BIO-DATA OF M.R.YADAV
Name
:
Dr. M. R. Yadav
PERSONAL
Address
:
Official
Faculty of Pharmacy,
The M. S. University of Baroda,
Kalabhavan
Vadodara– 390 001, Gujarat
Date of Birth
E-mail address
Phone No.
:
:
:
Residential
B-1, Kalyan Nagar
(Opp. Anant Park, Near Sabari
School) Vasna Road,
Vadodara-390 015
Gujarat
21st September 1954
msumryadav@gmail.com, mryadav-phar@msubaroda.ac.in
(O): 0265-2434187
FAX: 0265-2418927, 2423898
(M): 09426721112
EDUCATIONAL
Educational Qualifications :
Degree
Institution
Field /Subject(s)
Year
Positions
B. Pharmacy
University of Delhi, Delhi
Pharmacy
1976
IInd Rank
M. Pharmacy
B.H.U., Varanasi
Pharmaceutical Chemistry
1982
Ist Rank
Ph. D.
Panjab University, Chandigarh
Pharmaceutical Chemistry
1986
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PRESENT POSITION
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PROFESSOR & HEAD OF THE DEPARTMENT
Pharmacy Department, Faculty of Technology, Kalabhavan,
The M. S. University of Baroda, Vadodara- 390 001
SPECIAL RECOGNITION
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Organized Graduate Pharmacy Aptitude Test for Pharmacy Graduates [GPAT-2010
Examination (AICTE, New Delhi)] as Co-ordinator, for the FIRST TIME in INDIA.
Organized GPAT-2011 & GPAT-2012 Examinations, an All India level examination
organized under the aegis of AICTE, New Delhi, for Pharmacy Graduates consecutively
for THREE years, wherein about forty five thousand students appeared each year.
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REPRESENTATION IN NATIONAL BODIES
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Member, Scientific Body, National Pharmacopoeia Commission, Ministry of Health &
Family Welfare, Govt. of India
Chairman, Pharmacy Accreditation Evaluation Committee of National Board of
Accreditation, New Delhi for a period of three years from 31st May 2010.
Chairman, National Advisory/Monitoring Committee for GPAT, AICTE, New Delhi from
Nov 2009 –Oct 2011
Coordinator, National Monitoring Committee-GPAT, AICTE, New Delhi from Nov 2010 to
June 2012.
Expert Member, Project Evaluation Committee, UGC, New Delhi
Member, Executive Committee of National Board of Accreditation for empanelment of
Chairpersons/Experts in the field of Pharmacy, NBA, New Delhi
Member National Board of Accreditation (NBA), AICTE, New Delhi from May 2010 for
three years.
Member of South Central Regional Committee, AICTE, Hyderabad, from May 2010 for
three years.
Member of All India Board for Pharmacy Education (AIB-PE), AICTE, New Delhi from June
2006-May 2009.
Member of Sectoral Committee, National Board of Accreditation (NBA) for Management
and Pharmacy, AICTE, New Delhi from Aug 2006-July 2009.
Member, Scientific Services Committee, IPC, from 2004-2006
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AWARDS RECEIVED
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‘UGC-Visiting Fellow Award’ by University Institute of Pharmaceutical Sciences, Panjab
University, Chandigarh, Feb 2015
‘Professor V. M. Kulkarni Visiting Fellow Award in Pharmaceutical Sciences’ by Institute
of Chemical Technology (Autonomous University), Mumbai for the year 2013-14 under
“Professor V. M. Kulkarni Endowment Fund”.
‘Best Teacher of the Year (2013) Award’ in “3rd Annual National Convention of
Pharmacy Professionals” at Faculty of Pharmacy, D.D. University, Nadiad, Gujarat, on 18th
Jan. 2014
‘Pharmacy Teacher of the Year – 2010 Award’ of Association of Pharmacy Teachers of
India
Best Paper prize in oral session of Medicinal Chemistry at 57th IPC, Hyderabad, December
2005
Subhash C. Verma Memorial Prize for Best Research Paper presented in the oral
scientific session of 18th All Gujarat Annual Meeting of Indian Pharmacological Society
held at Anand Pharmacy college, Anand, January 2004
Ranbaxy Laboratories’ Silver Medal in B. Pharmacy at University of Delhi, 1976
EMPLOYMENT
PRESENT POSITION:

DEAN, Pharmacy Faculty of, The M.S. University of Baroda, Vadodara-390 001 From 3rd
December 2015 till date
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PROFESSOR & HEAD, Pharmacy Department, Faculty of Technology and Engineering, The
M.S. University of Baroda, Vadodara-390 001 From 27th February 2010 till date
POSITIONS HELD
ACADEMIC:
1. Professor of Pharmacy (Pharmaceutical Chemistry), Pharmacy Department, Faculty of
Tech. & Engg., Kalabhavan, The M.S. University of Baroda, Vadodara-390 001
 From 1st July 1996 till date
2. Assistant Professor at College of Pharmacy (Currently, DIPSAR, Delhi Institute of
Pharmaceutical Sciences and Research), Government of National Capital Territory of Delhi,
Pushp Vihar, Phase-III, New Delhi-110 017
 From 2nd Feb. 1992 to 30th June 1996
3. Lecturer at Dept. of Pharm. Sciences (Currently, University Institute of Pharmaceutical
Sciences), Panjab University, Chandigarh-160 014
 From 20th November 1985 to 31st January 1992
INDUSTRIAL:
1. Approved Manufacturing Chemist at M/S Tribhavan Injectables, Kirti Nagar Industrial Area,
New Delhi
 From 1st Aug. 1976 to 31st July 1980
ADMINISTRATIVE:
1. Head, Pharmacy Department, Faculty of Tech. & Engg., The M. S. University of Baroda,
Vadodara
 From February 27th 2010 till date.
2. Principal Coordinator, Q.I.P. (Pharmacy), AICTE at Pharmacy Department
 From March 2012 to June 2013.
3. Co-ordinator, Quality Improvement programme in Pharmacy (AICTE), Pharmacy
Department, The M.S. University of Baroda, Vadodara.
 From May 2003 to July 2005
4. Co-ordinator, Centre for Post graduate Studies and Research at Shri G.H. Patel Pharmacy
Building, Pharmacy Department, The M.S. University of Baroda, Vadodara.
 From 1st Aug. 2005 to 31st July 2007
5. Co-ordinator, IPR Cell, The M. S. University of Baroda, Vadodara
6. Head, Department of Pharmaceutical Chemistry, College of Pharmacy (currently DIPSAR)
New Delhi.
 From Jan. 1994 to June 1996
RESEARCH CONTRIBUTION
RESEARCH INTERESTS:
Designing and Synthesis of Medicinal Agents belonging to the following categories:
 Selective COX-II inhibitors
 Steroidal Aromatase inhibitors
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 TACE inhibitors
 Newer anti-hypertensive agents using dual targeted approach
 Protease inhibitors as Antimalarial agents
 Diaryl diazepines as potential anticancer agents
 Development of Non-Nucleoside Reverse Transcriptase Inhibitors
(NNRTI) as antiviral agents
 Preparation of metal complexes of some known antibiotics as H .pylori Inhibitors
 ACAT inhibitors as anti-hyperlipidemic agents
 Virtual screening of chemical databases for anticancer and antimalarial leads
 Computational studies on selective COX-2, Farnesyltransferase, TACE,
integrase, Telomerase Inhibitors
HIV
RESEARCH PROJECTS HANDLED:
1. AICTE-RPS project entitled, “Design and synthesis of peripherally actingCB1 receptor
antagonists as anti-obesity agents”, March 2015 to March 2018, Rs. 10.0 Lacs.
2. “Design and Development of Novel anti-malarial agents”, UGC, New Delhi, Major
Research Project from October 2015 to Septemberr 2018, Rs. 12.53 Lakhs
3. “UGC-BSR One time Grant Scheme” of UGC, New Delhi of Rs. 7.0 Lacs, March 2015.
4. DSA Phase-I program of UGC, New Delhi as Co-ordinator, March 2013 to Feb 2018, Rs. 98
Lakhs
5. “FIST Program of DST on Molecular Modeling”, March 2011, Rs. 48 Lacs, Continuing
from June 2011
6. AICTE-MODROB project entitled, “Evaluation of serotinergic and dopaminergic potential
of some novel ligands”, March 2013 to March 2014, Rs. 15.0 Lacs.
7. “Design and Development of Novel Steroidal Aromatase Inhibitors”, RPS (AICTE) Project
From April 2008 to March 2010, Rs. 19.5 Lacs
8. “Design and Development of New Specific COX-II Inhibitors”, UGC, New Delhi, Major
Research Project from April 2002 to March 2005, Rs. 5.83 Lacs
9. “Development of Protease Inhibitors as Antimalarial Drugs using Computer Aided Drug
Design”, TAPTEC Research Project supported by AICTE, New Delhi
From April 2003 to Mar. 2007, Rs. 14.0 Lacs
10. “Design and Development of New Drugs with Potential Applications in Inflammatory
Disorders”, TAPTEC Research Project supported by AICTE, New Delhi
From April 1998 to Mar. 2000, Rs. 10.0 Lacs
11. “Studies in Neuromuscular Blocking Agents Azasteroids”, UGC (Minor) Research Project
From June 1993 to May 1995, Rs. 38,000/-
ACADEMIC ACHIEVEMENTS:
Research Supervision:
 Ph. D. (Annexure 1)

M. Pharm (Dissertation)
:
:
Awarded
Thesis submitted
Synopsis submitted
Presently Registered
Supervised
Under Guidance
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06
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45
03
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Ph.D. Examiner at Universities:
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Chhatrapati Shahuji Maharaj University, Kanpur
University of Delhi, Delhi
University of Pune, Pune
Panjab University, Chandigarh
Kakatiya Univeristy, Warangal
Hemchandracharya North Gujarat University, Gujarat
Swami Ramanad Teerth Marathwada University, Nanded, Maharashtra
Devi Ahilya Vishwavidyalaya, Indore
Guru Jambheshwar University, Hissar
North Maharashtra University, Jalgoan
Banaras Hindu University, Varanasi
Dr H.S. Gaur Vishwavidyalaya, Sagar
Mumbai University, Mumbai
Rajiv Gandhi Prodyogiki Vishwavidyalaya, Bhopal
Hamdard University (Jamia Hamdard), New Delhi
Bharti Vidyapeeth Deemed University, Pune
Rajasthan University of Health Sciences, Jaipur
Sant Tukadoji Maharaj Nagpur University, Nagpur
Jawaharlal Nehru Technical University, Hyderabad
Nagarjuna University, Guntur
NMIMS University, Mumbai
AFFILIATION TO PROFESSIONAL/ACADEMIC/SCIENTIFIC BODIES
EXPERT MEMBER OF VARIOUS STATUTATIORY BODIES
 Expert member, UGC, New Delhi for evaluation of projects.
 All India Council for Technical Education, New Delhi, for Approval/Renewal of Various
Pharmacy Courses of Colleges throughout India
 Pharmacy Council of India, New Delhi, for Approval/Renewal of Degree/Diploma in
Pharmacy courses as PCI Inspector.
 Expert member of Local Inspection Committee of Gujarat University, Ahmadabad and
Hemchandracharya North Gujarat University, Patan for Affiliation of Colleges to the
concern Universities.
REPRESENTATION IN BOARDS/COMMITTEES OF THE M.S. UNIVERSITY OF BARODA
 Chairman, Screening cum evaluation committee
 Convener, Committee for appointment of dual professor
 Convener, Computer purchase committee
 Convener, Committee for installation of air conditioning system in H.M. Library
 Convener, Workload Committee
 Member, Finance and Establishment Standing Committee The M.S. University of Baroda,
Vadodara since 4th March 2012 till date
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Member, Committee for recommending the names for the appointments for the
Wardens of Halls of Residences, The M.S. University of Baroda, Vadodara since 28th Jan
2015 till date
Member, Standing Committee for monitoring disaster management efforts, The M.S.
University of Baroda, Vadodara
Member, IQAC
Member, RCC, Advisory Committee
Member, Core committee to compile and finalize UGC XII
Member for cases of unfairness committee
Member, Press Supervisory Committee
Member, Medicine Purchase Committee
Member, Advisory Committee for Rashtriya Uchchaatar Siksha Abhiyan (RUSA)
Member, Purchase Committee, The M.S. University of Baroda, Vadodara since 4th March
2012 till date
Member, Unfairmeans Committee
Member Ad-hoc committee for declaration of results, The M.S. University of Baroda,
Vadodara since 4th March 2012 till date
Chairman, Board of Studies (Pharmacy), The M. S. University of Baroda, Vadodara,
2011-14
Chairman, Board of Studies (Pharmacy), The M.S. University of Baroda, Vadodara, 2010
Member, Board of Studies (Pharmacy), The M.S. University of Baroda, Vadodara,
1997 - 2009
UNIVERSITY BOARDS
 Member, Academic Council, Faculty of Pharmacy, Parul University, Vadodara
 Member, Board of Studies in Pharmaceutical Chemistry, Lachoo Memorial College of
Science and Technology (Autonomous), Jodhpur, Rajasthan, 1st July 2012 to 30th June
2014
 Member, Faculty of Pharmacy, Ganpat University, Ganpat Vidyanagar, Kherva, Mehsana,
Gujarat, 1st March 2012 to 7th Jan 2015
 Member, Board of Studies (Pharmacy), Kakatiya University, Warangal, A.P., Jan 2012 to
Dec 2014
 Member, Board of Studies (Pharmacy), Saurashtra University, Rajkot, 2011 onwards
 Member, Board of Studies, Ganpat University, Ganpatnagar, Mehsana, 2009-2012
 Member, Board of Studies (Pharmacy), Devi Ahilya Vishwavidyalaya, Indore, 2010-2013
 Member, Board of Studies, NMIMS, Mumbai, 2007 – 2009
 Member, Subject Area Committee, Nirma University, Ahmedabad
EXPERT MEMBER OF SELECTION COMMITTEES
1. Acted as Expert member of Selection Committee in Subject field Bio-pharmacology for
selection of candidates for the Award of DAAD Fellowship, Ministry of Human Resource
Development, Government of India, New Delhi.
2. Expert Member Selection Committee for the Posts of Professors/Readers/Lecturers at :
 Kakatiya University, Warangal, A.P.
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 Jivaji University, Gwalior, M.P.
 Guru Gobind Singh Indraprashta University, Delhi
 Shri G.S. Institute of Technology and Science, Indore
 Birla Institute of Technology, Ranchi
 NMIMS, School of Pharmacy, Mumbai
 Panjab University, Chandigarh
 Jamia Hamdard (Deemed University), New Delhi
 Sardar Patel University, Vallabh Vidya Nagar
 Gujarat University, Ahmedabad
 J. N. Vyas University, Jodhpur
CHAIRMAN/C0-CHAIRMAN OF SCIENTIFIC SESSIONS
 Chairman in Scientific Session E, Pharmaceutical and Medical Sciences XXVI Gujarat
Science Congress 2012 organized by The M.S.University of Baroda and Gujarat Science
Academy Ahmadabad on 26th Feb 2012.
 Chairperson, two day National conference on ‘Particle technology with special emphasis
on nanotechnology’ organized by Parul Institute of Pharmacy, Vadodara, 22nd-23rd April
2011
 Acted as Chairman, Plenary lecture in IPA Convention 2011, Indore, hosted by IPA M.P.
State Branch, Indore (M.P.) held on 19th & 20th Feb 2011.
 Acted as Chairman of Medicinal Chemistry Session at Indian Pharmaceutical Congress
held at Pune (2002), Chennai (2003), Hyderabad (2005), Mumbai (2006), Varanasi (2007),
New Delhi (2008) and Ahmedabad (2009)
 Acted a Co-Chairman of Medicinal Chemistry section at Indore (1999), Hyderabad (2000)
and New Delhi (2001).
JUDGING OF SCIENTIFIC PRESENTATIONS
 Acted as a Judge for the Scientific Poster Presentation “Radiotracers in Drug
Development”, XXIV Annual Conference of Indian Association of Biomedical Scientists
organised by Institute of Nuclear Medicine and Allied Sciences, DRDO, New Delhi.
ORGANIZING OF SCIENTIFIC/PROFESSIONAL EVENTS
 Organized one day GUJCOST-sponsored National Seminar on “Ethics and plagiarism in
academic research” on 24th August 2015 at Pharmacy Department, Faculty of Tech. &
Engg., The M. S. University of Baroda, Vadodara
 Organized one day UGC-sponsored National Seminar on “Fostering innovation in
pharmaceutical research : Planning to innovation” on 20 th March 2015 at Pharmacy
Department, Faculty of Tech. & Engg., The M. S. University of Baroda, Vadodara
 Organized one week AICTE sponsored QIP on “Spectra based structural insights into
drugs” from 19th to 24th Jan 2015 at Pharmacy Department, Faculty of Tech. & Engg., The
M. S. University of Baroda, Vadodara
 Organized two-days AICTE sponsored National Seminar on “Approached in drug discovery” at
Pharmacy Department, The M. S. University of Baroda., Vadodara, on 26 – 27 Feb 2013.
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Organized UGC sponsored Two days National Seminar on ‘Statistical Analysis in Drug
Development and Discovery’, at Pharmacy Department, The M. S. University of Baroda,
Vadodara, on 20th and 21st Jan 2012
Dy. Co-odinator, National seminar on ‘Neutraceuticals and plants in human health’,
Department of Botany, The M. S. University of Baroda, Vadodara, Dec 10-11, 2011.
Organized one week AICTE sponsored QIP Staff Development Programme on “Glimpses
of Current Advances in The Field of Pharmaceutical Sciences”, at Pharmacy Department,
The M. S. University of Baroda from 2nd - 8th June 2010 as Convener.
Organized two days regional seminar on “Intellectual Property and Innovation
Management in Knowledge Era” held on 26th and 27th August 2009 at The M. S.
University of Baroda, Vadodara as Co-ordinator.
Organised Two weeks ISTE Sponsored Summer School on “Trends in Developments of
Drugs & Delivery Systems-A Futuristic Approach” as Co-ordinator at Pharmacy
Department, The M.S. University of Baroda, Vadodara From 19th to 31st May 1997.
TRAINING PROGRAMMES ATTENDED
 Workshop cum Retreat on “IP Management in Public Private partnership” organized by
INDO-US SCIENCE AND TECHNOLOGY FORUM, TIFAC-DST, Govt. of India at National
Center for biological sciences (NCBS), Bangalore, from February 8-10, 2006
 “Internet Training Programme”, organized by Computer Center, The M.S.University of
Baroda, Vadodara, 11-17th Jan 2000
 “Computer Aided Drug Design’, Summer school organised by National Institute of
Pharmaceutical Education and Research, S.A.S.Nagar, Punjab, 15 -19th June 1998
 ISTE Sponsored Summer School on “Quality Control of Drugs and Pharmaceuticals by
Modern Instruments” organized by L. M. College of Pharmacy, Ahmedabad, 8 -21st May
1995.
 Post Graduate Teachers Workshop in Medicinal & Analytical Chemistry, organized by
K.L.E. College of Pharmacy, Belgaum, 5 -6th June 1993
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UGC/DSA Supported Certificate “Course Course-cum-Workshop on QSAR”, organized by
Department of Chemical Technology, Matunga, Bombay, Feb 6-8, 1992
 ISTE Sponsored course on “Application of Computer Programming in Pharmaceutical
Sciences” organized by L.M.College of Pharmacy, Ahmedabad, 8 -28th May 1988.
EDITORIAL ADVISORY BOARD
 Member, Editorial Review Board, ‘International Journal of Quantitative Structure
Property Relationships (IJQSPR), IGI Global, Hershey, Pennsylvania (USA)
 Member, Editorial Board, ‘International Journal of Pharmaceutical Sciences and
Nanotechnology’, Pharma Book Syndicate, Hyderabad
 Member of Editorial Advisory Board of ‘The Open Drug Discovery Journal’ ISSN: 1877
3818, Bentham Open.
 Member, Advisory Board for Rajeev Gandhi University of Health Sciences Journal of
Pharmaceutical Sciences, Bangalore
JOURNAL REFEREE
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Bio-organic Medicinal Chemistry (Science Direct)
European Journal of Medicinal Chemistry (Science Direct)
Journal of Molecular Structure (Science Direct)
Immunology and Cell Biology (Nature Publishing Group)
Computer-Aided Molecular Design (Springer Link)
Journal of Heterocyclic Chemistry (Wiley Interscience)
Chemical Biology and Drug Design (Wiley Interscience)
Molecular Informatics (Wiley Interscience)
Current Medicinal Chemistry (Bentham Science)
Medicinal Chemistry (Bentham Science)
Medicinal Chemistry Research (Bentham Science)
Letters in Drug Design and Discovery (Bentham Science)
Mini Reviews in Medicinal Chemistry (Bentham Science)
PROFESSIONAL BODIES
 IPA Vadodara Branch: President since June 2012 for four years.
 Life Member of:
 Society of Pharmaceutical Education and Research (SPER/LM/GU/009)
 Indian Society of Technical Education (LM-4312)
 Indian Pharmaceutical Association (DEL/LM/101)
 India Pharmacy Graduate Association (LM-363)
 Indian Pharmacological Society (GULM-519)
 Association of Pharmacy Teachers of India (GU/LM-060)
SPECIAL LECTURE/TALK DELIVERED ABROAD AS RESOURCE PERSON
1. Scientific talk entitled, ‘Dual α1- and AT-1 inhibitors as potential antihypertensive agents’
delivered in Indo-Russian Seminar at National Medical University, Volgograd, Russia held
during 8th to 10th Sept 2011
SPECIAL LECTURES/TALKS DELIVERED AS RESOURCE PERSON (NATIONAL)
1. Invited talk entitled, “Concept & applications of molecular modeling” in 10th National
conference on Thermodynamics of pharmaceutical, chemical and biological systems, under
the aegis of The thermodynamics society at UIPS & Department of Chemistry, PU,
Chandigarh on 20th Nov 2015 held during 2o -21 November 2015.
2. Resource person in the awareness program on “Intellectual property rights (IPR”) 19 th
September 2015, conducted by Research and Consultancy Cell, The M. S. University of
Baroda, Vadodara
3. Invited talk entitled, “Design and development of some α1- and AII-blocking dual inhibitors
as potential antihypertensive drugs” in UGC Networking Resource Centre at UIPS, on
“Contemporary trends in the realm of medicinal chemistry ” on 14th Sept 2015 at University
Institute of Pharmaceutical Sciences, Panjab University, Chandigarh, held during 14 th to 19th
September 2015.
4. Invited talk entitled, “Fundamentals of NMR spectroscopy” in one day GUJCOST-sponsored
National Seminar and workshop on “Structural characterisation of organic compounds by
spectroscopy” on 11th Sept 2015 at L. M .College of Pharmacy, Ahemedabad, held during 11th
and 12th September 2015.
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5. Invited talk entitled, “Ethics and morality in academic research” in one day GUJCOSTsponsored National Seminar on “Ethics and plagiarism in academic research” on 24th August
2015 at Pharmacy Department, Faculty of Tech. & Engg., The M. S. University of Baroda,
Vadodara
6. Invited talk entitled, “Plagiarism and scientific misconduct” in one day Seminar on
“Plagiarism and Intellectual property rights laws” on 16th May 2015 at Sumandeep
Vidyapeeth (Deemed University), Vadodara
7. Invited talk entitled, “Changing paradigms in drug discovery” in one day UGC-sponsored
National Seminar on “Fostering innovation in pharmaceutical research : Planning to
innovation” on 20th March 2015 at Pharmacy Department, Faculty of Tech. & Engg., The M.
S. University of Baroda, Vadodara
8. Invited talk entitled, “Changing paradigms in drug discovery” on 1st March 2015 at DST-ICMR
sponsored National Seminar on “Emerging frontiers and challenges in nanotechnology and
drug design” at Department of Pharmaceutical Sciences, Dr H. S. Gour Vishwavidyalaya,
Sagar, M. P.
9. Invited talk entitled, “Design and development of site specific chemical delivery systems
for antiarthritic drugs” on 4th Feb 2015 at UGC Networking Resource Center, UIPS, Panjab
University, Chandigarah in the training school on “Attaining excellence and compliance
through drug delivery and pharmaceutical technology” during 2nd to 7th Feb 2015.
10. Invited talk entitled, “Basics of NMR” delivered at AICTE-QIP entitled, ‘Spectra based
structural insights into drugs’ organized during 19 th – 24th Jan 2015 on 20th Jan 2015, at
Pharmacy Department, Faculty of Tech. & Engg., The M.S. University of Baroda, Vadodara.
11. Invited talk entitled, “Cracking the API Jargon”, at MSVSS meeting at The M. S. University of
Baroda, Vadodara, on 18th Nov 2014
12. Invited talk entitled, “Role of phytoconstituents in the development of new drug entities” on
18th Jan. 2014 at “3rd Annual National Convention of Pharmacy Professionals” at Faculty of
Pharmacy, D.D. University, Nadiad, Gujarat.
13. Invited talk entitled, “Theoretical basis of NMR Spectroscopy for interpretation of structures
of drugs” on 12th Dec. 2013 under AICTE sponsored Quality Improvement programme on
“Enhancement of teaching and Learning Skills in Pharmaceutical Chemistry Through Problem
Solving Approach” held at Bharati Vidyapeeth Deemed University, Poona College of
Pharmacy, Pune, India From 09th Dec. to 21st December 2013
14. Invited talk entitled, “Phytoconstituents in development of new therapeutics,” under the
AICTE sponsored two weeks summer-winter school entitled, “Recent trends in natural
products drug development and delivery in health care,” on 13th Nov. 2013 organized by B.K.
Modi Government Pharmacy College, Rajkot.
15. Invited talk entitled, “Introduction of 2D-QSAR” under AICTE sponsored Two weeks faculty
development programme on “Recent Trends in Computer Aided Drug Design and Discovery”
on 9th Dec 2013 organized by Parul Group of Institute, Vadodara from 9-21st Dec. 2013.
16. Key note address entitled, “Ever expanding horizons of computational chemistry” on the
occasion of DST-SERB sponsored winter school on Computational Chemistry (WSCC-2013) on
9th Dec. 2013 organized by Department of Chemistry, Sardar Patel University, Vallabh
Vidyanagar from 9-13th Dec. 2013.
17. Invited talk entitled “Synthetic carriers in gene delivery” under the workshop on “Green
nanotechnology and modern industries” organized by CII Government of Gujarat,
Ahmedabad on 25th Oct 2013.
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18. Invited talk entitled, “Molecular modelling in designing of drugs,” under the GUJCOST
sponsored state level seminar on “Advances and emerging trends in new drug design by
molecular modelling, QSAR and retrosynthesis” organized by Pioneer Pharmacy Degree
College, Vadodara on 18th Oct. 2013.
19. Invited lecture entitled, “Strategies for structure elucidation using UV, IR, NMR & MS spectral data”,
organized by Sardar Patel College of Pharmacy, Bakrlol, Anand, Gujarat, in the GUJCOST SPONSORED
one day National seminar on “Structural analysis by various spectroscopic techniques” on 1 st Oct
2013
20. Invited lecture entitled, ‘Modeling techniques in drug discovery’ delivered at B.N. Institute of
Pharmaceutical Sciences, Udaipur, AICTE sponsored Faculty Development Programme on “ An
approach to develop new models in the field of medicinal chemistry” from 16th 28th Sept 2013 on
16th Sept 2013.
21. Invited lecture entitled, ‘Refurbishing the image of pharmacy education in the changing scenario’
delivered at Sigma Institute of Pharmacy, Vadodara in AICTE sponsored National level Pharma
Carnival on Road map for strengthening pharmacy education in changing scenario (17 th 18th Aug
2013) on 17th August 2013.
22. Invited lecture entitled, ‘High resolution mass spectrometery in drug research’, delivered at Babaria
Institute of Pharmacy, Vadodara in AICTE sponsored National Seminar on Quality assurance issues in
drug discovery and formulation development, on 27th July 2013.
23. Invited lecture entitled, Targets for cancer chemotherapy’, delivered at Pune District Education
Association’s Seth Govind Raghunath Sable College of Pharmacy, Saswad, Pune in AICTE sponsored
National Seminar on Frontiers in cancer chemotherapy, on 26th July 2013.
24. Invited lecture entitled, ‘Exploring QSAR for lead optimization’ delivered at B.V. Patel PERD Center,
Ahmedabad, on 14th May 2013.
25. Expert
lecture
entitled,
‘Selectivity
in
mono,
di
and
tri-alkylation
of
3-benzazepine scaffold’ at Gujarat Technological University, Ahmedabad on 9th April in
“Research week 2013” during April 3-16, 2013.
26. Invited lecture entitled, ‘Plants as a source of lead molecules in drug discovery’, delivered at Shree
S.K. Patel College of Pharmaceutical Sciences and Research, Ganpat University, Ganpat Vidyanagar,
Mehsana, in AICTE sponsored two days National seminar on “Recent advances in drug discovery from
natural resources” on 29th March 2013.
27. Invited lecture entitled, ‘Design and development of multi-targeted 6,7-dimethoxyquinazoline
analogs as dual α1- and AII-receptor antagonists’, delivered at Bombay College of Pharmacy, Kalina,
Santacruz, Mumbai on 28th Feb 2013 in AICTE sponsored Faculty development programme on “New
facets of medicinal chemistry in drug discovery” during 18th Feb to 2nd March 2013.
28. Invited lecture entitled, ‘Changing paradigm in drug discovery’, delivered at Pharmacy Department,
The M.S.University of Baroda, Vadodara in AICTE sponsored two-days National Seminar on
“Approached in drug discovery” during 26 – 27 Feb 2013 on 27th Feb 2013
29. Invited lecture entitled, ‘Design and development of multi-targeted 6,7-dimethoxyquinazoline
analogs as dual α1- and AII-receptor antagonists’, delivered at Pharmacy Department, The
M.S.University of Baroda, Vadodara in AICTE sponsored two-days National Seminar on “Approached
in drug discovery” during 26 – 27 Feb 2013 on 26th Feb 2013
30. Invited lecture entitled, ‘Facing GPAT Examination made easy’, in Continuing Pharmacy Education
programme of Indian Pharmacy Association, Vadodara branch on 25th Feb 2013
31. Invited lecture entitled, ‘Design and synthesis of some multi-targeted ligands as anti-hypertensive
agents’, delivered at Department of Pharmacy, Sumandeep Vidyapeeth Waghodia Distt, Vadodara, in
a Two-days National Seminar on “Pharma Rendezous” during 22 – 23 Feb 2013, on 23rd Feb 2013
32. Invited lecture entitled, ‘LC-MS: A versatile technique for pharmaceutical Analysis’ in one day
National seminar on “Advanced in analysis of pharmaceuticals dosage forms by chromatography”
11
33.
34.
35.
36.
37.
38.
39.
40.
41.
sponsored by GUJCOST, organized by Shankarsinh Vaghela Bapu Institute of Pharmacy, GandhinagarMansa Road, Vasan, Gandhinagar on 16th Feb 2013
Invited lecture entitled, ‘Alternative methods and techniques in pharmaceutical analysis’ in State
level seminar on “Justification for selection of Pharmaceutical analytical techniques” organized by
Atmiya Pharmacy College, Ankodiya, Vadodara on 4th Feb 2013
Invited lecture entitled, ‘Virtual screening for the discovery of new drugs’ delivered during the
training school on ‘Computer aided drug design: Hands on workshop’(from 28th January to 9th
February 2013) at UGC Networking Resource Center, University Institute of Pharmaceutical Sciences,
Panjab University, Chandigarh on 29th Jan 2013
Invited lecture entitled, ‘Exploring QSAR for lead optimization’ delivered during the training school on
‘Computer aided drug design: Hands on workshop’(from 28th January to 9th February 2013) at UGC
Networking Resource Center, University Institute of Pharmaceutical Sciences, Panjab University,
Chandigarh on 28th Jan 2013.
Invited lecture entitled, ‘Virtual screening – A versatile tool for new drug discovery process’ in two
day CSIR Sponsored workshop on Hands on training on software related to computer aided drug
design, at Nirma Institute of Pharmacy, Ahmedabad on 22nd Jan 2013
Invited talk entitled, ‘Accreditation- NBA perspective’ on 9th Dec 2012 at 64th Indian Pharmaceutical
Congress, SRM University, Chennai, organized by Indian Pharmaceutical Congress Association during
7th to 9th Dec 2012
Invited talk entitled, ‘Design and development of steroidal aromatase inhibitors as potential drugs for
breast cancer’, on 24th Nov 2012 at International conference on recent advances in pharmaceutical
sciences RAPS-2012’ at University College of Pharmaceutical Sciences, Kakatiya University, Warangal506009, Andhra Pradesh, from 22nd -24th Nov 2012
Invited talk entitled, Do we need regulatory bodies for the growth of higher education?’ delivered on
13th Oct 2012 at NAAC sponsored National Level Seminar on ‘Higher education: Excellence towards
quality management and assurance’, organized by Anand Pharmacy College, Anand, Gujarat on 12th
and 13th Oct 2012
Invited talk as mentor scientist entitled, ‘Wonders of Pharmaceutical Analysis’, delivered in the
science camp on 4th Oct 2012 on ‘Innovation in science pursuit for inspired research internship 2012’
from 1st Oct to 6th Oct 2012 at SPP School of Pharmacy & Technology Management, NMIMS, Mumbai
Invited talk on ‘NMR Spectroscopy’ under the “CPE Programme” of Indian Pharmaceutical
Association, Vadodara Branch on 24th Aug 2012 at Faculty of Technology Auditorium, The
M.S.University of Baroda, Vadodara
42. Invited talk on ‘New Steroidal aromatase inhibitors as potential anticancer agents in breast
cancer, at Shri Sarvajanik College of Pharmacy, Mehsana, Gujarat on 21st July 2012.
43. Invited lecture on ‘Design and development of site specific chemical delivery systems for
anti-arthritic agents’, delivered at Pioneer Pharmacy Degree College, Vadodara, in a One day state
level seminar & poster competition on ‘Advances and emerging trends in pharmaceutical Sciences’
on 7th April 2012
44. Invited lecture on ‘Dual α1- and AT-1 inhibitors as potential antihypertensive agents’,
delivered at Shri B.M. Shah College of Pharmaceutical Education & Research, Modasa, during
GUJCOST sponsored National Seminar on “Pharmaceutical Education: Need of Academia and
Industry Harmonization” on March 3, 2012
45. Invited lecture on ‘Rrelevance of different analytical technique in pharmaceutical analysis – current
perspectives’ delivered at Pharmacy Department, The M. S. University of Baroda, under Ms. Kanan
Ishwar Mehta Memorial Annual lectures on 27th Sept 2011.
46. Invited lecture on ‘Application of Spectroscopy in Pharmacy Field’ delivered in one day
symposium on “Novel technologies to expedite drug discovery and development”, organized
by Saraswati Institute of Pharmaceutical Sciences, Gandhinagar on 24th Sept 2011.
12
47. Invited talk on ‘New Steroidal aromatase inhibitors as potential anticancer agents in breast
cancer, at Al-Ameen College of Pharmacy, Bangalore, on 20th Sept 2011
48. Invited talk on ‘Simulation techniques in drug design and development’ at Department of
Chemistry, Faculty of Science, The M. S. University of Baroda, Vadodara in a Five day Winter
School of Bio-inorganic Chemistry from 8th -12th March 2011, under UGC-CAS Program, on
10th March 2011.
49. Invited talk on ‘Interpretation of NMR spectra and identification of organic compounds by
spectroscopy’ at Saraswathi Vidya Bhavan’s College of Pharmacy, Dombivli (E), in two days
National workshop on ‘NMR & Co-relation spectroscopy’, on 4th & 5th February 2011.
50. Invited talk on ‘Structural elucidation of organic compounds’ delivered at Sinhgad College of
Pharmacy, Pune, under University of Pune sponsored seminar grant, 18th -20th Jan 2011.
51. Invited talk ‘Steroidal aromatase inhibitors as potential drugs for breast carcinoma’ delivered
in International conference on Recent Advances in Pharmaceutical sciences- 2010, organized
by Department of Pharmaceutics, IT-BHU, Varanasi, 22-23rd Dec 2010.
52. Invited talk on ‘Spectroscopic techniques- Recent developments’, delivered at Ravishankar
College of Pharmacy, Bhopal, on 18th Dec 2010.
53. Invited talk on ‘Structure elucidation using spectroscopic techniques’ delivered in National
Seminar on ‘Quality assurance issues in drug discovery & formulation development’ at
Babaria Institute of Pharmacy, Vadodara, on 3rd - 4th December 2010.
54. Invited talk on ‘New aromatase inhibitors: Steroids as potential therapeutics for breast
cancer’, delivered in ‘6th International symposium on Innovations in pharmaceutical sciences
and technology’ organized by B. V. Patel Education Trust and B. V. Patel PERD Centre,
Ahmedabad, Gujarat from 26-28th Nov 2010.
55. Invited talk on ‘Discovery of some novel TACE inhibitors: A journey through desktop to
benchtop’ delivered in ‘International conference on Recent Advances in Drug Discovery’
organized by the University College of Pharmaceutical Sciences, Kakatiya University,
Warangal, A.P. from 22nd to 24th Oct 2010.
56. Invited talk on ‘Theoretical principles of NMR Spectroscopy’ delivered at Parul College of
Pharmacy, Gujarat, under the SDP on the topic, on 4th Sept 2010.
57. Invited talk on Interpretation of NMR spectra for structure elucidation in "Structural
elucidation of organic compounds through spectroscopic data” on 28th and 29th June, 2010
organized by Satara College of Pharmacy, Satara, Maharashtra, 29th June, 2010.
58. Invited talk on ‘QSAR and Molecular Modelling’ in AICTE sponsored Quality Improvement
Programme 2010 on ‘Glimpses of current Advances in the Field of Pharmaceutical Sciences’
on June 7th, 2010, organized by Pharmacy Department, The M. S. University of Baroda,
Vadodara, 7th to 12th June 2010.
59. Invited talk on ‘Research Methodology in synthetic Medicinal Chemistry’ in AICTE sponsored
Quality Improvement Programme 2010 on ‘Glimpses of current Advances in the Field of
Pharmaceutical Sciences’ on June 7th, 2010, organized by Pharmacy Department, The M. S.
University of Baroda, Vadodara, 7th to 12th June 2010.
60. Invited talk on ‘Peptidomimetics in Drug Discovery’ at University Institute of Pharmaceutical
Sciences, Panjab University, Chandigarh on 1st June 2010 in UGC Networking Resource
Centre under the theme of ‘Emerging Trends in Drug Discovery’ and Development from 31 st
May to 12th June 2010.
61. Invited talk on ‘Indian Patent and PCT Applications’ at The M. S. University of Baroda in UGC
sponsored Symposium on ‘Patent awareness and Scientific writing’, 27 th March 2009
13
62. Invited talk delivered on “High Throughput Screening in Drug Discovery” at Poona College of
Pharmacy, Pune, Maharashtra under AICTE sponsored staff development programme for
Pharmacy teachers on 27th Feb 2009.
63. Invited talk delivered on “CoMFA and CoMSIA techniques in Drug Design and Discovery” at
R.C.Patel Institute of Pharmaceutical Education and Research, Shirpur, Maharashtra under
AICTE sponsored staff development programme for Pharmacy teachers on 13th Feb 2009.
64. Invited talk entitled, ‘Stereochemistry’ delivered at STE’s Sinhgad College of Pharmacy,
Vadgaon, Pune on 10th Feb 2009.
65. Invited lecture delivered on the topic “Spectrophotometric techniques” at Baroda college of
Pharmacy, Vadodara on 8th Sept. 2008.
66. Lecture Delivered on “Peptides in Drug Design” in PCI Sponsored State level Orientation
Programme for Pharmacy Teachers” held at Shri Sarvajanic Pharmacy College, Mehasana,
Gujarat, 1st Feb. 2008.
67. Invited Talk entitled, “Pharmacy Education - Current Scenario and Future Directions”,
delivered at Annual Convention of APTI organised by UIPS, Panjab University, Chandigarh,
25th Oct. 2007.
68. Invited Talk on “3D-QSAR and Docking Studies in Drug Design” delivered at National Seminar
and Workshop of Pharmacoinformatics organised by PSG College of Pharmacy, Coimbatore,
23rd March 2007.
69. Guest Lecture at Shri Sarvajanic Pharmacy College, Mehsana, on the topic “3D-QSAR and
Docking Studies in Drug Design” on 23rd Oct. 2007.
70. Invited Lecture in AICTE Sponsored Two Weeks Staff Development Programme entitled, “3DQSAR and Docking Studies in Drug Design” organized by S.K. Patel College of Pharmaceutical
Education and Research, Ganpat University, Kherva, Mehsana from 13th to 27th April 2007.
71. Invited lecture in AICTE Sponsored Two Weeks Staff Development Programme entitled,
“Advances in Characterization of Phytochemical Constituents” organized by S.K. Patel College
of Pharmaceutical Education and Research, Ganpat University, Kherva, Mehsana from Jan.
29th to 11th Feb. 2007.
72. Invited Lecture under Continuing Pharmacy Education Programme of Indian Pharmaceutical
Association, Vadodara Branch on “Licensing of Intellectual Property Rights” on 14 th Oct.
2006.
73. Invited Lecture in Workshop on “Contemporary Topics in Pharmaceutical Sciences on
“Peptidomimetics in Drug Discovery” organized by QIP Centre AICTE and TIFAC Centre of
Relevance and Excellence in New Drug Delivery System at Pharmacy Department, The M.S.
University of Baroda on 21st June 2006.
74. Invited Lecture entitled “Protease Inhibitors as Potential Drugs” delivered at C.U. Shah
College of Pharmacy, SNDT Women’s University, Mumbai on 16th Feb 2006 during their Silver
Jubilee Celebrations.
75. Special Lecture entitled “Designing of Peptidomemetics as Potential Drugs” delivered at Shri
Sarvajanic Pharmacy College, Mehsana, Gujarat, during National Pharmacy Week on 26 th
Oct. 2005.
76. Invited Lecture entitled, “Computer Assisted Drug Design” on a One day Workshop on
“Computer Assisted Drug Design” organized by Prin. K.M. Kundanani College of Pharmacy,
Mumbai on 15th Oct. 2005.
77. Guest lecture entitled, “Importance of Organic Chemistry in Pharmacy” delivered at S.B.
College of Pharmacy, Sivakasi, TN, on the Annual Celebrations on 23rd March 2005.
14
78. Invited Lecture entitled, “QSAR in Dosage form Designing” delivered at AICTE-ISTE Sponsored
Short Term Training Programme Organized by A.R. College of Pharmacy, Vallabh Vidyanagar,
from 25th May to 5th June 2004.
79. Invited Lecture entitled, “Radiotracers in in vitro and Preclinical Studies” delivered in 24th
Annual Conference of Indian Association of Biomedical Scientist on the topic Radiotracers in
Drug Development, organized by Institute of Nuclear Medicine and Allied Sciences, DRDO,
New Delhi on 2nd Nov. 2003.
80. Invited Lecture entitled “Peptide Leads in New Drug Discovery” delivered at UGC Sponsored
Refresher Course in Pharmaceutical Sciences on Current Concept in Drug Design and
Formulation Development organized by Department of Pharm. Sciences, Guru Jambheshwar
University Hisar from Oct. 1st to Oct. 21st 2003.
81. Invited Lecture entitled “Applications of Computers in Drug Discovery” delivered at UGC
Sponsored Refresher Course in Pharmaceutical Sciences on Recent Advances in
Pharmaceutical Technology and Computer Applications, organized by Department of Pharm.
Sciences, Guru Jambheshwar University Hisar from Feb. 20th to March 12th 2003.
82. Invited Lecture entitled “Protease Inhibitors as New Drugs” delivered at UGC Sponsored
Refresher Course in Pharmaceutical Sciences on Recent Advances in Pharmaceutical
Technology and Computer Applications organized by Department of Pharm. Sciences, Guru
Jambheshwar University, Hisar from Feb. 20th to March 12th 2003.
83. Invited Lecture entitled “Drug Discovery- In Retrospect” delivered at UGC Sponsored
Refresher Course in Pharmaceutical Sciences organized by Department of Pharm. Sciences,
Guru Jambheshwar University Hisar from Jan 30th to Feb.19th 2002.
84. Invited Lecture entitled “Molecular Modelling and Drug Designing” delivered at UGC
Sponsored Refresher Course in Pharmaceutical Sciences organized by Department of Pharm.
Sciences, Guru Jambheshwar University Hisar from Jan 30th to Feb.19th 2002.
85. Invited Lecture entitled “Computers and Drug Discovery” delivered at AICTE-ISTE Sponsored
Short Term Training programme on Pharm. Sciences in the New Millennium- Emerging
Trends & Challenges Ahead, organized by A.R. College of Pharmacy, Vallabh Vidyanagar,
from 30th April 2001 to 12th May 2001.
86. Invited Lecture entitled “Basic Test for Common Medicines”, WHO Sponsored Professional
Training Programme organized by Pharmacy Department, The M.S. University of Baroda on
23rd April 2001.
87. Invited Lecture entitled, “Rational Drug Design” on 1st March at Department of Pharm.
Sciences, Dr. Harisingh Gour Vishwavidyalaya, Sagar during 28th Feb. to 12th March 2000.
88. Invited Lecture entitled, “Drug Discovery- In Retrospect” on 1st March 2000 in AICTE
Sponsored Short Term Training Programme on “Frontiers in Pharmaceutical Chemistry”
organized by ISTE at Department of Pharm. Sciences, Dr. Harisingh Gour Vishwavidyalaya,
Sagar during 28th Feb. to 12th March 2000.
89. Invited Lecture delivered AICTE and ISTE Sponsored Short Term Training Programme on
Recent Developments in Pharm. Sciences organized by A.R. College of Pharmacy, Vallabh
Vidyanagar from 26th Oct. to 7th Nov. 1998.
90. Invited Lecture in ISTE Summer School on Trends in Development of Drugs and Delivery
Systems-A Futuristic Approach organized by Pharmacy Department, The M.S. University of
Baroda, Vadodara from 19th to 31st March 1997.
SCIENTIFIC PUBLICATIONS
15
Research Papers
Reviews
Book Chapters
Patents
: 110
: 26
: 04
: 17
List of Research Articles:
Sr.
No.
1.
Name of Journal,
Vol. & Page No.
Year
Journal
of Pharmaceutical
Prajapati, Ashish M.
Sciences and
Kanhed, Kirti Patel, Rajani
Pharmacology
Giridhar, Mange Ram
In
Press
Title of the Paper
D3 antagonist
and antipsychotic potential of
some novel benzazepines
Author(s)
Jatin Machhi, Navnit
Yadav
2.
3.
4.
5.
Combined atom-based 3DQSAR and structure-based
modelling for identifying new
leads – A new approach
applied to discover potential
non-nucleoside reverse
transcriptase inhibitors
Neuroprotective potential of
novel multi-targeted
isoalloxazine derivatives in
rodent models of Alzheimer's
disease through activation of
canonical Wnt/β-catenin
signalling pathway.
Synthesis and SAR of
substituted 3-benzazepines as
potent and selective 5-HT2C
receptor agonists
Neuroprotective role of novel
benzazepine derivative
through D1 agonism in 6OHDA-induced Parkinson's
model of rat
Radha Charan Dash,
Ashish M. Kanhed,
Mugdha R. Suryawanshi,
Sharad H. Bobsale, Mange
Ram Yadav
J. Chem. Inf. Mod.
In
Press
Jatin Machhi, Anshuman
Sinha, Pratik Patel, Ashish
M. Kanhed, Ashutosh
Tripathi, Zalak S. Parikh,
Ragitha Chaturvedi,
Prakash p. Pillai, Sarita
Gupta, Kirti Patel, Rajani
Giridhar, Mange Ram
Yadav
N. Prajapati, A. Sinha,
R.Giridhar and M.R.Yadav
Neurotoxicity
Research
In
Press
Curr. Med. Chem.
In
Press
Anshuman Sinha, Jatin
Machhi, Navnit Prajapati,
Ashish M Kanhed,
Ashutosh Tripathi, Zalak S
Parikh Prakash P Pillai,
Rajani Giridhar, Mange
Ram Yadav
European Journal of
Pharmacology
In
Press
16
6.
3-Substituted 1-methyl-3benzazepin-2-ones as 5-HT2C
receptor agonists
Mahesh Mohan
Shidore, Jatin
Machhi, Prashant
Murumkar, Mahesh
Barmade, Jigar
Thanki and Mange Ram
Yadav
RSC Adv., 5, 91908 91021
2015
7.
Benzo[e]pyrimido[5,4b][1,4]diazepin-6(11H)-one
Derivatives as Aurora A Kinase
Inhibitors: LQTA-QSAR Analysis
and Detailed Systematic
Validation of the Developed
Model
Exploring structural
requirements for peripherally
acting 1,5-diaryl pyrazole
containing cannabinoid 1
receptor antagonists for the
treatment of obesity
Discovery of isoalloxazine
derivatives as a new class of
potential anti-Alzheimer
agents and their synthesis
Ashish M. Kanhed, Radha
Charan Dash, Nishant
Parmar, Tarun Kumar Das,
Rajani Giridhar, Mange
Ram Yadav
Molecular Diversity,
19, 965-974
2015
Mayank Kumar Sharma,
Prashant R. Murumkar,
Rajani Giridhar, Mange
Ram Yadav
Molecular Diversity,
19, 871-893
2015
Ashish M Kanhed,
Anshuman Sinha, Jatin
Machhi, Ashutosh Tripathi,
Zalak Parikh, Prakash Pillai,
Rajani Giridhar and Mange
Ram Yadav
R.S.Tamboli, R.Giridhar,
H.Gandhi, A.M.Kanhed,
H.M.Mande and
M.R.Yadav
Bioorganic
Chemistry, 61, 7-12
2015
J. Enz. Inh. Med.
Chem.
Accept
ed
Mange Ram Yadav, Riyaj S
Tamboli, Hemant M
Mande, Haribhai A Rabari,
Rajani Giridhar
Navnit Prajapati, Rajani
Giridhar, Anshuman Sinha,
Ashish M. Kanhed,
Mange Ram Yadav
Tetrahedron Lett.,
56, 3858–3860
2015
Molecular Diversity,
19, 653-667
2015
8.
9.
10.
11.
12.
Design, green synthesis and
pharmacological evaluation of
novel 5,6-diaryl-1,2,4-triazines
bearing 3-morpholinoethylamine moiety as potential
antithrombotic agents
Base catalyzed novel
rearrangement of steroidal
[3,4-c]furoxans
Regioselective alkylation of
1,3,4,5-tetrahydrobenzo[d]
azepin-2-one and biological
evaluation of the resulting
alkylated products as
potentially selective 5-HT2C
17
agonists
13.
14.
15.
16.
17.
18.
19.
20.
Enhancing Skin Permeation of
Biphenylacetic acid (BPA)
Using Salt Formation with
Organic and Alkali Metal Bases
Neuroprotective role of novel
triazine derivatives by acting
on Wnt/β catenin signalling
pathway in rodent models of
Alzheimer’s disease
Potential of
piperazinylalkylester prodrugs
of 6-methoxy-2-naphthylacetic
acid (6-MNA) for percutaneous
drug delivery
6,7-Dimethoxyquinazolines as
Potential Cytotoxic agents:
synthesis and in vitro activity
Virtual screening-based
identification of lead
molecules as selective TACE
inhibitors
Structural requirements for
imidazo[1,2-a]pyrazine
derivatives
as Aurora A kinase inhibitors
and validation of the model
Synthesis and biological
evaluation of some novel
pyrido[1,2-a]pyrimidin-4-ones
as anti-malarial agents
Room-temperature ionic
liquid–DMSO Promoted and
improved one-pot synthesis
Of 5,6-diaryl-1,2,4-triazines
Vijay Pawar, Prashant
Naik, Rajani Giridhar,
Mange Ram Yadav
AAPS PharmSciTech,
In
press
Sinha A.., Tamboli R.S.,
Seth B., Kanhed A.M.,
Tiwari S., Agrawal S., Nair
S., Giridhar R., Chaturvedi
R.K., Yadav M.R.
Molecular
Neurobiology
In
press
Vijay Pawar, R.Thosani, A.
Kanhed, R.Giridhar and
M.R.Yadav
AAPS
PharmSciTech, 16,
518-27
2015
M. R. Yadav, B. S.
Chauhan, P. P. Naik,
Hardik Gandhi,
R. Giridhar
Prashant R. Murumkar,
Mayank Kumar Sharma,
Rajani Giridhar, Mange
Ram Yadav
Lett. Drug Des. Dis.,
12, 190 - 205
2015
Med. Chem. Res.,
24, 226-244
2015
Ashish M. Kanhed, Vishal
P. Zambre, Vijay A. Pawar,
Mayank Kumar Sharma,
Rajani Giridhar, Mange
Ram Yadav
Med. Chem. Res.,
23, 5215–5223
2014
Uttam R. Mane, D.
Mohanakrishnan, Dinkar
Sahal, Prashant R.
Murumkar,
Rajani Giridhar, Mange
Ram Yadav
Riyaj S. Tamboli , Rajani
Giridhar, Hemant M.
Mande, Shailesh
R. Shah & Mange Ram
Yadav
Eur. J. Med. Chem.
79, 422-435
2014
Synt. Comm.
44, 2192–2204.
2014
18
21.
22.
23.
24.
25.
26.
27.
An HPTLC method for
quantification of cholesteryl
esters from human plasma and
rat liver microsomes
Enhanced skin permeation of
6-methoxy-2-naphthylacetic
acid by salt formation
Hardik Gandhi, Palash Pal,
Rajani Giridhar,
M.R.Yadav
Biomedical
Chromatography.
28, 583–588
2014
Vijay Pawar, H. Yogish
Kumar, Rajani Giridhar,
and Mange Ram Yadav
Drug Deliv.
(DOI: .3109/107
17544.2014.894595)
2014
Molecular Modeling Studies of
Some Triazine Derivatives as
G-quadruplex binders for
inhibition of telomerase
enzyme
Synthesis of novel 4,6-diaryl-2aminopyrimidines as potential
antiplasmodial agents
Vishal P Zambre, Rajani
Giridhar and Mange Ram
Yadav
Med. Chem. Res.,
22, 4685-4699
2013
R. Giridhar,
R.S. Tamboli,
D.G.Prajapati, S. Soni, S.
Gupta and M.R.Yadav
P. Naik, H. Gandhi, B.S.
Chauhan, R. Giridhar,
M.R.Yadav
Med. Chem. Res.,
22 (7), 3309-3315
2013
Bio-org. Med. Chem.
Lett., 23, 3959-3966
2013
Amit Verma, N.
Prajapati,S. Salecha,R.
Giridhar, M.R. Yadav
Tet. Lett., 54, 2029 2032
2013
M. R. Yadav, U. R. Mane,
R. Giridhar, H. Li, J. Huang,
R. C. Gupta, S. S. Nadkani,
C. Dutt, V. Chouthaiwale
and P. P. Naik
Amit Verma, R.Giridhar
and M. R. Yadav
Bio-org. Med. Chem.
20, 6296 - 6304
2012
Tet. Lett., 53, 2954 2958
2012
Rajani Giridhar, Riyaj S.
Tamboli, R. Ramajayam,
Dhaval G. Prajapati and
M.R.Yadav
Eur. J. Med. Chem.,
50, 428-432
2012
Design and synthesis of 6,7dimethoxyquinazoline analogs
as multi-targeted ligands for
<alpha>1- and AII-receptors
antagonism
Microwave Assisted Palladium
Catalyzed Intermolecular αArylation of Copper-Amide
Enolate.of Benzazepine
Pyrido[1,2-a]pyrimidin-4-ones
as
potential
plasmodial
falcipain-2 inhibitors
28. 8A facile IL-DMSO assisted
3synthesis of benzo annelated
five-, six- and sevenmembered heterocycles
29. 8Assessment of antiplatelet
2activity of 2-aminopyrimidines
19
30. 8Steroidal carbonitriles as
1Potential aromatase inhibitor
Mange Ram Yadav,
Prafulla M. Sabale, Rajani
Giridhar, Christina Zimmer
and Rolf W. Hartmann
31. 8Cytotoxic potential of novel M. R. Yadav, Fedora
Grande ; Bishram S
06,7-dimethoxyquinazolines
Chouhan ; Prashant P Naik
; Rajani Giridhar ; Antonio
Garofalo; Nouri Neamati
32. 7Revelation on the potency of α1- M. R. Yadav, H. P. Gandhi,
P. P. Naik and R. Giridhar
9blockers – Parallel blockade of
33.
34.
Angiotensin II receptor: A new
finding
Improved percutaneous delivery
of some NSAIDs for the
treatment of arthritis
Cartilage tartgeted chemical
delivery of naproxen and
ibuprofen for the treatment of
arthritis
Steroids, 77, 850 857
2012
Eur. J. Med. Chem.,
48, 231 -247
2012
Pharm. Biol., 50, 439
-442
2012
R. Thosani, V. Pawar, R. J. Pharm. Bioallied
Giridhar and M.R.Yadav
Sciences, 4(S), S12-3
2012
V.Pawar,
V.
Gohil, J. Pharm. Bioallied
R.Tamboli, R.Giridhar and Sciences, 4(S), S10-1
M.R.Yadav
2012
35. 7Synthesis,
preliminary
8biological evaluation and
molecular modeling of some
new heterocyclic inhibitors of
TACE
P. Sengupta, C. S. Puri, H.
A. Chokshi, C. K. Sheth,
A. S. Midha, T. Rao C.,
Rajamannar T., P. R.
Murumkar and M.R.
Yadav
Eur. J. Med. Chem.,
46, 5549-55
36. 7Synthesis and Preliminary
7Screening of Novel A- and DRing Modified Steroids as
Aromatase Inhibitors
M. R. Yadav, Prafulla M. Let. Drug Des. Dis.,
Sabale, Rajani Giridhar, 8, (10), 943-950
Dharmendra
Baria,
Christina Zimmer and Rolf
W. Hartmann
37. 7Determining of Structural
6Requirements of Influenza
Neuraminidase Type A
Inhibitors and Binding
Interaction Analysis with the
Active Site of A/H1N1 by 3DQSAR CoMFA and CoMSIA
Modeling
38. 7Synthesis of Some Novel
5Androstanes as Potential
Aromatase Inhibitors
Murumkar P. , Le Ly,
Truong Thanh and
M.R.Yadav
Med. Chem.
Commun., 2, 710719
M. R. Yadav, P. M. Sabale,
R. Giridhar,
C. Zimmer and R. W.
Hartmann
Steroids, 76, 464-70
2011
2011
2011
2011
20
39. 73D-QSAR studies of 44quinolone derivatives as highaffinity ligands at the
benzodiazepine site of brain
GABAA receptors
40. 7Development of highly
3predictive 3D-QSAR CoMSIA
models for anthraquinone and
acridone derivatives as
telomerase inhibitors which
target G-quadruplex DNA
telomere
41. 7Development of predictive
2pharmacophore model for in
silico screening, and 3D QSAR
CoMFA and CoMSIA studies
for lead optimization, for
designing of potent tumor
necrosis factor alpha
converting enzyme inhibitors
42. 7Synthesis and anti-HIV-1
1integrase activitiy of cyano
pyrimidinones
A. Gaurav, M.R.Yadav, R.
Giridhar, V. Gautam, R.
Singh
Medicinal Chemistry
Research, 20, 192-97
V.P. Zambre, P.R.
Murumkar, R. Giridhar, M.
R. Yadav
Journal of Molecular
Graphics and
Modelling, 29, 229239
Murumkar, P.R., Zambre,
V.P., Yadav, M.R.
Journal of
Computer-Aided
Molecular Design 24
(2), pp. 143-156
Ramajayam, R., Mahera,
N.B., Neamati, N., Yadav,
M.R., Giridhar, R.
Archiv der
Pharmazie
342 (12), 710-715
43. 7QSAR studies on 4-quinolone
0derivatives as high-affinity
ligands at the benzodiazepine
site of brain GABAA receptors
44. 6Metalloantibiotics: synthesis,
9characterization and
antimicrobial evaluation of
bismuth-fluoroquinolone
antibiotic complexes against
Helicobacter pylori
45. 6Studies on novel 28imidazolidinones and
tetrahydropyrimidin-2(1H)ones as potential TACE
inhibitors: Design, synthesis,
molecular modeling, and
preliminary biological
evaluation
46. 6Structural investigation of
7acridine derivatives by CoMFA
and CoMSIA reveals novel
Gaurav, A., Yadav, M.R.,
Giridhar, R., Gautam, V.,
Singh, R.
Medicinal Chemistry
5 (4), 353-358
Anwar Shaikh, Rajani
Giridhar, Francis Mgraud
and M.R.Yadav
Acta Pharm. 59 (3),
pp. 259-271
Shirshendu DasGupta,
Prashant R Murumkar,
Rajani Giridhar and M. R.
Yadav
Bio-org. Med.
Chem., 17, 3604-17
Vishal P Zambre, Prashant
R Murumkar, Rajani
J. Chem. Info. Mod.
49,5, 1298-1311
2011
2010
2010
2009
2009
2009
2009
2009
21
insight towards DNA Gquadruplex mediated
telomerase inhibition and
offer a highly predictive 3Dmodel for substituted
acridines
47. 6Design, synthesis and
6preliminary screening of some
new conformationally
constrained Falcipain-2
inhibitors as potential
antimalerial agents
48. 6Development of predictive 3D5QSAR CoMFA and CoMSIA
Models for βAminohydroxamic AcidDerived Tumor Necrosis-α
Converting Enzyme Inhibitors
49. 6Synthesis, antileukemic and
4antiplatelet activities of 2,3diaryl-6,7-dihydro-5H-1,4diazepines
Giridhar and M. R. Yadav
A. K. Shinde, B. S.
Chauhan, S. D. Gupta, R.
Giridhar, P. Rosenthal, J.
Gut and M.R.Yadav
Letters in Drug
Design & Discovery,
6 (4), 258-267
Prashant R. Murumkar,
Vishal P. Zambre, Rajani
Giridhar and M. R. Yadav
Chem. Biol. Drug
Des., 73, 97-107
R.Ramajayam, R.Giridhar,
M.R.Yadav, R.Balraman,
H.Djaballah, D.Shum and
C.Rady
M.R. Yadav, Vijay Pawar,
P.K. Halen, R. Giridhar
Eu. J. Med. Chem.,
43, 2004-2010
2008
50. 6Site specific chemical delivery
3of NSAIDs to inflamed joints:
Synthesis, biological activity
and γ-imaging studies of
quaternary ammonium salts of
tropinol esters of some NSAIDs
51. 6Peptidomimetics 2M.R.Yadav, A.K. Shinde,
2Cyanopyrrolidine as Potential
B.S. Chauhan, R. Giridhar,
Selective Cathepsin L
Robert Menard
Inhibitors
Bio-org. Med.
Chem., 16(21) 94439449
2008
J. Enz. Inh. Med.
Chem., 23(2), 190197
2008
52. 63D-Quantitative Structure1Activity Relationship Studies
on Benzothiadiazapine
Hydroxamates as Inhibitors of
Tumor Necrosis Factor-α
Converting Enzyme
Prashant R. Murumkar,
R.Giridhar and Mange
Ram Yadav
Chem. Biol. Drug
Des., 71, 363-373
2008
53. 6Studies on crystal forms of
0Pefloxacine: Preparation,
Characterization and
Dissolution Profile
M.R.Yadav, Anwar Shaikh,
V. Ganesan, Rajani
Giridhar, Renu C.
J. Pharm. Sci., 26372648
2008
2009
2009
22
54. 5Synthesis antiproliferative
9activity of some
diaryldiazepines and
diarylpyrimidines
55. 5Combining antocholinergic and
8anti-inflammatory activities
into a single moiety: A novel
approach to reduce
gastrointestinal toxicity of
ibuprofen and ketoprofen
56. 5Substituted aminoalcohol
7ester analogs of indomethacin
with reduced toxic effects
57. 5Insights into the structural
6requirements of
farnesyltransferase inhibitors
as potential anti-tumor agents
based on 3D QSAR CoMFA and
CoMSIA models
58. 5Bismuth -norfloxacin complex:
5Synthesis, physicochemical
and antimicrobial evaluation
59. 5Studies in 3,4-diaryl-1,2,54oxadiazoles and their Noxides: Search for better COX2 inhibitors
60. 5Synthesis and Evaluation of
3some Gastrointestinal sparing
anti-inflammatory amino ethyl
ester derivatives and
naphthalene-based NSAIDs
61. 5Synthesis and Pharmacological
2Investigation of Novel 1-Alkyl4-(4-substituted
aryl/heteroaryl)-1,2,4triazolo[4,3-a]quinazolin5(4H)-ones as a New Class of
H1-Antihistaminic Agents
62. 5Synthesis of new chemical
1entities from paracetamol and
NSAIDs with improved
pharmacodynamics profile
R. Ramajayam, R. Giridhar,
M.R.Yadav, H.Djaballah,
D.Shun and C.Radu
J. Enz. Inhib. Med.
Chem., 22(6), 716721
P.K Halen, K.K. Chagti,
R.Giridhar, M.R.Yadav
Chem. Biol. Drug
Des., 70, 450-455
P.K Halen, K.K. Chagti,
R.Giridhar, M.R.Yadav
Med. Chem. Res.,
16, 101-111
2007
D. S. Puntambekar, R.
Giridhar, M. R. Yadav
Eur. J. Med. Chem.,
41 (11) 1279-1292
2007
A.R. Shaikh, R. Giridhar,
M.R. Yadav
Int. J.
Pharmaceutics, 332 ,
24–30
Acta Pharm. 57, 13–
30
2007
Arch. Pharm. Chem.
LifeSci.340, 88-94
2007
M. R.Yadav, S.T. Shirude,
D. S. Puntambekar, P.J.
Patel, H.B. Prajapati, A.
Parmar R. Balaraman, R.
Giridhar
P.K.Halen, Manisha Rawal,
K.K. Chagti, R. Giridhar,
M.R. Yadav
V.Alagarsamy, M.R.Yadav
and R. Giridhar
Arznein.-Forsch., 56
(12), 834-841
P.K.Halen, S.T. Shirode, R.
Giridhar, M.R. Yadav
Biorg. & Med.
Chem., 14, 87018706
2007
2007
2007
2006
2006
23
63. 5Anti-HIV, Antibacterial,
0Antifungal activities of some
novel 1, 4-disubstituted 1,2,4triazolo[4,3-a] Quinazolin5(4H)-ones
64. 4Synthesis of new chemical
9entities from paracetamol and
NSAIDS with improved
pharmacodynamic profile
V. Alagarsamy, R. Giridhar,
M. R.Yadav, R. Revathi, E.
deCercq, K. Rukmani
Indian J. Pharm. Sci.,
68, 532-535
2006
M.R.Yadav, D.M.
Biorg. Med. Chem.,
Brahamkshatriya, S.T.
14, 8701-8706
Shirude, A. Parmar, R.
Balaraman and R. Giridhar
2006
65. 4Synthesis and pharmacological
8evaluation of some dual acting
aminoalcohol esters
derivatives of flubiprofen and
biphenyl acetic acid
66. 4Synthesis and Anti7Inflammatory activity of 2,3Diaryl-4-(3H)quinazolinones
P.K. Halen, M. R. Yadav,
K.K Chagti, and R. Giridhar
Chem. Biodiv., 3,
1238-1248
2006
M.R.Yadav, S.T. Shirude,
A. Parmar, R. Balaraman
and R. Giridhar
Khim. Geterotsikl.
Soedin., 42, 11981205
2006
67. 4Understanding the Antitumor
6activity of tricyclicpiperazinyl
derivatives as
farnesyltransferase inhibitors
using CoMFA and CoMSIA
68. 4Synthesis of Novel substituted
5diaryl 1,4-Diazepines
D.S. Puntambekar, R.
Giridhar and M.R.Yadav
Eur. J. Med. Chem.,
41, 1279–1292
2006
R.Ramajayam, R. Giridhar
and M.R.Yadav
69. 4An efficient and time saving
4microwave-assisted selenium
dioxide oxidation of 1,2diarylethanones
70. 43D-QSAR studies of farnesyl
3transferase inhibitors: A
comparative molecular field
analysis study
71. 43D QSAR CoMFA/CoMSIA
S.T. Shirude, P. Patel, R.
Giridhar and M.R.Yadav
Chemistry of
2006
Heterocyclic
Compounds, 42 (7),
901-906
Indian J. Chem., 45B, 2006
1080-1085
D.S. Puntambekar, R.
Giridhar and M.R. Yadav
Biorg. Med. Chem.
Lett. 16, 1821-1827
2006
D.S. Puntambekar, R.
Acta Pharm. 56, 157
2006
24
72.
73.
74.
75.
2studies on 5-aryl-2,2-dialkyl-4phenyl-3H)furanone
derivatives as selective COX-II
inhibitors
4Synthesis and evaluation of
1dual acting esters of aspirin
and ketorolac
4Synthesis and pharmacological
0investigation of novel 1substituted 4(methoxyphenyl)-1,2,4triazolo[4,3-a] Quinazolin5(4H)-ones as a new class of
H1-antihisttaminic agents
3Identification of novel non9Nucleoside reverse
transcriptase inhibitors using
fragment-based lead
generation
3QSAR studies of
8diarylimidazoles as selective
COX-2 inhibitors
Giridhar and M.R. Yadav
P.K. Halen, M.R. Yadav,
K.K Chagti, C.S. Reshmi,R.
Giridhar
V Alagarsamy , R. Giridhar,
M.R. Yadav
Ars. Pharm., 47, 6179
R .Ramajayam, R. Giridhar,
M.R.Yadav, E. deClercq, C.
Pannecouque and G.P.
Dhaval
Med. Chem. Res, 14,
475-487
M.R.Yadav,
D.S.Puntambekar,
K.P.Sarathy, S.
Vengurlekar, R. Giridhar
M.R.Yadav, P.Halen, K.
Chagti, B. Hemalatha
R.Giridhar
V. Alagarsamy, R. Giridhar,
M.R.Yadav
Indian J. Chem., 45B, 2005
475-482
76. 3A novel approach towards
therapeutic optimization of
7
diclofenac
77. 3Synthesis and pharmacological
6investigation of novel 1. substituted-4-phenyl-1,2,4triazolo[4,3-a]quinazolin5(4H)-ones as a new class of
H1-antihistaminic agents
78. 3Effect of bis[Curcumino]
J.B.Majithia, R.Balaraman,
5oxovanadium complex on non- R. Giridhar, M.R.Yadav
. diabetic and Streptozotocininduced Diabetic Rats
Alagarsamy V, Giridhar
79. Synthesis and H1antihistaminic activity of some
novel 1-substituted-4-(3methylphenyl)-1,2,4-triazolo
[4,3-a]quinazolin-5(4H)-ones.
R, Yadav M.R.
2006
J Pharm. Pharmacol., 2006
58, 1249- 1255
2005
ARS Pharma., 46,
263-267
2005
Bioorganic Med.
Chem. Lett., 15,
1877-1880
2005
J. Trace Elem. Med.
Biol., 18, 211-217
2005
Biol. Pharm. Bull., 28
(8), 1531-34
2005
25
80. 3Studies on the Development of
4Taste Masked Suspension of
. Chloroquine
81. 3Synthesis of 3-Oxo-4-aza-53System from (25R)-3-oxo-A. norspristone
82. 3QSAR Study by Fujita-Ban of
2Some Substituted α,β-Diaryl
. Five Membered Heterocyclic
as COX-1/COX-2 Inhibitors
83. 3New Azasteroidal
1Neuromuscular Blocking Agent
. Possessing Acetylcholine-like
Moiety in Ring A
84. 3Crystal Forms of Nimesulide-A
0Sulfonanilide(NSAID)
.
85. 2Phosphite Deoxygenation of
9Steroidal[3,4-c] and [16,17-c]
. furazan N-oxides
86. 2Chemical and Pharmacological
8Studies on Fixed Oil of Ocimum
. sanctum
87. 2Synthesis of some Novel
7Hetrocyclic Steroids by
. Beckmann Rearrangement
88. 2Naproxen-L-Phenylalanine
6alkyl ester prodrugs: Synthesis
. and Biological Evaluation
89. 2Synthesis and Biological
5Activity of [16,17-c]furaxano. 5α/β-androstano[3,4c]furazans
90. 2Synthesis and Biological
4Activity of Steroidal[3,4. d]triazoles
V.Chandibhamar,
M.R.Yadav and R.S.R.
Murthy
M.R.Yadav, M.M.Ganesh,
R.Giridhar, M.Kumar
Bull. Chim. Farmac.,
143, 377-382
2004
Asian J. Chem.,
16(2), 1027-1033
2004
K.P.Sarathy, R.Giridhar
and M.R.Yadav
Indian Drugs, 40(1),
9-18
2003
M.R.Yadav, R.Giridhar,
S.P.Rathod, M.Mahatma
and P.M.Sabale
Indian J. Chem., 40B, 2001
1177-1185
A.Kapoor, D.K.Majumdar
and M.R.Yadav
Indian J. Chem., 37B, 1998
372-375
D.P.Jindal, R.Gupta,
I.B.Singh, J.S.R.A.Sharma
and M.R.Yadav
S.Singh, D.K.Majumdar
and M.R.Yadav
Indian J. Chem., 36B, 1997
14-16
D.P.Jindal, R.Gupta,
R.Kaushal, I.B.Singh and
M.R.Yadav
V.K.Sharma, M.R.Yadav
and S.Singh
Indian J. Chem., 35B, 1996
775-778
D.P.Jindal, R.Gupta,
I.B.Singh, N.Sharma and
M.R.Yadav
Indian J. Chem., 34B, 1995
560-562
A.K.Verma, R.Gupta,
M.R.Yadav and D.P.Jindal
Indian J. Chem., 34B, 1995
215-220
91. 2Wolf-Kishner reduction
3Studies on Steroidal
. hydrazoneoximes
92. 2Studies in Synthesis of Some
A.K.Verma, N.Sharma,
M.R.Yadav D.P.Jindal
J. Indian Chem.
Soc.,71, 283-284
M.R.Yadav
Indian J. Chem., 32B, 1993
Indian J. Exp.
Biol.,34, 1212-1215
Inflamm. Res.,44,
S287-S287
1996
1995
1994
26
93.
94.
95.
96.
97.
98.
99.
100.
101.
102.
103.
104.
2Potential Neuromuscular
. Blocking Azasteroids
2Studies in 17a1Azasteroidal[3,2-c]furoxans
.
217-methyl-3β-pyrrilidino-170aza-D-homo-5-androstene
. dimethiodide
1Certain Steroidal[3,4-c]-1’,2’,5’
9oxadiazoles
.
15 α-Androstano[3,4-c][16,178c]bisfuroxan
.
1Hetroaromatic-ring fused
7steroids
.
1Synthesis and Study of
6Azatriterpenes
.
1Novel Camphorimideoximes
5and Camphorquinone dioxime
.
1Studies in Steroidal[3,4-c]41’,2’,5’ oxadiazoles
.
1Synthesis and Study of
3Heterocyclic Oxadiazoles
.
15-Pregneno[3,4-c]-1’,2’,5’
2oxadiazoles
.
12’-Phenyl;-5 α-pregnano[3,41c]-1’,2’,5’-triazole-20-one
.
1Synthesis and Anti0inflammatory Activity of Some
. Camphor Analogues
746-753
D.P. Jindal, J. Abraham and Indian J. Chem., 31B, 1992
M.R. Yadav
664-666
M.R.Yadav
Indian J. Chem., 31B, 1992
1-2
M.R.Yadav and D.P.Jindal
Indian J. Chem., 30B, 1991
473-476
D.P.Jindal and M.R.Yadav
Indian J. Chem., 30B, 1991
515-516
M.R.Yadav and D.P.Jindal
Indian J. Pharm. Sci.,
52, 42-42
1990
M.S.Y.Khan, S.Ahmed,
M.R.Yadav and D.P.Jindal
J. Indian Chem.
Soc.,67, 330-331
1990
V.K.Kapoor, K.K.Chagti,
M.R.Yadav and D.P.Jindal
Indian J. Chem., 29B, 1990
971-972
M.R.Yadav, J.Abraham
and D.P.Jindal
Indian J. Chem., 29B, 1990
26-28
D.P.Jindal, I.B.Singh and
M.R.Yadav
Indian J. Pharm. Sci.,
51, 153-153
M.R.Yadav, D.P.Jindal and
H.Singh
Indian J. Chem., 27B, 1988
205-208
D.P.Jindal, N.Sharma and
M.R.Yadav
Indian J. Pharm. Sci.,
49, 116-116
1987
V.K.Kapoor, K.K.Chagti,
M.R.Yadav and D.P.Jindal
Indian J. Pharm. Sci.,
49, 116-116
1987
1989
27
105. 017-Oxo-17a-aza-D-homo-5 α9androstano[3,4-c]-1’,2’,5’
. oxadiazole N-oxide
106. 0Pregneno[3,4-c]-1’,2’,5’
8oxadiazol-20-ones
.
107. 017α-preg-20-yno[3,4-c]-1’,2’,5’
7oxadiazol-17-ols
.
108. 0Steroidal 5-eno[3,4-c]-1’,2’,5’
6oxadiazoles
.
109. 05-Pregnenol[3,4-c]-1’,2’,5’
5oxadiazoles
.
110. 0Substituted thiocarbonimidic
4diamide Derivatives and Their
. Antihistaminic properties
111. 017 Hydroxy-5ξ,17α-preg-203yno[3,4-c]-1’,2’,5’ oxadiazoles
.
112. 0Steroidal [3,4-c]-1’,2’,5’
2oxadiazoles
.
D.P.Jindal, J.Abraham and
M.R.Yadav
Indian J. Pharm. Sci.,
49, 115-115
1987
D.P.Jindal, M.R.Yadav,
R.K.Sharma,V.R.Agrawal
and H.Singh
H.Singh, M.R.Yadav and
D.P.Jindal
Indian J. Chem., 26B, 1987
100-103
D. Paul, M.R.Yadav and
H.Singh
Indian J. Pharm. Sci.,
48, 108-108
1986
H.Singh, D. Paul,
M.R.Yadav R.K.Sharma
and V.R.Agrawal
S.N.Pandya, M.R.Yadav
and K.Gupta
Indian J. Pharm. Sci.,
47, 55-55
1985
113. 05ξ-Pregnanol[3,4-c]-1’,2’,5’
1oxadiazoles
.
Indian J. Chem., 26B, 1987
95-99
Eastern
Phamacist,28, 211212
H.Singh, M.R.Yadav and D. Indian J. Chem., 2B,
Paul
1158-1158
1985
H.Singh, M.R.Yadav,
S.P.Garg, R.K.Sharma and
D. Paul
Heterocycles,23,
2929-2938
1985
D. Paul, M.R.Yadav,
R.K.Sharma, V.R.Agrawal
and H.Singh
Indian J. Chem, 24B,
1-1
1985
1985
List of Reviews:
Sr. No.
1.
2.
Name of Journal,
Vol. & Page No.
Title of the Review
Author(s)
Developing steroidal
aromatase inhibitors-an
effective armament to win
the battle against breast
cancer
Management of
Hypertension – Journey from
Mange Ram Yadav,
Mahesh A. Barmade, Riyaj
S. Tamboli, Prashant R.
Murumkar
Eur. J. Med. Chem.,
105, 1-38
Prashant P. Naik. Vijay A.
Pawar, Rajani Giridhar,
Current Clinical
Pharmacology
Year
2015
2015
28
3.
Single Drug Therapy to
Multitargeted Ligand
Therapy: A Clinical Overview
A comprehensive patents
review on cannabinoid 1
receptor antagonists as antiobesity agents
Discovery of Anti-malarial
Agents Through Application
of In silico Studies
4.
5.
6.
7.
8.
9.
Prospective therapeutic
agents for obesity: Molecular
modification
approaches of centrally and
peripherally acting selective
cannabinoid
1 receptor antagonists
Nitrogen containing
privileged structures and
their solid phase
combinatorial synthesis
Mange Ram Yadav
10.2174/15748847)
Mayank Kumar Sharma,
Prashant R. Murumkar,
Mahesh A. Barmade,
Rajani Giridhar, Mange
Ram Yadav
Mahesh A. Barmade,
Prashant R. Murumkar,
Mayank Kumar Sharma,
Kaushik P. Shingala, Rajani
R. Giridhar and Mange
Ram Yadav
Mayank Kumar Sharma,
Prashant R. Murumkar,
Ashish M. Kanhed, Rajani
Giridhar, Mange Ram
Yadav
Expert Opin Ther
Pat., 25(10), 1093116
Amit Verma, M.R.Yadav,
Rajani Giridhar, Navnit
Prajapati, Avinash C.
Tripathi and Shailendra K.
Saraf
Uttam Mane and
M. R. Yadav
Comb Chem High
Throughput
Screen.16(5),
345-93.
Falcipain-2 inhibitors as
potential therapeutics for
resistant strains of malaria: a
patent review
Novel methods and strategies Prashant Murumkar, R.
in the discovery of TACE
Giridhar and M. R. Yadav
Inhibitors
ACAT Inhibitors: The Search
for Novel Cholesterol
Lowering Agents
10.
Novel TACE inhibitors in drug
discovery: A review of
patented compounds
11.
Gemini Amphiphiles: A Novel
(DOI:
Combinatorial
Chemistry & High
Throughput
Screening, 18, 151 -
2015
187
Eur. J. Med. Chem.
79, 298-339
2014
Expert Opin Ther
Pat., 23(2), 165-187
Expert Opin Drug
Discov., 8(2),
157-181
Palash Pal, Hardik Gandhi, Mini-Reviews in
Rajani Giridhar and Mange Med. Chem., 13,
Ram Yadav
1195-1219
Murumkar, P.R.,
DasGupta, S., Chandani,
S.R., Giridhar, R. M.R.
Yadav
Mukesh Kumar, Kaustub
2015
Expert Opinion on
Therapeutic Patents
20 (1), pp. 31-57
Critical Reviews™ in
2013
2013
2013
2013
2010
2010
29
12.
Class of
Nonviral Gene Delivery
Vectors
Jinturkar, M.R. Yadav,
& A.N. Misra
Therapeutic Drug
Carrier Systems,
27(3), 237-278
Angiotensin II Receptor Type
1 (AT1) Selective Nonpeptidic
Antagonists - A Perspective
Prashant Naik, Prashant
Murumkar, Rajani Giridhar
and M. R. Yadav
P.K. Halen,
P.R. Murumkar, R.
Giridhar and M. R. Yadav
Bioorganic and
Medicinal Chemistry,
18, pp. 8418-56.
Prodrug Designing of NSAIDS
13.
14.
15.
16.
Current perspective of TACE
inhibitors: A review
The search for potent, small
molecule NNRTIs: A review
Recent Advances in Selective
α1-Adrenoreceptor
Antagonists as
Antihypertensive Agents
17.
Inhibition of
farnesyltransferase: A
rational approach to treat
cancer?
18.
Current Scenario of 1,4Diazepines as potent
biomolecules- A mini review
19.
Protease Inhibitors as
Potential Drugs
20.
21.
22.
Intellectual Property- Related
Issues
The Multifaceted Profile of
Cox-2 Enzyme and Emerging
Therapeutic Uses of Cox-2
Inhibitors
Some Interesting Facets of
Chiral Drugs
DasGupta, S Murumkar, P.
R., Giridhar, R., M.R.
Yadav
Mini-Reviews in
Med. Chem., (9),
124-139
Bioorganic and
Medicinal Chemistry
Chem. (17) 444-459
Bioorganic and
Medicinal Chemistry
17 (16), pp. 57445762
K. S. Jain, J. B Bariwal, M. Bio-org. Med.
Kathiravan, M. S Phoujdar, Chem., (16) 4759R. S Sahne, B. S Chauhan, 4800
A. K Shah, M. R. Yadav
Prajapati, D.G.,
Ramajayam, R., M.R.
Yadav, Giridhar, R.
D.S. Puntambekar,
R.Giridhar, M.R. Yadav
J. Enz. Inh. Med.
Chem.,22, 127-40
Mini-Reviews in
R .Ramajayam, R. Giridhar,
Med. Chem., 7 (8)
M.R.Yadav
793-812
M.R.Yadav
M.R.Yadav
Hetal B. Prajapati, R.
Giridhar and M.R.Yadav
Halen P.K., Giridhar R. and
Yadav M.R
Chronicle
Pharmabiz, March
21, 65-68
Pharma Glimpses,
15-17
Indian J. Pharm. Sci.
65, 557-564
Indian Drugs, 39,
457-464
2010
2009
2009
2009
2008
2007
2007
2006
2006
2003
2002
30
23.
24.
Industry- Academy
Interaction- Need of the Hour
RU-486: A Multifaceted
Antihormonal Drug
Mange Ram Yadav
Mange Ram Yadav and
Manoj Kumar
25.
Antimicrobial Agents in
Pharmaceutical Products
Dharam Paul Jindal and
Mange Ram Yadav
26.
Role of Antioxidants in
Pharmaceutical Products
Dharam Paul Jindal and
Mange Ram Yadav
Assoc. Pharm.
Technocrt., 73-74
Indian Drugs, 29,
387-394
Eastern Pharmacist,
29, 47-60
Indian Drugs, 22, 117
1994
1992
1986
1985
Patents:
Sr.
No.
1.
2.
3.
4.
5.
Title of the Patent
Author(s)
3-Benzazepin-2-one derivatives as 5HT2C receptor agonists and the process
for their preparation
Yadav M.R.,
Mahesh Shidore,
Jatin Machhi,
Prashant
Murumkar and
Rajani Giridhar
Yadav M.R.,
Kumar M. and
Misra A.N.
Gemini amphiphile based formulations
and their method of preparation for
polynucleotide delivery
Benzimidazolyl, benzoxazolyl and 2pyridylimidazolyl derivatives as
potential anticancer agents and the
process for their preparation
Piperazinylalkyl esters and the salts of
some NSAIDs for improved
percutaneous delivery and the process
for their preparation
Quaternary ammonium 8-methyl8azabicyclo[3.2.1]octan-3-yl esters as
muscarinic receptor antagonists and
their method of preparation
Registration/Application
No., Year
Indian patent,
Appl./959/MUM/2015
Indian patent,
Appl./1828/MUM/2013
Yadav M.R.,
Srinivasan B.P.,
Yogishkumar H.
and Pawar V.A.
Yadav M.R. and
Pawar V.A.
Indian patent,
Appl./192/MUM/2013
Yadav M.R.
Pawar V.A. and
Huchanna Y.K.
Indian patent,
Appl.//MUM/2012
Indian patent,
Appl.//MUM/2012
31
6.
7.
8.
9.
10.
11.
12.
13.
14.
4-Amino-2-piperazinoquinazoline
derivatives as potential
antihypertensive agents and their
method of preparation
2-Substituted 4-amino-6,7dimethoxyquinazolines as dual acting
antihypertensive agents and the
process for their preparation
Benzazepine derivatives and the
process for their preparation
M.R.Yadav,
P.R.Naik and
R.Giridhar
Indian Patent,
Appl./253/MUM/2012
M.R.Yadav,
R.Giridhar and
Prashant P. Naik
Indian Patent,
Appl./3412/MUM/2011
(Under Physical
Examination)
Indian Patent,
Appl./3480/MUM/2010
4-(Arylthia)-16 –cyano-17-oxo-4androsten-3-ones, reduced derivatives
17–ols and the process for their
preparation
Some polar diquaternary Gemini
amphiphiles and the process for their
preparation
R. Giridhar,
M.R.Yadav and A.
Verma
M.R.Yadav, P.M.
Sabale,
P.R.Murumkar
and R.Giridhar
M.R.Yadav, M.
Kumar and
A.N.Misra
1-Aryl-2-imidazolidinones as potential
TACE Inhibitors and the process for
their preparation
M.R.Yadav,Shirsh
endu DasGupta
and R.Giridhar
Indian patent,
Appl./ 2469/Mum/2008
Trisciprofloxacinatobismuth and the
Process for its Preparation
M.R.Yadav,
Anwar R. Shaikh
and R. Giridhar
M.R.Yadav,
R.Giridhar and
Hetal B. Prajapati
Indian Patent,
Appl./1449/Mum/2007
M.R.Yadav,
R.Balaraman and
R.Giridhar
D.P.Jindal and
M.R.Yadav
Indian Patent,
No. 191025
dated 24.09.2001
A Process for the preparation of 3-[o-mp- Mono/Disubstituted phenyl]-4-[o/psubstituted phenyl] Furazans and
Furoxans’.
A Process for the Preparation of
Biscurcumino-oxvanadium(iv)
A Process for the Preparation of 17α15. dMethyl-4-oxo-5α-androstano[2,3ad]pyrazol-17-ol
16.
17.
A process for the Preparation of 4,17βDihydroxy-3-oxo-4-androstene-2ξcarbonitrile17-acetate
A Process for the Preparation of 17αMethyl-4-androstano[3,2-c]isoxazol-
Indian patent,
Appl./ 3309/Mum/2010
(Under Physical
Examination)
Indian patent,
Appl./ 2633/Mum/2010
Indian Patent,
Appl./109/Mum/2004
D.P.Jindal and
M.R.Yadav
Indian Patent,
Appl.1041/Del/94,
Chem.Abstr.,124,1996,90
95W
Indian Patent,
Appl.1041/Del/88
D.P.Jindal and
M.R.Yadav
Indian Patent,166480,
1986, Appl.999/Del/86
32
4,17-diol
BOOK/ BOOK CHAPTER
1. Mange Ram Yadav, Prashant R. Murumkar and Vishal Zambre, “Advances in Studies on
Collagenase Inhibitors”, Advances in Studies on Matrix Metalloproteinase Inhibitors
(Springer Basel AG), Experientia Supplementum Volume 103, 2012, pp 83-135.
2. Mange Ram Yadav, Shirshendu Das Gupta, Prashant R. Murumkar and Rajani Giridhar,
“Small Molecule Selective TACE Inhibitors: Potential Therapeutic Agents”, NOVA
international publication, Volume 3, USA, 2010,
3. Kanchan Kohli and Mange Ram Yadav, Pharmaceutical Chemistry-II, Piyush Publications,
Delhi, 1995.
4. Harkishan Singh, Dharam Paul Jindal, Mange Ram Yadav and Manoj Kumar,
“Heterosteroids in Drug Research” in Progress in Medicinal Chemistry, G.P. Ellis and G.B.
West, Eds., Elsevier/ North-Holland Biomedical Press, Amsterdam, Vol. 28, 1991.
SCIENTIFIC PAPER PRESENTATIONS
International Presentations:
1. Mange Ram Yadav, “Green synthesis and antiplatelet potential of diaryl 1,2,4-triazines”
during 23-25th Jan. 2014 at NIPiCON-2014, Nirma Institute of Pharmacy, Ahmedabad,
Gujarat.
2. Mange Ram Yadav, “Synthesis of quinazoline based cyclic guanidines as potent AchE and
BuchE antagonist for AD” during 23-25th Jan. 2014 at NIPiCON-2014, Nirma Institute of
Pharmacy, Ahmedabad, Gujarat.
3. Mange Ram Yadav, “Pharmacological approaches for evaluating 5HT2c agonistic potentials
of some novel ligands using murine models” during 16-18th Dec. 2013 at 46th Annual
conference of Indian Pharmacological society, NIMHANS Bangalore, India
4. Mange Ram Yadav, “Modulatory effect of MCR-1329, a novel quinazoline derivative on
DOCA-salt induced hypertension in rats” during 16-18th Dec. 2013 at 46th Annual
conference of Indian Pharmacological society, NIMHANS Bangalore, India
5. Mange Ram Yadav, “In vitro pharmacological evaluation of some novel benzazepine
derivatives for their dopaminergic potential” during 16-18th Dec. 2013 at 46th Annual
conference of Indian Pharmacological society, NIMHANS Bangalore, India
6. Mange Ram Yadav, “A non-radiometric method for estimation of cholesteryl esters”
during 2-5th June 2013 at 81st Annual Conference Of the European Atherosclerosis
Society, Lyon, France.
7. Mange Ram Yadav, “Synthesis and Evaluation of a Series of 3-Benzazepine Derivatives as
Anxiolytics and Antidepressants” during 18-20th Jan. 2013 at NIPiCON-2013, Nirma
Institute of Pharmacy, Ahmedabad, Gujarat.
33
8. Mange Ram Yadav, “Synthesis , Docking and antiplatelet potential of 1,3-benzooxazin-4ones and their diamides” during 18-20th Jan. 2013 at NIPiCON-2013, Nirma Institute of
Pharmacy, Ahmedabad, Gujarat
9. Mange Ram Yadav, “Design and synthesis of triaryl imidazoles as antiplatelet agents”
during 18-20th Jan. 2013 at NIPiCON-2013, Nirma Institute of Pharmacy, Ahmedabad,
Gujarat
10. Mange Ram Yadav, “Searching for new isosterically modified analogues of imatinib to
overcome resistance in chronic myelogenous leukemia” during 26-29th June 2012 at 13th
Tetrahedron Symposium, Amsterdam, Netherlands.
11. Mange Ram Yadav, “Design, Synthesis and Bioactivity of Substituted Pyrimidine as PTP1B
Inhibitors” during 9-11th Jan. 2011 at CHARUSAT, University of Science and Technology,
Chhanga, Gujarat.
12. Mange Ram Yadav, “Synthesis and Neurotropic activity of 3-Benzazepine derivatives”
during 22-24th Oct. 2010 at University College of Pharm. Sciences, Warangal, Andhra
Pradesh.
13. Vishal P Zambre, Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav DNA Gquadruplex ligands – anthraquinones and acridones: 3D - QSAR studies for a quantitative
prediction of the telomerase inhibitory activity based on comparative molecular similarity
indices analysis, 239th ACS Annual National Meeting, 2009 San Francisco, CA, USA.
14. Vishal P Zambre, Prashant Murumkar, Rajani Giridhar and Mange Ram Yadav, “3DQSAR
studies on DNA G-quadruplex interactive agents as telomerase inhibitors” 17th European
Symposium on QSAR in “Omics” and Systems Biology during 21-26 Sept. 2008 at Uppsala,
Sweden.
15. Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav Identification of ligand
feature essential for TACE inhibitors by pharmacophore modeling. 237 th ACS Annual
National Meeting, 2009, Salt lake City, Utah, USA.
16. Vishal P Zambre Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav, Ligandbased molecular modeling study on DNA G-quadruplex mediated telomerase inhibitors: A
3D-QSAR CoMFA, CoMSIA approach. 237th ACS Annual National Meeting, 2009, Salt lake
City, Utah, USA.
17. Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav 3D-QSAR studies on
Benzodiazepine Hydroxamates as Tumor Necrosis Factor- alpha Converting Enzyme
Inhibitors, 235th ACS Annual National Meeting, 2008, New Orleans, LA, USA.
18. Bishram Singh Chouhan, Rajani Giridhar and Mange Ram Yadav, Microwave Assisted
Synthesis of Substituted 4-Quinazolones, Medchem. India, 2007, Select Biosciences (UK),
Hyderabad, India.
34
19. R.Ramajayam, Rajani Giridhar and Mange Ram Yadav Design, Synthesis and Evaluation of
2,3-diaryl-1-4-diazepinesas Potential Anti-Proliferative Agents, 230th ACS Annual National
Meeting, Washington DC,USA.
20. Devendra Puntambekar, Rajani Giridhar and Mange Ram Yadav, Development of
Predictive CoMFA and CoMSIA Models for Alkoxylated and Hydroxylated Chalcones as AntiMalarial Agents, 230th ACS Annual National Meeting, Washington DC, USA.
21. Devendra Puntambekar, Rajani Giridhar and Mange Ram Yadav, Insight into the Structural
Requirements of Farnesyltransferase Inhibitors as Potential Anti-tumor Agents Based on
3D-QSAR, CoMSIA and CoMFA models, 233th ACS Annual National Meeting, Chicago, USA.
22. Bishram Singh Chouhan, Rajani Giridhar and Mange Ram Yadav Design and Synthesis of
Some Multitargeted Ligand as Potential Anti-hypertensive Agents, 234th ACS Annual
National Meeting, Boston, USA.
23. Vijay Kumar Sharma, Mange Ram Yadav and Surender Singh, Naproxen-L-phenylalanine
Alkyl Ester Prodrugs: Synthesis and biologicsl evaluation, Second World Congress on
Inflammation, Brighton, U.K., Sept. 17-22, 1995, Abstract No. W19/5.
24. Anjali Bhasin, D.K. Majumdar and Mange Ram Yadav, Dissolution characteristics of
diclofenac crystals obtained from various solvents, International Symposium on Recent
Trends in Pharmaceutical Sciences, Ootacamund, Feb 18-20, 1995, Abstract No. D27.
25. S. Bhatia, Mange Ram Yadav, M. S. Y. Khan, A. Kar and S. Singh, Synthesis and CNS Profile
of some 2-phenylindole derivatives, International Symposium on Recent Trends in
Pharmaceutical Sciences, Ootacamund, Feb 18-20, 1995, Abstract No. B43.
26. Harkishan Singh, Mange Ram Yadav and Dharam Paul, Steroidal [3,4-c]-1’,2’,5’-Oxadiazoles
as potential bioactive molecules, in 10th International Congress of Heterocyclic Chemistry,
University, University of Waterloo, Canada, 11-16th Aug. 1985, Abstract No. P9-284.
National:
1. Dushyant Patel, Nirav Patel, Rajani Giridhar, Mange Ram Yadav, “Synthesis and biological
evaluation of some vicinyl diaryl thiazole urea derivatives as potential ACAT inhibitors”
during 7th Feb. 2014 in “Pharma-FEST- 2014” at , Parul Institute of Pharmacy, Baroda.
2. Chetna Dhakada, Navneet Prajapati, Jatin Machi, Rajani Giridhar, Mange Ram Yadav,
“Synthesis of cyclic guanidines as potent cholinesterase inhibitors for AD” during 7th Feb.
2014 in “Pharma-FEST- 2014” at , Parul Institute of Pharmacy, Baroda
3. Neetesh Agrawal, Virendra Rathwa, Prashant Naik, Prashant R Murumkar, Rajani Giridhar
Mange Ram Yadav, “Synthesis and evaluation of a series of 6,7-dimethyl-2-(4arylsubstituted piperazine-1-yl quinazolin-4-amine) derivatives as multitargeted ligands as
potential antihypertensive agents ” during , 18th Jan. 2014 in “3rd Annual National
Convention Of Pharmacy Professionals” at Faculty of Pharmacy, D.D. University Nadiad,
Gujarat.
35
4. Mahesh Shidore, Jigar Thanki, Jatin Machi, Prashant R. Murumar, Rajani Giridhar Mange
Ram Yadav, “Synthesis and biological evaluation of 4,5-dihydro-1-methyl-1-benzazepin-2one derivatives as 5-HT2c receptor agonist” during , 18th Jan. 2014 in “3rd Annual National
Convention Of Pharmacy Professionals” at Faculty of Pharmacy, D.D.University Nadiad,
Gujarat.
5. Virendra Rathwa, Vaishali Desai, Neetesh Agrawal, Prashant Naik, Prashant R Murumkar,
Rajani Giridhar, Mange Ram Yadav, “Synthesis and evaluation of series of 6,7-dimethoxy2-(4-substituted piperazine-1yl)quinazoline-4-amine derivatives as dual acting potential
antihypertensive agents” during 20-22 Dec. 2013 in “65th Indian Pharmaceutical Congress”
at Amity University, Delhi.
6. Jigar Thanki, Mahesh Shidore, Jatin Machi, Prashant R. Murumar, Rajani Giridhar, Mange
Ram Yadav, “Synthesis and biological evaluation of 4,5-dihydro-1- methyl-1(H)benzo(d)azpine-2(3H)- one derivatives as 5-HT2C receptor agonist” during 20-22 Dec.
2013 in “65th Indian Pharmaceutical Congress” at Amity University, Delhi.
7. Niral Patel, R.S. Tamboli, A.M. Ravani, Mange Ram Yadav, Rajani Giridhar “Synthesis and
antiplatelet activity of some 2,4,5-triaryl imidazoles” during 20-22 Dec. 2013 in “65th Indian
Pharmaceutical Congress” at Amity University, Delhi.
8. Mayank Kumar Sharma, Uttam Mane, Prashant R. Murumar, D. Sahal, Rajani Giridhar,
Mange Ram Yadav, “Synthesis and biological evaluation of some novel pyrido[1,2a]pyrimidin-4-ones as antimalarial agents” during 20-22 Dec. 2013 in “65th Indian
Pharmaceutical Congress” at Amity University, Delhi.
9. Mayank Kumar Sharma, Prashant R. Murumkar, Rajani Giridhar, Mange Ram Yadav,
“Virtual screening based discovery of lead molecules as selective TACE inhibitors” during ,
20-22 Dec. 2013 in “65th Indian Pharmaceutical Congress” at Amity University, Delhi.
10. Dushyant Patel, Karan Samyani, Navneet prajapati, Rajani Giridhar, Mange Ram Yadav,
“Palladium–catalysed α-Methylation of carbonyl compounds using dimethylformamide as
methylating agent” during , 20-22 Dec. 2013 in “65th Indian Pharmaceutical Congress” at
Amity University, Delhi.
11. Sujata Salecha, Amit Verma, Navneet Prajapati, Jatin Machi, Rajani Giridhar, Mange Ram
Yadav, “Synthesis of benzazepine derivatives using palladium catalyst and their potential
as dopamine receptors modulators” during 22-23rd, Feb 2013 in “Pharmarendezvous” at
Sumandeep college of Pharmacy, Vadodara.
12. Anand Mantri, Viral Dhaluk, Pradeep Mali, Mange Ram Yadav, Rajani Giridhar “Synthesis of
Thiazolidin-4-ones as potent PTP1B inhibitors” during 26-27th Feb. 2013 in “Approaches in
Drug Discovery” at Pharmacy Department, The M.S. University of Baroda, Vadodara.
13. Neetesh Agrawal, Vaishali Desai, Rajani Giridhar, Mange Ram Yadav, “Design and synthesis
of some multi-targeted ligands as potential antihypertensive agents” during 26-27th Feb.
2013 in “Approaches in Drug Discovery” at Pharmacy Department, The M.S. University of
Baroda, Vadodara.
36
14. Palasha Pal, Satish Balda, Rajani Giridhar, Mange Ram Yadav, “Synthesis of compounds
possessing vicinal diaryl heterocyclic urea derivatives as an ACAT inhibitors” during 26-27th
Feb. 2013 in “Approaches in Drug Discovery” at Pharmacy Department, The M.S. University
of Baroda, Vadodara.
15. Vijay Pawar, Pardip Patel, Rajani Giridhar, Mange Ram Yadav, “Design and development of
non-viral vector for efficient transfection of pDNA” during 26-27th Feb. 2013 in
“Approaches in Drug Discovery” at Pharmacy Department, The M.S. University of Baroda,
Vadodara.
16. Sujata Salecha, Amit Verma, Anshuman Sinha, Ashish Kanhed, Navnit Prajapati, Mange
Ram Yadav, Rajani Giridhar “Novel quinazolinone based cyclic guanidines as potent
neuroprotective agents” during 26-27th Feb. 2013 in “Approaches in Drug Discovery” at
Pharmacy Department, The M.S. University of Baroda, Vadodara.
17. Mange Ram Yadav, “In vitro seretonergic potential of some novel ligands” during 16 Dec.
2011 at 63rd Indian Pharmaceutical Congress, MCPS, Manipal University, Manipal.
18. Mange Ram Yadav, “A new bearing on multiple-targeted ligands: α1blockers and AT1R
antagonism” during 16 Dec. 2011 at 63rd Indian Pharmaceutical Congress, MCPS, Manipal
University, Manipal.
19. P. P. Naik, B. S. Chouhan, R. Giridhar and Mange Ram Yadav, Synthesis and cytotoxic
activity of a series of novel 2-substitutedaryl 4-amino- 6,7-dimethoxyquinazolines, 61st
Indian Pharmaceutical Congress, Ahmedabad, Dec. 2009 Abstract No. B-259
20. D.G. Prajapati, A. V. Mantri, R. Giridhar, and Mange Ram Yadav, Synthesis of Allyloxy
Substituted 4,6-diarylpyrimidines as Potential HIV Reverse Transcriptase Inhibitors, 61st
Indian Pharmaceutical Congress, Ahmedabad, Dec. 2009 Abstract No. B-253
21. Dharmendrasinh A. Baria, Prafulla M. Sable, Rajani Giridhar, Mange Ram Yadav, D-ring
modified hetero-steroids as potential aromatase inhibitors, 61st Indian Pharmaceutical
Congress, Ahmedabad, Dec. 2009. Abstract No. B-232
22. D.G. Prajapati, R. S. Tamboli, R. Giridhar, and Mange Ram Yadav, Assessment of Antiplatelet activity of 2-aminopyrimidines, 61st Indian Pharmaceutical Congres Ahmedabad,
Dec, 2009. Abstract No. B-215
23. Prafulla M. Sabale, Umang Shah, Rajani Giridhar and Mange Ram Yadav Design and
Synthesis of Novel Steroidal Aromatase Inhibitors, 61st Indian Pharmaceutical Congress,
Ahmedabad, Dec. 2009. Abstract No. B-205
24. Prashant R Murumkar, Sneha R Chandani, Rajani Giridhar and Mange Ram Yadav,
“Pharmacophore alignment based CoMFA and CoMSIA studies for Tumor Necrosis Factor
Alpha Converting Enzyme Inhibitors” presented in 61st Indian Pharmaceutical Sciences to
be held at Ahmedabad in 2009. Abstract No. B-59
25. Vishal P Zambre Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav,
“Comparative Molecular Similarity Indices Analysis of DNA G-Quadruplex Mediating
37
Telomerase Inhibitors, 61st Indian Pharmaceutical Congress, Ahmedabad, Dec. 2009
Abstract No. B-58
26. Prashant R. Murumkar, Vishal P. Zambre, Rajani Giridhar, Mange Ram Yadav, “Structure
Guided 3D-QSAR: A Useful Approach for Designing of TACE Inhibitors” in 60th Indian
Pharmaceutical Sciences at New Delhi in Dec. 2008
27. Prashant R. Murumkar, Rajani Giridhar, Mange Ram Yadav “Development of predictive 3DQSAR CoMFA and CoMSIA Models for-aminohydoxamic acid-derived TNF-converting
enzyme inhibitors” in 59th Indian Pharmaceutical Sciences at Varanasi on 21st Dec. 2007.
28. Ramajayam R, Rajani Giridhar and Mange Ram Yadav, ‘2,3-substituted diaryl-6,7-dihydro5H-1,4-diazepine as potential medicinal agents’ 57th Indian Pharmaceutical Congress,
Hyderabad, Dec. 02 to 04 2005, Abstract no. BP-54
29. A.K.Shinde, Rajani Giridhar, Robert Menard, Mange Ram Yadav, ‘Synthesis and Evaluation
of dipeptide nitrites as selective cathepsin-L inhibitors.’ 57th Indian Pharmaceutical
Congress, Hyderabad, Dec. 02 to 04 2005, Abstract no. B-16
30. Mange Ram Yadav, D.S.Puntambekar, K.P. Sarathi, S. vengurlekar and Rajani Giridhar,
‘Quantitative Structure Activity Relationship studies of diarylimidazoles as selective COX-II
inhibitors’ 56th Indian Pharmaceutical Congress, Kolkata, Dec. 03 to 05 2004, Abstract no.
BP-39
31. V. Alagarsami, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis and Pharmacological
investigation of some novel 1,2,4-triazoloquinazoline-5(4H)-ones as antihistaminic agents’
56th Indian Pharmaceutical Congress, Kolkata, Dec. 03 to 05 2004, Abstract no. B-11
32. H.B. Prajapati, Shrikant T. Shirude, Rajani Giridhar, R.Balaraman, A. Parmar and Mange
Ram Yadav, ‘Synthesis and evaluation of 3,4-diaryl-1,2,5-oxadiazoles and corresponding NOxides as selective COX-II inhibitors’ 56th Indian Pharmaceutical Congress, Kolkata, Dec. 03
to 05 2004, Abstract no. B-5
33. A.K.Shinde, Rajani Giridhar and Mange Ram Yadav, ‘Cysteine protease inhibitors as
potential anti-malarial drugs.’ 56th Indian Pharmaceutical Congress, Kolkata, Dec. 03 to 05
2004, Abstract no. B-3
34. Dharmendra G. Patel, Rajani Giridhar and Mange Ram Yadav, ‘Fujita Ban modified DeNovo studies on triazolinone-based balanced AT1-AT2 receptor antagonists.’ 55th Indian
Pharmaceutical Congress, Chennai, Dec. 19 to 21 2003, Abstract no. BP-43
35. Datta M. Nimekar, Pathik S Brahmhkshatria, Rajani Giridhar and Mange Ram Yadav, paminophenol and acetylated phenol derivatives of certain commonly available NSAIDs as
more COX-II selective inhibitors, 55th Indian Pharmaceutical Congress, Chennai, Dec. 19 to
21 2003, Abstract no. BP-42
38
36. Shitesh R. Patel, M.M.Ganesh, R.Ramajayam, Rajani Giridhar and Mange Ram Yadav, ‘16ξdimethylamine-3-pyrrolidino-5-androstane dimethiodide as a potential neuromuscular
blocking agents’ 55th Indian Pharmaceutical Congress, Chennai, Dec. 19 to 21 2003,
Abstract no. BP-41
37. P.K.Halen, K.K.Chagti, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis and evaluation of
certain ketorolac analogs with an improved therapeutic profile’ 55th Indian Pharmaceutical
Congress, Chennai, Dec. 19 to 21 2003, Abstract no. BP-40
38. Sudha Vengurlekar, K.P.Sarathi, Rajani Giridhar and Mange Ram Yadav, ‘Structural
requirements for 1,2-diarylimidazole as COX-II inhibitors: Hansch Analysis.’ 55th Indian
Pharmaceutical Congress, Chennai, Dec. 19 to 21 2003, Abstract no. BP-39
39. K.K.Chagti, P.K.Halen, Rajani Giridhar and Mange Ram Yadav, ‘Indomethacin Derivatives
with a better pharmacokinetics and pharmacodynamic profile’ 55 th Indian Pharmaceutical
Congress, Chennai, Dec. 19 to 21 2003, Abstract no. B-36
40. K.K.Chagti, P.K.Halen, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis, Pharmacokinetics
and Pharmacodynamic Profile of beta-amino ester derivatives of Ketoprofen’ 54th Indian
Pharmaceutical Congress, Pune, Dec. 13 to 15 2002, Abstract no. BP-46
41. P.K.Halen, K.K.Chagti, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis and Evaluation of
certain Diclofenac analogues with therapeutic advantage over the parent drug.’ 54th
Indian Pharmaceutical Congress, Pune, Dec. 13 to 15 2002, Abstract no. B-33
42. J.B. Majethia, R. Balaraman, Rajani Giridhar, Mange Ram Yadav, ‘Effect of vanadium and its
complex on the blood glucose and lipid profile of Strptozocin induced diabetic rats’ 53nd
Indian Pharmaceutical Congress, New Delhi, Dec. 21 to 23 2001, Abstract no. E-23
43. K.P.Sarathi, Rajani Giridhar and Mange Ram Yadav, ‘Structural Requirements for COX-1 and
COX-II activity in 3,4-diaryl five membered ring system: Fujita Ban QSAR Approach
Combined with Hansch Analysis ’ 53nd Indian Pharmaceutical Congress, New Delhi, Dec. 21
to 23 2001, Abstract no. B-36
44. P.K.Halen, K.K.Chagti, R.Giridhar and Mange Ram Yadav, ‘Synthesis and Evaluation of Some
Naproxen analogues as dual acting potential drugs.’ 53nd Indian Pharmaceutical Congress,
New Delhi, Dec. 21 to 23 2001, Abstract no. B-22
45. V. Ganeshan, Rajani Giridhar, Hetal Prajapati and Mange Ram Yadav, ‘Polymorphism in
Sparfloxacine: Characterization and Dissolution studies.’ 53nd Indian Pharmaceutical
Congress, New Delhi, Dec. 21 to 23 2001, Abstract no. A-72
46. Revathi R, Rajani Giridhar and Mange Ram Yadav, ‘Studies on some metal complexes of
curcumin’ 52nd Indian Pharmaceutical Congress, Hyderabad, Dec. 1 to 3 2000, Abstract no.
BP-34
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47. Reshmi C.S, Kewal K. Chagti, Rajani Giridhar and Mange Ram Yadav, ‘A New Approach in
the Direction of Therapeutic optimization of NSAIDs- A Study in the Synthesis and Kinetics
of Some NSAIDs Derivatives’ 52nd Indian Pharmaceutical Congress, Hyderabad, Dec. 1 to 3
2000, Abstract no. BP-26
48. Hemalatha B, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis and biological activity of
Gastroprotective analogues of some NSAIDs.’ 52nd Indian Pharmaceutical Congress,
Hyderabad, Dec. 1 to 3 2000, Abstract no. B-11
49. M.M. Ganesh, Hetal B. Prajapati, Rajani Giridhar and Mange Ram Yadav, ‘COX-1 Vs COX-II
selectivity: A Molecular Modeling and QSAR study on 7-tertialrybutyl-2,3-dihydro-3,3dimethylbenzofuran derivatives.’ 52nd Indian Pharmaceutical Congress, Hyderabad, Dec. 1
to 3 2000, Abstract no. B-6
50. Mange Ram Yadav, Rajani Giridhar, Mukesh Mahatma and Prafulla M.Sabale, 4ξ-acetoxy17A, methyl-3ξ-pyrrolidino-17A-aza-D-homo 5α-androstene-dimethiodide: A new
neuromuscular blocking agent. 17th Asian Congress of Pharmaceutical Sciences, Mumbai,
Dec. 10 to 13 1998, Abstract No. IBP-23
51. Anjali Kapoor, D.K.Majumdar and Mange Ram Yadav, Dissolution Characteristics of various
physical forms of Nimesulide. 48th Indian Pharmaceutical Congress, Chennai, Dec. 25th to
27th 1996, Abstract No. AP-25.
52. Nirmal Sharma, Sharda Sushil, A.K. Sharma, Mange Ram Yadav, Sumitra Yadav, Sangeeta
Bhatia, S. Singh, R. Verma and V.K. Sharma, Teaching and reasearch- oriented to team
work, 46th Indian Pharmaceutical Congress, Chandigarh, Dec 28-30, 1994.
53. Surendra N. Pandeya, and Mange Ram Yadav, Synthesis and Biological Activity of α,α'Thiobisformamidine (Amidine) Salts, 46th Indian Pharmaceutical Congress, Chandigarh, Dec
28-30, 1994, Abstract No. B-41.
54. Mange Ram Yadav and Dharam Paul Jindal, 17-Substituted Steroidal [3,4-c]-1',2',5'oxadiazole, 42th Indian Pharmaceutical Congress, Manipal, Dec 28-30, 1990, Abstract No.
A20.
55. Mange Ram Yadav and Dharam Paul Jindal, Heteroaromatic Ring- fused Steroids, 41th
Indian Pharmaceutical Congress, Bombay, Dec 16-18, 1989, Abstract No. A19.
56. Jojy Abraham, Mange Ram Yadav and Dharam Paul Jindal, Certain Heterocycle- fused
Azasteroids, 41th Indian Pharmaceutical Congress, Bombay, Dec 16-18, 1989, Abstract No.
A7.
57. Dharam Paul Jindal, Inder Bir Singh and Mange Ram Yadav, Synthesis and Study of
Heterocyclic Steroids, 40th Indian Pharmaceutical Congress, Calcutta, Dec 26-28 , 1988,
Abstract No. A16.
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58. Dharam Paul Jindal, Jojy Abraham and Mange Ram Yadav, 17a-methyl-17a-aza-D-homo-5αandrostano[3,4-c]-1',2',5'-oxadiazole, 39th Indian Pharmaceutical Congress, Madras, Dec
27-29 , 1986, Abstract No. A15.
59. Dharam Paul Jindal, J.S.R.A. Sharma and Mange Ram Yadav, Synthesis and Study of
Steroidal [3,4-c]-1',2',5'-oxadiazole N-oxide, 39th Indian Pharmaceutical Congress, Madras,
Dec 27-29 , 1986, Abstract No. A14.
60. Vijay K. Kapoor, Kewal Krishan, Mange Ram Yadav and Dharam Paul Jindal Synthesis and
Anti-inflamatory activity of some camphor analouges, 38th Indian Pharmaceutical Congress,
Ahmedabad, Dec 21-23, 1986, Abstract No. A15.
61. Dharam Paul Jindal, Neeta Sharma, and Mange Ram Yadav, 2'-Phenyl-5α-pregnano [3,4-c]1',2',3'-triazol-20-one, 38th Indian Pharmaceutical Congress, Ahmedabad, Dec 21-23, 1986,
Abstract No. A16.
62. Dharam Paul Jindal, Jojy Abraham and Mange Ram Yadav, 17-oxo-17a-aza-D-homo-5αandrostano[3,4-c]-1',2',5'-oxadiazole N-oxide, 38th Indian Pharmaceutical Congress,
Ahmedabad, Dec 21-23, 1986, Abstract No. A5.
63. Dharam Paul, Mange Ram Yadav, and Harkishan Singh, Studies in the Synthesis of Steroidal
5-eno [3,4-c]-1',2',5'-oxadiazole, 37th Indian Pharmaceutical Congress, New Delhi, Dec 2628, 1985, Abstract No. A10.
64. Harkishan Singh, Mange Ram Yadav, and Dharam Paul, Steroidal [3,4-c]-1',2',5'-oxadiazoles
a Potential Bioactive Molecules, 10th International Congress of Heterocyclic Chemistry.
Aug 11-16, 1985, University Of Waterloo, Ontario, Canada, Abstract No. p-284.
65. Harkishan Singh, Dharam Paul, Mange Ram Yadav, Rakesh Kumar Sharma and Vijaykumar
R. Agrawal, 5-Pregnano[3,4-c]-1',2',5'-oxadiazoles, 36th Indian Pharmaceutical Congress,
Bangalore, Feb 9-11, 1985, Abstract No. A15.
66. Harkishan Singh, Mange Ram Yadav, Dharam Paul, Sat Paul Garg and Rakesh Kumar
Sharma, Steroidal [3,4-c]-1',2',5'-oxadiazoles, 35th Indian Pharmaceutical Congress,
Hyderabad, Dec 18-20,1983, Abstract No. A28.
(Dr M. R. Yadav)
10th Dec 2015
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