Hepatitis Update 2013 Brendan M. McGuire, MD UAB Liver Center Introduction • Hepatitis - Inflammation of the liver • Five types – – – – – A B C D E Characteristics of Hepatitis Viruses Virus Genome Family Major mode of Chronicity Transmission Fecal - oral No HAV RNA Picornavirus HBV DNA Hepadnavirus Blood Yes HCV RNA Flaviviridae Blood Yes HDV RNA Satellite Blood Yes HEV RNA Caliciviridae? Fecal - oral No 14 Hepatitis A 12 10 8 6 4 Hepatitis B Hepatitis C 2 2000 1998 1996 1994 1992 1990 1988 1986 1984 0 1982 Cases / 100,000 population US Incidence of Reported Cases of Acute Viral Hepatitis, 1982-2001 16 Mortality Rate for acute hepatitis is approximately 0.2% US Esimates of Acute & Chronic Disease Burden for Viral Hepatitis HAV HBV HCV New Infections 25,000 43,000 17,000 Chronic Infections 0 1.2 million 3.2 million Chronic liver disease deaths/year 0 3,000 12,000 Based on CDC estimated annual incidence 2007 Hepatitis A • • • • Usually a self-limiting disease Severity of illness increases with age Transmission is fecal-oral Rarely transmitted by blood to blood transfer • Incubation period is about 28 days • Diagnosis by anti-HAV IgM http://ocw.jhsph.edu/imageLibrary Geographic Distribution of HAV Infection Symptoms & Signs of HAV Infection • Some persons, particularly young children, are asymptomatic. • When symptoms are present, can include: – Constitutional: fever, fatigue & joint pain – Gastrointestinal: loss of appetite, nausea & emesis – Hyperbilirubinemia: jaundice, dark urine & claycolored bowel movements Concentration of HAV in Various Body Fluids Body Fluids Feces Serum Saliva Urine 100 102 104 106 108 1010 Infectious Doses per mL Viral Hepatitis and Liver Disease 1984;9-22 J Infect Dis 1989;160:887-890 Risk Factors Associated with Reported HAV in the US (1990-2000) Source: National Notifiable Diseases Surveillance System Unknown 45% Personal contact 14% IVD use 6% Food/waterborne outbreaks 4% International travel 5% Other 8% Daycare centers 8% Men who have sex with men 10% Sequence of Serologic Changes in Acute HAV Relative Concentration Jaundice Symptoms ALT HAV Stool Anti-HAV Anti-HAV IgG Anti-HAV IgM Viremia TIME Persons at Risk for Acquiring HAV • Travelers to regions with intermediate or high rates of HAV • Sex contacts of infected persons • Household members or caregivers of infected persons • Injection & non-injection illegal drug users • Persons working with nonhuman primates susceptible to HAV infection Prevention of HAV • Hygiene – Hand washing • Sanitation – Clean water source • Immune globulin – Pre-exposure – Post-exposure • Hepatitis A vaccine HAV Prevention Immune Globulin • Pre-exposure – Travelers to intermediate & high HAVendemic regions without enough time for HAV vaccine • Post-exposure (within 14 days) – Household & other intimate contacts – Selected situations in institutions & common source exposure HAV Vaccine • Two single-antigen vaccines are available (HAVRIX® & VAQTA®) • A combination vaccine, TWINRIX®, contains both HAV & HBV antigens • All are inactivated vaccines • Schedule is 0 and 6 months • Not recommended for children < 1 years old Persons Currently Considered to Have an Indication for HAV Vaccine by ACIP • All children ages 12-23 months • Travelers to countries with intermediate & high rates of disease • Individuals who engage in high risk behaviors – Homosexual activities – Intravenous drug use • Chronic liver disease • Individuals with occupational risk of disease – Primate handlers Advisory Committee on Immunization Practices (ACIP) Recommendations 2006 Advisory Committee on Immunization Practices = ACIP Hepatitis B Virus (HBV) • DNA virus • Worldwide: 350 million infected & 620,000 die annually from HBV-related liver disease • 1.2 million persons in the US with chronic HBV infection • Incubation period is 120 days • Causes acute & chronic disease http:ocw.jhsph.edu/imageLibrary www.cdc.org Prevalence of Chronic HBV Infection www.cdc.org Symptoms & Signs of HBV Infection • Most children < 5 years old are asymptomatic. • 30-50% of persons > 5 years of age have signs & symptoms. • Symptoms when present can include: – Constitutional: fever, fatigue & joint pain – Gastrointestinal: loss of appetite, nausea & emesis – Hyperbilirubinemia: jaundice, dark urine & claycolored bowel movements – Decompensated cirrhosis Concentration of HBV in Body Fluids High Blood Serum Wound exudate Moderate Semen Vaginal fluid Saliva Low/not detectable Urine Feces Sweat Tears Breast milk Reported Risk Factors for Acute HBV in the US (1990-2000) Heterosexual activity 45% Men who have sex with men 13% Other 6% IVD use 21% Other include household contact, institutionalization, hemodialysis, blood transfusion, occupational exposure Unknown 15% Source: CDC Natural History of HBV in Infants Acute HBV infection 5% 95% Recovery and immunity Chronic HBV Replication High Low Progressive liver injury Fibrosis and cirrhosis Asymptomatic infection Hepatocellular carcinoma Natural History of HBV in Adults Acute HBV infection 95% 5% Recovery and immunity Chronic HBV Replication High Low Progressive liver injury Fibrosis and cirrhosis Asymptomatic infection Hepatocellular carcinoma Cellular Immune Responses to HBV NEJM 2004;350:1118 Acute HBV with Recovery Symptoms HBeAg anti-HBe Total anti-HBc Titer HBsAg 0 4 8 IgM anti-HBc 12 16 20 24 28 32 36 Weeks after Exposure anti-HBs 52 100 Serological Markers of Acute HBV Infection Clinical Significance HBsAg HBsAb Early + - Window - Recovery + HBeAg + - - HBeAb - + + HBcAb IgM + + - HBcAb IgG HBV DNA +++ - + - Progression to Chronic HBV Infection Acute (6 months) Chronic (Years) HBeAg anti-HBe HBsAg Titer Total anti-HBc IgM anti-HBc 0 4 8 12 16 20 24 28 32 36 52 Weeks after Exposure Years Chronic HBV Disease Types • HBeAg positive – Also known as “wild type” – Antibody to HBeAg is negative – HBV DNA > 20,000 IU/mL (> 105 copies/mL) • HBeAg negative – Also known as “precore mutant” – Antibody to HBeAg is positive – HBV DNA > 2000 IU/mL (> 104 copies/mL) Keeffe EB, et al. Clin Gastroenterol Hepatol. 2004;2:87-106. Chu CJ, et al. Gastroenterology. 2003;125:444-451. 4 Phases of Chronic HBV Current Understanding of HBV Infection HBeAg Anti-HBeAg ALT activity HBV DNA Phase Liver Immune Tolerant Immune Clearance Inactive Carrier State Minimal inflammation and fibrosis Chronic active inflammation Mild hepatitis and minimal fibrosis Yim HJ, et al. Hepatology. 2006;43:S173-S181. Reactivation Active inflammation Optimal treatment times Hepatitis B Viral (HBV) Markers Laboratory Results HBsAg + HBsAb + HBeAg + HBeAb + Comments HBcAb IgM + HBcAb IgG + HBV DNA + Acute or prior exposure Prior exposure Active viral replication Active viral replication Prior exposure or immunity Active viral replication Acute or prior exposure or chronic infection Markers of Chronic HBV Infection Clinical Significance Phase Replicative Low, Flare of or nonreplicative, chronic HBV or inactive Reactivation carrier Precore/core promotor mutants HBsAg HBsAb + - + - + - + - HBeAg + +/- +/- - HBeAb - -/+ -/+ + HBcAb IgM - - +/- - HBcAb IgG HBV DNA + +++ + +/- -/+ ++ + + The Replication Cycle of HBV NEJM 2004;350:1118 Therapeutic Approaches to HBV • Interferon • Nucleoside analogues – Lamivudine & Entecavir • Nucloetide analogues – Adefovir & Tenofovir • Monoclonal antibody to HBsAg • Vaccination for prevention Hepatitis B Immune Globulin (HBIG) • Prepared from plasma containing high titers of antibody to HBsAg • Used for post-exposure prophylaxis to prevent infection from: – Perinatal – Sexual – Occupational • Must be given within 2 weeks of exposure to be effective • Confers no protection against future exposure Hepatitis B Vaccine • Became available in 1981. • All are produced with yeast & recombinant techniques to generate the HBsAg protein. • Advisory Committee on Immunization Practices recommended universal vaccinations of – All infants, in 1991. – All adolescents, in 1995. – All persons up to age 18, in 1999. Adults Considered to Have an Indication for HBV Vaccine By ACIP • • • • • • • • • • Sexual or household contacts of people infected with HBV Multiple sexual partners IVD user Job that involves contact with blood or blood products Prisoner in a correctional facility Residents/staff in institutions for the developmentally disabled Travelers to countries with high rates of HBV HIV positive Chronic liver disease, renal failure or dialysis Unvaccinated adults with diabetes ages 19 - 59 years HCV: RNA Genomic Organization 0 3000 6000 9000 NEJM 2001;345:41 Hepatitis C Virus (HCV) • RNA virus • 17,000 cases new annually in the US (2007) • Approximately 12,000 deaths each year in the US secondary to chronic HCV www.cdc.org Identifying Estimated 170 Million Persons With HCV Infection Worldwide Americas 13.1 million (1.7%) Europe 8.9 million (1.03%) Africa 31.9 million (5.3%) W Pacific 62.2 million (3.9%) SE Asia E Mediterranean 32.3 million (2.15%) 21.3 million (4.6%) World Health Organization (WHO). Wkly Epid Rec .1999;74:425-427. WHO. Hepatitis C: Global Prevalence: Update. 2003. Farci P, et al. Semin Liver Dis. 2000;20:103-126. Wasley A, et al. Semin Liver Dis. 2000;20:1-16. Prevalence of Chronic HCV Infection In the US, 2.7–4 million people are living with chronic HCV infection; 75% are unaware they are infected CDC & Prevention. HCV. Available at: http://www.cdc.gov/hepatitis/HCV/HCVfaq.htm. Accessed June 26, 2011. Institute of Medicine. Hepatitis & Liver Cancer: A National Strategy for Prevention & Control of Hepatitis B & C; 2010. Epidemiology of HCV in the US • 2.7-4 M Americans infected (2%) • High prevalence rates – 2.5% of males – 3.2% of African Americans – 2.1% of Hispanic Americans – People born between 1946 - 1964 Two-Thirds of Those With Chronic HCV in the U.S. Were Born Between 1946 & 1964 Individuals (n) Estimated Prevalence by Age Group 1.6M 1.4M 1.2M 1M 800k 600k 400k 200K 0 <1920 19201929 19301939 19401949 19501959 19601969 1970- 19801979 1989 1990+ Birth Year Group Pyenson B, et al. Consequences of Hepatitis C Virus (HCV): Costs of a Baby Boomer Epidemic of Liver Disease. New York, NY: Milliman, Inc; 2009. Natural History of HCV Infection A cute H C V Infection (100) R ecov ery & C learance of H C V (20) M ild (24) C hronic H epatitis C hronic Infection (8 0 ) M oderate (32) S ev ere (24) C irrhosis E nd-S tage Liv er D isease H epatocellular CA Clin Liver Dis 2005;9:383-398. Eur J Gastroenterol Hepatol 1996;8:324-328. Hepatology 2002;36(suppl):S1-S2. Hepatology 2002;36(suppl):S35-S46. Ann Intern Med 2000;132:296-305. Gastroenterology 1997;112:463-472. Immunopathogenesis of HCV CD4 T-Helper Cells HCV Antigen APC MHC Class II TCR/CD3 CD-4 Th1 IL-12 INF-g Th0 IL-4 Th3 TGF-b, IL-10 Th2 IL-2, TNF-a/b, IFN-g IL-4, IL-6, IL-6, IL-10 Greater Immunopathology Lesser Immunopathology Number of cases Projected Cases of Hepatocellular Carcinoma & Decompensated Cirrhosis Due to HCV 160,000 140,000 120,000 Decompensated 100,000 cirrhosis 80,000 60,000 40,000 Hepatocellular cancer 20,000 0 1950 1960 1970 1980 1990 2000 2010 2020 2030 Year Gastroenterology 2010;138:513-521 Patient Survival Rates with HCV (+) & HCV (–) After Liver Transplantation HCV (+) 4439 HCV (-) 6597 3035 4784 1951 3343 1134 2117 519 98 1003 220 Gastro 2002;122(4):889. Risk Factors for HCV • Transfusion of blood or blood products before 1992 • Intravenous drug use • Intranasal cocaine • Hemodialysis • High-risk sexual contact • Tattooing or body piercing • Occupational exposure to blood or blood products • An organ, graft, or tissue transplant from an HCV+ donor Reported Risk Factors for Acute HCV in the US, 2007 • • • • • Injection drug use – 48% Multiple sex partners – 42% Men who have sex with men – 10% Sex with someone known to have HCV -10% Risk factors are not mutually exclusive Low Risk of HCV Transmission Between Monogamous Sexual Partners • 776 serodiscordant spouses followed for 10 yrs – Intercourse mean: 1.8/wk – No condom use, no anal sex – 3 new infections (incidence 0.37/1000 pt-yrs), but all 3 differed from partner’s strain – Net incidence of transmission: 0 Vandelli C, et al. Am J Gastroenterol. 2004;99:855-859 Counseling HCV Patients • Potentially infectious • Keep cuts and skin lesions covered • Potential for sexual transmission • Potential for perinatal transmission – no evidence to advise against pregnancy or breastfeeding • Should not • Donate blood, organs, tissue, or semen • Share household articles (e.g., toothbrushes, razors) Typical Course for Resolution of Acute HCV Symptoms Titer anti-HCV Normal 0 1 2 3 Months 4 5 6 1 2 3 4 ALT HCV RNA Years Time after exposure Hepatology. 2002;36:S65-S73. Typical Course for Chronic HCV Infection HCV RNA Symptoms Titer anti-HCV ALT Normal 0 1 2 3 Months 4 5 6 1 2 3 4 Years Time after exposure Hepatology. 2002;36:S65-S73. Enzyme Immunoassay (EIA) anti-HCV • Main screening test • Detects circulating antibodies – 2 months after exposure • Advantages are ease of use, low variability, ease of automation & relatively low expense • Sensitivity is 97-100% • Positive predictive value varies on prevalence – 95% with risk factors & elevated ALT – 50% without risk factors & normal ALT Quantitative HCV RNA by PCR • Important for measuring the level of circulating HCV RNA (viral load) • Diagnosis within 1 to 2 weeks after exposure • Evaluation of patients with false positive EIA • Diagnosis of patients who fail to develop antibodies • Detection limit > 12 IU/ml Hepatology. 2009;49:1335-1374. False Negative Molecular Tests • Ribonucleases are ubiquitous & makes RNA inherently unstable • Serum specimens should be separated from whole blood < 4 hours of venipuncture • Rapid storage of serum specimens at -70 oC • Minimal freezing & thawing Nucleic Acid Testing For HCV • Allows very small amounts of RNA to be detected by a process of massive copying of a gene fragment. • A rapid test to determine RNA in the blood. • Can identify RNA in the blood 12 days after exposure. • Used by organ and blood banks for identifying acute cases of HCV from donors. Transfusion 2010; 50:1495–1504 Prevalence of HCV Genotypes & Subtypes in the USA 1&2 3 4 2b 2a 1a & 1b 1b (39%) 1a (36%) Patterns of Virologic Response PegIFN alfa & RBV HCV RNA (log10 IU/mL) 7 Null Response* 6 5 Partial Response* 4 3 Relapse 2 1 Undetectable 0 -8 -4 -2 0 *Subset of Nonresponse RVR 4 EVR 8 12 ETR 16 20 24 32 40 48 SVR 52 60 72 Wks After Start of Therapy 4 weeks - RVR: rapid virological response 12 weeks - eRVR: extended RVR & EVR: early virological response 24 - 48 weeks - ETR: end of treatment response 24 weeks after treatment - SVR: sustained virological response Hepatology 2009;49:1335-1374. Treatment Evolution of HCV Sustained Viral Response (SVR) 100 1999 1991 2001 2002 2011 70-80% 80 54-56% 60 40 34% 42% 39% 16% 20 6% 0 IFN 6m IFN 12m IFN/RBV 6m IFN/RBV 12m Peg-IFN 12m Peg-IFN/ RBV 12m Peg-IFN/ RBV + PI 6-12m IFN: Interferon; m: months; RBV: Ribavirin; Peg: Pegylated; PI: Protease inhibitor Adapted from Strader DB et al. Hepatology 2004;39:1147-1171 Guidelines for HCV Testing: Acute Infection Suspected • Baseline HCV Ab • 4-6 weeks - HCV antibody & HCV RNA • 2-3 months – HCV RNA – If positive, consider treatment • 4-6 months - HCV antibody & HCV RNA JAMA. 2007;297:724-732. Spontaneous Clearance for Symptomatic Acute HCV High, Justifies Treatment Delay • 60 patients with acute HCV (36 genotype 1) followed[1] – Spontaneous clearance in 52% of 51 symptomatic cases • No asymptomatic patient cleared virus spontaneously – SVR achieved in 81% of symptomatic patients without spontaneous clearance who were treated > 3 mos after symptom onset with IFN ± RBV • Recent study showed similar SVR rates in symptomatic adherent patients who delayed therapy for 12 wks vs those who received immediate treatment[2] 1. Gerlach JT, et al. Gastroenterol. 2003;125:80-88. 2. Deterding K, et al. EASL 2009. Abstract 1047. Randomized Trial of Treatment for Acute HCV at Variable Times After Onset – 37% genotype 1 – 41% genotype 4 • Randomized to treatment at Wk 8, 12, or 20 • Treatment with pegIFN alfa2b 1.5 µg/kg/wk x 12 wks 100 95* 92 76 80 SVR (%) • 129 patients entered treatment for lack of spontaneous clearance within 8 wks of presentation 60 40 20 0 43 43 43 8 wks 12 wks 20 wks Time of Treatment Initiation *SVR rates significantly higher for genotype 1 patients who received treatment after 8 wks vs either 12 or 20 wks (P = .01 and P = .004, respectively). Gastroenterol. 2006;130:632-638. Acute HCV Infection: Summary of Recommendations • Patients with acute HCV infection should be considered for IFN-based therapy (either standard or pegIFN). • Treatment can be delayed 8-12 weeks after acute onset to allow for spontaneous resolution • No definitive recommendation about optimal duration of treatment for acute HCV; however, it is reasonable to treat for ≥ 12 weeks, & 24 weeks may be considered • Decision to use RBV made on a case-by-case basis Ghany MG, et al. Hepatology. 2009;49:1335-1374.