HYGIA INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH,
Faizullahganj, Prabhandh Nagar, Ghaila Road, Lucknow-226020 (U.P)
Subject Name
Subject Code
Semester
Subject Teacher Name
No of Lectures
:
S.No
1.
Unit
2.
4.
5.
6.
7.
8.
9.
10.
11.
12.
13.
14.
15.
Unit-I
Antihistaminic agents, Gastric proton-pump inhibitors,
Anti-neoplastic agents
3.
LECTURE PLAN
MEDICINAL CHEMISTRY – II
BP501T
V
Rajni Devi
Approx 56
Topic
Basic introduction and syllabus of medicinal
chemistry.
Histamine, receptors and their distribution in
the human body.
H1–antagonist: Diphenhydramine
hydrochloride*, Dimenhydrinate, Doxylamine
succinate,
Clemastine fumarate, Diphenylpyraline
hydrochloride, Triphelenamine
hydrochloride, Chlorcyclizine hydrochloride,
Meclizine hydrochloride, Buclizine
hydrochloride,
Chlorpheniramine maleate, Triprolidine
hydrochloride*, Phenidamine tartrate,
Promethazine hydrochloride*,
Trimeprazine tartrate, Cyproheptadine
hydrochloride, Azatidine maleate,
Astemizole, Loratadine, Cetirizine,
Levocetrizine, Cromolyn sodium.
H2-antagonists: Cimetidine*, Famotidine,
Ranitidine. Gastric proton-pump inhibitors:
Omeprazole, Lansoprazole, Rabeprazole,
Pantoprazole.
Alkylating agents: Meclorethamine*,
Cyclophosphamide, Melphalan,
Chlorambucil, Busulfan, Thiotepa.
Antimetabolites: Mercaptopurine*,
Thioguanine, Fluorouracil, Floxuridine,
Cytarabine, Methotrexate*, Azathioprine.
Antibiotics: Dactinomycin, Daunorubicin,
Doxorubicin, Bleomycin.
Plant products: Etoposide, Vinblastine
sulphate, Vincristine sulphate.
Miscellaneous: Cisplatin, Mitotane.
Anti-anginal: Vasodilators: Amyl Nitrite,
Nitroglycerin*,
Pentaerythritol tetranitrate,
Isosorbide dinitrite*, Dipyridamole.
Calcium channel blockers: Verapamil,
Bepridil hydrochloride, Diltiazem
Date
20/09/2021
Day
Monday
21/09/2021
Tuesday
22/09/2021
Wednesday
23/09/2021
Thursday
24/09/2021
Friday
27/09/2021
Monday
28/09/2021
Tuesday
29/09/2021
Wednesday
30/09/2021
Thursday
01/10/2021
Friday
04/10/2021
Monday
05/10/2021
06/10/2021
Tuesday
Wednesday
07/10/2021
Thursday
08/10/2021
Friday
Remark
hydrochloride,
16.
19.
20.
21.
22.
23.
24.
25.
26.
27.
28.
29.
30.
31.
32.
33.
34.
35.
Unit-III
Anti-arrhythmic Drugs, Anti-hyperlipidemic
agents, Coagulant & Anticoagulants, Drugs used
in Congestive Heart Failure
18.
Unit-II
Anti-anginal, Diuretics, Anti-hypertensive
Agents
17.
36.
37. Unit-IV
38.
Drugs
acting on
Nifedipine, Amlodipine, Felodipine,
Nicardipine, Nimodipine.
Diuretics: Carbonic Anhydrase Inhibitors:
09/10/2021
Saturday
11/10/2021
Monday
Acetazolamide*, Methazolamide,
Dichlorphenamide.
Thiazides: Chlorthiazide*,
Hydrochlorothiazide, Hydroflumethiazide,
Cyclothiazide,
12/10/2021
Tuesday
13/10/2021
Wednesday
Loop Diuretics: Furosemide*, Bumetanide,
Ethacrynic acid.
Potassium sparing Diuretics: Spironolactone,
Triamterene, Amiloride. Osmotic Diuretics:
Mannitol.
Anti-hypertensive Agents: Timolol,
Captopril, Lisinopril, Enalapril, Benazepril
hydrochloride,
Quinapril Hydrochloride, Methyldopate
Hydrochloride* Clonidine hydrochloride,
Guanethidine Monosulphate, Guanabenz
Acetate, Sodium Nitroprusside,
Diazoxide, Minoxidil, Reserpine, Hydralazine
hydrochloride.
Anti-arrhythmic Drugs
18/10/2021
Monday
20/10/2021
Wednesday
21/10/2021
Thursday
22/10/2021
Friday
23/10/2021
Saturday
25/10/2021
Monday
26/10/2021
Tuesday
Quinidine Sulphate, Procainamide
Hydrochloride,
Disopyramide
Phosphate*, Phenytoin Sodium,
Lidocaine Hydrochloride, Tocainide
Hydrochloride,
Mexiletine Hydrochloride,
Lorcainide Hydrochloride, Amiodarone,
Sotalol.
Anti-hyperlipidemic agents: Clofibrate,
01/11/2021
Monday
02/11/2021
Tuesday
03/11/2021
Wednesday
08/11/2021
Monday
09/11/2021
Tuesday
Lovastatin, Cholestyramine and Colestipol.
10/11/2021
Wednesday
Coagulant & Anticoagulants: Menadione,
11/11/2021
Thursday
Acetomenadione, Warfarin*, Anisindione,
Clopidogrel.
Drugs used in Congestive Heart Failure
12/11/2021
Friday
13/11/2021
Saturday
Digoxin, Digitoxin, Nesiritide, Bosentan,
Tezosentan.
Drugs acting on Endocrine system
15/11/2021
Monday
16/11/2021
Tuesday
Nomenclature, Stereochemistry and
metabolism of steroids.
Sex hormones: Testosterone, Andralone,
17/11/2021
Wednesday
18/11/2021
Thursday
39. Endocrine
40.
41.
42.
43.
44.
45.
system,
Sex
hormones,
Oral
contracept
ives,
Corticoste
roids,
Thyroid
and
antithyroi
d drugs
47.
48.
49.
50.
51.
52.
53.
54.
Unit-V
Antidiabetic agents, Local Anesthetics
46.
Progestrones, Oestriol, Oestradiol, Oestrione,
Diethyl Stilbestrol.
Drugs for erectile dysfunction: Sildenafil,
Tadalafil.
Oral contraceptives: Mifepristone,
Norgestrel, Levonorgestrel
Corticosteroids: Cortisone, Hydrocortisone,
22/11/2021
Monday
23/11/2021
Tuesday
25/11/2021
Thursday
26/11/2021
Friday
Prednisolone, Betamethasone,
Dexamethasone.
Thyroid and antithyroid drugs:
27/11/2021
Saturday
29/11/2021
Monday
L-Thyroxine, L-Thyronine, Propylthiouracil,
Methimazole.
30/11/2021
Tuesday
Antidiabetic agents: Insulin and its
preparations.
Sulfonylureas: Tolbutamide*,
Chlorpropamide, Glipizide, Glimepiride.
Biguanides: Metformin.
Thiazolidinediones: Pioglitazone,
Rosiglitazone, Meglitinides
Repaglinide, Nateglinide.
Glucosidase inhibitors: Acarbose, Voglibose.
Local Anesthetics: SAR of Local anesthetics.
Benzoic acid derivatives; Cocaine,
Hexylcaine,
Meprylcaine, Cyclomethycaine, Piperocaine.
Amino Benzoic acid derivatives:Benzocaine*,
Butamben, Procaine*, Butacaine,
Propoxycaine, Tetracaine, Benoxinate.
Lidocaine/Anilide derivatives: Lignocaine,
Mepivacaine, Prilocaine, Etidocaine.
Miscellaneous: Phenacaine, Diperodon,
Dibucaine.
01/12/2021
Wednesday
02/12/2021
Thursday
03/12/2021
Friday
06/12/2021
Monday
07/12/2021
Tuesday
08/12/2021
Wednesday
09/12/2021
Thursday
10/12/2021
Friday
11/12/2021
Saturday