, Shamsun Nahar Khan,
Muhammad Iqbal
Choudhary, Application Number: 11/553465, Publication Date, 05/01/2008.
33.
New treatment of diabetes mellitus, Viqar Uddin Ahmad, Nasir Rasool,
Muhammad Iqbal Choudhary, Shamsun Nihar Khan Application Number:
11/309013, Publication Date:12/13/2007.
34.
Collier, H.O J, Saeed, S.A, Schneider C and Mannuzza F. : "Method for
reducing endogenous prostaglandin synthesis". U.S. Patent No. 4, 129, 648
(1978).(Miles Laboratories Inc.), USA.
35.
Saeed S.A. : "Method for the preparation of prostaglandin synthetase". U.S.
Patent No. 4, 070, 242 (1978).(Miles Laboratories Inc.), USA. Canadian
Patent No. 1009181 (1977).
36.
Saeed SA. (Miles Laboratories, Inc.), USA."Apparatus for Large Scale Gel
Electrophoresis" U.S. Patent No. 3, 888, 758 (1975).
37.
Saeed SA, Schneider C and Phillips BM. : "Method of treating inflammation
utilizing alkyl esters of Gallic Acid". U.S. Patent No. 3, 833, 732
(1974).(Miles Laboratories Inc.), USA.
38.
Saeed SA and Saeed SO: Anti-platelet aggregation compositions N-Acetyl-2aminophenol. U.S. Patent (Applied). 2008. United States Patent application
20050084528.
LIST OF NON-US PATENTS
1. Development of process for preparation of new spasmolytic composition from
Psidium guajava leaves, Sabira Begum, Bina S. Siddiqui, S.I. Hassan, A.H. Gilani
and M. N. Ghayur , CBR # 1. The Patent Office, Govt. of Pakistan, Patent Serial
No. 140597 (2010).
2. A process for the preparation of pesticidal composition Biosal from the dried
neem seeds (Kernel), Bina S. Siddiqui, S. Naeem-ul-Hasan Naqvi, Syed Tariq Ali
and Shaheen Faizi, The Patent Office, Govt. of Pakistan, Patent Serial No.
140326, (2010).
3. A Process for the synthesis of new anti-Tuberculosis agents, Sabira Begum, S. N.
Ali and B.S. Siddiqui, Patent Application No. 1040/2009.
4. Antifungal formulation from Kalidium foliatum, Bina S. Siddiqui, Zh.Zh.
Karzhaubekova, G.Sh. Burasheva, and N.A.Sultanova, Patents Application No.
56218 (Kazakhistan) (2009).
5. Antibacterial formulation from Kalidium foliatum, Bina S. Siddiqui, Zh.Zh.
Karzhaubekova, G.Sh. Burasheva, and N.A.Sultanova, (2009).
6. Saeed S. A and Saeed S. O: N-Acetyl-2-aminophenol. UK Patent on
Orthacetamol. U.K. Patent No.2405092 (2008), UK Patent 9th April, 2005.
7. Neemex, A Biofertilizer-cum-pesticide based on the dried fruits (seeds) of
Azadirachta indica A. Juss, Bina S. Siddiqui, S.T. Ali and S.K. Ali, CBR # 3022
The Patent Office, Govt. of Pakistan, (2007).
8. Saeed SA and Saeed SO: Anti-platelet aggregation compositions. U.K. Patent No.
GB 2407040 (2007).
9. Bioaman – A botanical insecticidal composition for household use based on the
dried fruits (or kernel) of Azadirachta indica A.Juss, Bina S. Siddiqui, S.N.H.
Naqvi, S.T. Ali and S.K. Ali, CBR # 3021 The Patent Office, Govt. of Pakistan,
(2007).
10. Saeed SA and Saeed SO. : 2-hydroxyacetanilide to its pharmaceutical
composition containing it and its use as anti-inflammatory, analgesic, anti-pyretic
and anti-platelet agent. Pakistan Patent. SL No.138941 (2007).
11. The Manner of Obtaining Remedy Posses Antifungal Activity, B. K. Yeskalieva,
M. Iqbal Choudahry, G. Sh. Burasheva, N. A. Sultanova, Zh. A. Abilov, In print
2006.
12. The Manner of Obtaining Remedy Posses Antibacterial Activity, B. K.
Yeskalieva, M. Iqbal Choudhary, G. Sh. Burasheva, N. A. Sultanova, Zh. A.
Abilov, In print 2006.
13. The Manner for Obtaining of Antioxidant Polyphenols Complexes From Tamarix
laxa, A. K. Umbetova, M. Iqbal Choudhary, G. Sh. Burasheva, N. A., Sultanova,
Zh. A. Abilov, In print 2006.
14. The Manner for Obtaining of Antibacterial Polyphenols Complexes From
Kamphorosma monspeliacum, A. K. Umbetova, M. Iqbal Choudhary, G. Sh.
Burasheva, N. A Sultanova, Zh. A. Abilov, In print 2006.
15. Biosal-a pesticidal composition based on the whole fruits of Azedirachta indica
A. Juss. B. S. Siddiqui, S. N. H. Naqvi, S. T. Ali and Shaheen Faizi Serial number
# 2181 The Patent Office, Govt. of Pakistan Patent Application No. 1222/06,
2006.
16. Agrosal-a pesticidal composition based on the whole dry fruits (or kernel) of
Azadirachta indica A. Juss. Bina S. Siddiqui, S.N.H. Naqvi, Syed Tariq Ali,
Shaheen Faizi and Syed Kashif Ali, CBR # 2181 The Patent Office, Govt. of
Pakistan, (2006).
17. Development of a method for the production of bio-diesel, Bina S. Siddiqui, Syed
Tariq Ali and Jafar Nazir Usmani , CBR # 2180 The Patent Office, Govt. of
Pakistan (2006).
18. A process for preparing efficient and safe antioxidant and analgesic composition
containing xanthone-C-glucoside (Mangiferin) from Bombax ceiba, A. Dar,
Shaheen Faizi, S. Naqvi, T. Roome, S. Zikr-ur-Rehman, M. Ali Patent
Application No. 633/05, 2005.
19. Development of process for preparation of new spasmolytic composition from
Psidium guajava leaves, Sabira Begum, Bina S. Siddiqui, S.I. Hassan, A.H. Gilani
and M. N. Ghayur , CBR # 1. The Patent Office Govt. of Pakistan (2005).
20. A simple method of isolation of an antioxidant (patuletin) in large quantity from
flowers of Tagetes patula, A. Dar, Shaheen Faizi, S.Naqvi, H. Siddiqi, A. Naz, S.
Bano, Pakistan Patent, (2005).
21. A process for the development of an insecticidal composition based on neem
(Azadirachta indica) fruit coats., Bina S.Siddiqui, S.N.H. Naqvi, and S. Faizi ,
Patent # 138573 The Patent Office, Govt. of Pakistan, (2003).
22. A process for the preparation of a herbal composition for the skin treatment of
farm and pet animals, Bina S. Siddiqui, A.Dar and S. Faizi, Patent # 138572 The
Patent Office, Govt. of Pakistan (2003).
23. Some Fractions of Polyphenols of Tamarix ramosissima (Tamaricaceae) Posses
Antifungal Activity, N. A. Sultanova, T. Makhmoor, V. B. Omurkamzinova, M.
Iqbal Choudhary, Atta-ur-Rahman, Zh. A. Abilov, Patent No 11936, А 61К
35/78, Bulletin No 9 dated 16/09/2002.
24. Nematicidal composition NIMATICIDOL based on the aerial parts of Lantana
camara Linn, Sabira Begum, Bina S. Siddiqui, Aneela Wahab and Fatima Qamar,
Serial number 136887, The Patent office, Govt. of Pakistan, (2001).
25. Process for the Osmo-Drying of Fruits and Vegetables for the Production of New
Snacks, M. Iqbal Choudhary, Pakistan Patent Application No. 353/2000, dated
22/04/2000.
26. A process for preparing a composition to cure eczema from Melia azedarach
Linn, Shaheen Faizi, B. S. Siddiqui, R. Saleem, S. I. Ahmed and A. Wasi, Patent
Application No. 656/2000, S.I. No. 137331, 2000.
27. Antihypertensive medicine based on sahjana (Moringa olifera). Shaheen Faizi,
Bina S.Siddiqui, A.H.Gilani and Rubina Saleem, Serial number # 136438. The
Patent Office, Govt. of Pakistan, (2000).
28. Antihypertensive medicine aloedin based on Aloe barbadensis Mill, Rubeena
Saleem, Shaheen Faizi, Bina S. Siddiqui, Ahsana Dar, S. Iqbal Ahmed and M.H.
Qazi, Serial number # 136463. The Patent Office, Govt. of Pakistan, (2000).
29. A Novel Cholesterol-Lowering Edible Oil Composition Comprising of Garlic
Extract, M. Iqbal Choudhary, Pakistan Patent No. 135653, dated 23/01/1997.
30. Novel formulation of the antimicrobial composition, amoxycassia based on the
synergistic activity of Cassia fistula and amoxicillin, S.U. Kazmi, N. Hasan Ali
and Shaheen Faizi, Pakistan Patent (1999) Patent Application No. 1121/99, S.I.
No. 137124, 1999.
31. Nematicidal composition NIMATI-CIDOL base on the aerial parts of Lantana
camara Linn. Sabira Begum, Bina S. Siddiqui, Fatima Qamar and Aneela Wahab,
Serial number # 136887. The Patent Office, Govt. of Pakistan, (1999).
32. A
process
for
preparing
an
antihypertensive
composition
containing
anthraquinone from Aloe barbadensis Mill, R. Saleem, Shaheen Faizi, B.S.
Siddiqui, A. Dar, S.I. A. M.H. Qazi, Pakistan Patent 1998. Patent Application No.
862/98, 1998.
33. A process for preparing an antihypertensive composition containing Xanthone Cglucoside (Mangiferin) from Bombax ceiba Linn., Shaheen Faizi, R. Saleem, M.
Ali, S. I. Ahmed and M.H. Qazi, Pakistan Patent SI No. 136464 1998. Patent
Application No. 814/98, 1998.
34. Antihypotensive medicine Brassico based on Brassica rapa sb. sp. campestris,
A.H. Gilani, Irfanullah, F. Shaheen, S. Bibi, and Shaheen Faizi, Pakistan Patent SI
No. 136437 1998. Patent Application No. 871/98, 1998.
35. Antihypertensive composition containing thiocarbamate glycosides from Moringa
oleifera, Shaheen Faizi, B.S. Siddiqui, A.H. Gilani and R. Saleem, Pakistan Patent
1997. Patent Application No. 872/98, 1998.
36. A Preparation of Novel Composite Essential Oil Mixture Which is Identical to
Famous Garam Masala (Mixure of Spices), M. Iqbal Choudhary, Pakistan Patent
No. 135652, and dated 23/01/1997.
37. The Development of Simple Process for the High Yield Extraction of Essential
Oils From Different Aromatic Spices, Flowers and Nuts, M. Iqbal Choudhary,
Pakistan Patent No. 135689, dated 16/02/1997.
38. Demulsification of B. F. O/water in Oil Turbine Power Stations, M. Iqbal
Choudhary and K. M. Khan, Pakistan Patent Application No. 213/92, dated
10/5/1992.
39. Pesticidal composition based on neem, B.S. Siddiqui, N. H. Naqvi, and Shaheen
Faizi, Pakistan Patent SI No. 133662, 1995.
40. A processes for preparation of new cytotoxic composition from Nerium oleander,
Bina S. Siddiqui and Sabira Begum, Serial number # 133661. The Patent Office
Govt. of Pakistan, (1995).
41. Plant-Based Anti-diarrhoeal Drug and Abdominal Pain Reliever, M. Iqbal,
Choudhary, Pakistan Patent Application No. 236/92, dated 18/5/1992.
42. Demulsification of B. F. O/water in Oil Turbine Power Stations, M. Iqbal
Choudhary and K. M. Khan, Pakistan Patent Application No. 213/92, dated
10/5/1992.
43. Saeed SA. (Miles Laboratories, Inc.), USA."Apparatus for Large Scale Gel
Electrophoresis" British Patent No. 1, 359, 944 (1974). French Patent No. 2, 192,
857 (1974). German Patent legungsschrift No. 2, 336, 414 (1974).
44. Salimuzzaman Siddiqui and Viqar Uddin Ahmad - A process for the production
of mononitroajmaline; Pakistan Patent No. 122593 dated 4-2-1972.
45. Salimuzzaman Siddiqui and Viqar Uddin Ahmad - Improvement in and with
relation to the production of C-nitrosoajmaline; Pakistan Patent No. 122840 dated
25-1-1972.