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Drugs Used - D&A

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NALTREXONE Revia Vivint
usedto manage alcohol
ROA
RO
opioid antagonist
opioid dependence
by decreasing desire
most common
50mg tablet
In depot injection
SC implants
acute hepatitis
contraindicating
recent opioid use
sideeffects
a
or
liverfailure
710 days
diarrhea
wish at
vethdrand
on abdominalcramping
MOA
foropioiddependence
foralcoholdependence
blocks opioid receptors to attenuate
the effects ofopioids
blocking
KOR blocks actionof
endogenousopioid dynophir
instatesdrug seehing behaviour
SINCLAIR METHOD
continued
consumption
of alcohol in combination
with
naltrexone
naltrexone blocks action of endorphins which would provide
rounding experience when driving
i over time
cravings
brain learns to cut associate aleowd with pleasure
Tanth over alcohol
use
ACAMPROSATE
used withcounselling
ROA PO
psychosocial support
a
suicidalbehaviour
majordepressive
disorder
anxiety
Eton bindsto GABAA R
I EfOH
vomiting
depression
diarrhea
i
to treatalcoholdependence
nausea
kidney failure
MOA
positiveallostericmandafffter
hidacy damage
contraindications
sideeffects
NMDA R antagonist
CCampral
tolerance
desensitised GABA
R
physical withdraw sincenondGABAhas no effect
iGABAnormally inhibity
CABA
R desensitization
acamprosate enhances GABAsignalling
overexatation
as positive allostericmodulator
Etonusuallyinhibits NMDAR activity
chronic Eton consumption upregulates NMDA R
i HEINI canes Rautinty of excess NMDARs
withdrawals
withdrawal
glutarde surge whitefumeaetiaks NMDARs
s aeanprosate
decreases
glutante surge as NMDA R antagonist
at
DISULFIRAM
used
poA
acetaldehyde
Antabuse
as secondline drugforalcoholism
dehydrogenase inhibitor
by Asensitivity to alcohol
doesnottramings a compliance bad
poor
8D implant
contraindications
liver problems
recentalcohol use
sideeffects
with alcohol
02hours
common severe hangover symptoms
dyspnea
visualdisturbance
housed
confusion
vomiting
posturalsyncope
headache
without alcohol
to
circulatory collapse
headache
metallicgarlictaste in mouth
dlibido
linerproblems
Shih rush
neuropathy
MOA
disulfiram
1
alcohol
alcohol
dehydrogenase
acetaldehyde
i
Tautaldehyde
acetaldehyde
dehydrogenase
acetyl
coff
hangoversymptoms
DIAZEPAM
Valium
benzodiazepine
usedfor a variety of conditions including alohdwithdrawalsyndrome
ROA P O
PR
nasalspray
M
w
contraindications
side effects
ataxia
depression
hyperventilation
psychosis
liverproblems
pregnancy
kidney problems
sleepapnea
sedation
bronchitis
breastfeeding
copD
confusion
anterograde amnesia
MOA
myastheniagravis
a
ataxia
benzodiazepines are positive allosteric modulator of GABA R
AAAAA R
are
ligandgated d selective channels which when
activatedby GABA
i
Iv activity
Tirflax of Cl
hypepolarisation
of cortical andlimbic systems in CNS
Other benzos
chlordiazepoxide Clibrium alertedwithdrawal
Miran
diazepam lorazepam alcoholwithdnt in elderly and cirrhosis cases
alprazolam'Cxanax
bromazepan anxiety insomnia
clonazepam Cklonopin
seizures
non selective opioidreceptorantagonist
NALOXONE Narcan
used to blockthe effects of opioids
ROA
endotracheal
In
nasalspray
10
Cerg to increasebreathing
homespray
take
reverse OD
to
IV
contraindications
in opioidOD
new
available
heartconditions
hypersensitivity
sideeffects
hypotension
hypertension
tachycardia
nausea
seizures
vomiting
MOA
sweating
non selectively
prevents
a
acute opioid withdrawal syndrome
competitively binds
to opioidreceptors
the action ofboth endogenous and exogenous
opiates
BUPRENORPHINE
opioid
Buvidal
used to treat opioid user disorder
ROA
subnet
sublingual fun
pregnant
buccalinjection
as
well
as
transdermal
acute chronic pain
Buidal is depotinjection
weekly or monthly
implant
subcutaneous
IV
contraindications
sideeffects
hypersensitivity
nausea
a
vomiting
a
MOA
acts as
respiratory
dry
amnesia
miosis
perspiration
orthotichypotension
drowsiness
dizziness
mouth
headache
itchiness
depression
urinary retention
a
an opioid receptor modulator
weakpartialagonist of MOR
antagonist of KOR
antagonist of Pop
i
binds with high affinity to mop butonly activates partially
can bloch most nor agonistsand is usefulto treatdependence
NALOXONE CSuboxone
BUPRENORPHINE
combination
used to treat opioid use disorder with counselling
opioid
to
apah
giadgm.net
abusedeterrent
ROA sublingual
a
contraindications
side effects
a
severe respiratory liner impairment
create alcoholism
headaches
hypotension
opioid withdrawal syndrome
vomiting
nausea
pain
increased sweating
Mott
constipation
buprenorphine
acts as
an opioid receptor modulator
weakpartialagonist of MOR
antagonist of KOR
antagonist of pop
binds with high affinity to mop butonly activates partially
can bloch most nor agonistsand is usefulto treatdependence
naloxone
non selectively
prevents
works
as
competitively binds
to opioidreceptors
the action ofboth endogenous and exogenous
an
opiates
abusedeterrent
whentaken sublingually
as prescribed
buprenorphine
elfah
dominate naloxone is negligible dueto low oral absorption
if tries to misuse by
naloxone
acts as an
injection inhalation
antagonit to reduce opioideffects or even precipitate withdrawal
METHADONE Dolophihelmethadose
opioidagonist
NMDA Rantagoni
usedto treatopioid dependenceandchronicpain
post
a
pro mostcommon
II
fM
contraindicating i
a
use of anticonvulsants
use
side effects
a
a
vomiting
abund heat
diarrhea
dizziness
myths due to
prolonged QT
nausea
sleepiness
a
Mott
ofopioidantagonists
a
headache
a
respiratory depressin
sweating
releases neurotransmitter invoked in
paintransmission
opioid agonist
as
inhibits action of excitatory neurotransmitter glutamate
i
decreases development of tolerance to opioids by
disrupting memory pathways
as
NMDAN antagonist
SERTRALINE
antidepressant used to
ROA
selective serotoninreuptakeinhibitorcss.pe
Eleven
treat
Po
contraindications
a
use
of
depression
panicdisorders
OCD PTSD
monoamine oxidase Moto inhibitors
use of antipsychotic pineaide
age of disulfiram
care when prescribing
elderly
or patients
with
liver problems slower elimination
sideeffects
nausea
diarrhea
insomnia
dizziness
MOA
dry mouth
tremor
decreased libido
ejaculation failure
serotonin transporter SERT to inhibit
neuronalreuptake of serotonin and potentiate sentinergie
binds to
activity in the CNS
THIAMINE VITAMIN Bi
usedto that thiaminedeficiency in chromealcoholism alcoholmouse disorde
PO
ROA
1V
MOA
alcohol can damage stomach act lining
4 absorption of vitaminB
deficiency
beriberi
dry
a
wet
ACT
neuropathy
numbness
cardiac TNR
nausea
cerebral
vomiting
tingling hyperreflexia
edema dyspnea
abdominal
heatfailure
pain
Weniches encephalopathy Korsakoff'spsychosis
Wernicke's Korsakoff syndrome
abnormaleye movements
stance and gaitataxia
cognitive inpairments
gabapentinoid anticonvulsant anxiolytic
PREGABALIN Lupica
usedto treat epilepsy neuropathicpain fibromyalgia anxiety seizures
RoA Po
contraindications
a
suicidalthought
heat failure
COPD
kidney failure
side effects
a
weightgain
1cg edema
disturbedvision
sleepiness
a
fatigue
a
dinner
loss of coordination
euphoria
a
Vertigo
MOA
inhibits
i
certain voltage dependent calcium channels
fair
influx
VDCs
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