Program (会议日程安排)
The 10th SINO-US Chemistry Professors Conference
Jinan, China June 15-17, 2014
Date
Program & Venue
June 15
(Sunday)
Chairperson
Hao Fang &
Check-in (舜耕山庄 Shun geng Hill View Hotel)
June 16
Opening Ceremony & Plenary Lectures
(Monday)
(报告厅 Lecture Hall)
8:30-9:00
Opening Ceremony
9:00-9:30
Gunda I. Georg (University of Minnesota)
Small Molecule Probes and Leads for Male Contraception and
Minyong Li
Chairperson
Hao Fang
Binghe Wang
Cancer
9:30-10:00
Take Pictures and Coffee Break
10:00-10:30
Zhongyin Zhang (Indiana University School of Medicine)
Drugging the Undruggable: Therapeutic Potential of Targeting the
Xinshen Ye
Protein Tyrosine Phosphatases
10:30-11:00
Binghe Wang (Georgia State University)
Inducing MDM2 degradation as an anticancer strategy
11:00-12:30
Buffet (重华堂 Chonghua Hall)
Xiaodong Shi
有机化学分会场（会见厅）
June 16
Section I Organic Chemistry
(Monday)
(会见厅 VIP Hall)
13:30-13:50
Xumu Zhang (Wuhan University)
Chairperson
Practical Catalytic Hydrogenation
13:50-14:10
14:10-14:30
Xuefeng Jiang (East China Normal University)
Sulfur Atom Transfer (SAT) Reaction and Synthesis of
Robin
Sulfur-Containing Drugs and Natural Products
Yonggui Chi
Fushun Liang (Northeast Normal University)
Cascade reactions of activated cyclopropanes toward
aza/oxa-heterocycles
14:30-14:50
Robin Yonggui Chi (Nanyang Technological University)
Opportunities with NHC Organocatalysis: Toward New Activation
Modes
14:50-15:10
Ang Li (Shanghai Institute of Organic Chemistry, Chinese
Xumu Zhang
Academy of Sciences)
Total Synthesis of Sespenine: a Bio-Inspired Aza-Prins Approach
15:10-15:30
Coffee Break
15:30-15:50
Weiping Tang (University of Wisconsin)
Rh(I)-catalyzed Tandem Annulation and Cycloaddition for the
Synthesis of Privileged Heterocycles
15:50-16:10
Qing Gu (Shanghai Institute of Organic Chemistry, Chinese
Academy of Sciences)
Enantioselective Synthesis of Planar Chiral Ferrocenes via
Hao Xu
Pd-Catalyzed Direct C-H Bond Arylation
16:10-16:30
Sunliang Cui (Zhejiang University)
Rh(III)-Catalyzed Cyclization and Desymmetrization for
Heterocycles Synthesis
16:30-16:50
Hao Xu (Georgia State University)
Iron-Catalyzed Nitrogen Atom Transfer for Stereoselective
Difunctionalization of Unsaturated Hydrocarbons
16:50-17:10
Bingfeng Shi (Zhejiang University)
Pd-Catalyzed C (sp3)-H Bonds Functionalization: Synthetic Scope
and Application
17:10-17:30
Weiping Tang
Meixin Zhao (East China University of Science and Technology)
Cinchona alkaloid derivatives catalyzed diastereo- and
enantioselective Mannich-type reactions of isocyanoacetates with
ketimines
18:00-20:00
Welcome Dinner Reception (重华堂 Chonghua Hall)
Fengshan
Wang
June 17
Section I Organic Chemistry
Chairperson
(Tuesday)
(会见厅 VIP Hall)
8:00-8:20
Andrew Evans (Queen’s University)
Development of Higher-Order Carbocyclization Reactions:
Emulating Terpene Biosynthesis
8:20-8:50
Yuehai Shen (Kunming University of Science and Technology)
Studies towards convergent total synthesis of autolytimycin
8:50-9:10
Gong Cheng
Weiliang Duan (Shanghai Institute of Organic Chemistry, Chinese
Academy of Sciences)
Palladium-Catalyzed Asymmetric Synthesis of Chiral Phosphorus
Compounds
9:10-9:30
Xiaodong Shi (West Virigina University)
Triazole-Gold and Triazole-Pd Pormoted Catalysis
9:30-9:50
Renhua Fan (Fudan University)
Break and Rebuild the Aromaticity:Application of
Dearomatization Strategy in the Synthesis of Heterocyclic
Compounds
9:50-10:10
Andrew
Evans
Zhihui Shao (Yunnan University)
Structural Unit-Directed Asymmetric Catalysis and Divergent
Total Synthesis
10:10-10:30
Coffee Break
10:30-10:50
Gong Cheng (Penn State University)
Development of Useful C-H Functionalization Chemistry for
Organic Synthesis
10:50-11:10
Hegui Gong (Shanghai University)
Ni-catalyzed reductive coupling of tertiary alkyl halides
11:10-11:30
Shouyun Yu (Nanjing University)
De novo synthesis of nitrogen aromatic compounds enabled by
somophilic isocyanide insertions
11:30-11:50
Shuanhu Gao (East China Normal University)
Total Synthesis of Bioactive Natural Products: Taiwaniaquinol B
and Gracilamine
12:00-13:00
Buffet (重华堂 Chonghua Hall)
Xiaodong Shi
June 17
(Tuesday)
Section I Organic Chemistry
(拱北楼四楼会议室 The 4th Floor Meeting Room, Gongbei
Chairperson
Building)
13:30-13:50
Lei Liu (Shandong University)
Catalytic enantioselective C-H functionalization of heterocycles
13:50-14:10
Jian Xiao (Qingdao Agricultural University)
sp3 C-H functionalization of azarenes under metal free and
catalyst free conditions
14:10-14:30
Zhenghu Xu
Huadong Xu (Changzhou University)
A novel cyclization/aza-Claisen rearrangement cascade initiated
by ketenimine formation: highly efficient synthesis of β-allyl
cyclic amidines
14:30-14:50
Zhenghu Xu (Shandong University)
Tandem Metal Relay Catalysis for Heterocycles
14:50-15:10
Zhenghui Guan (Northwest University)
Synthesis of azaheterocycles via cyclization of enamides and
alkynes
15:10-15:30
Shifa Zhu (South China University of Technology)
Lei Liu
Transition Metal-Catalyzed Generation and Trapping of the
o-QDMs: The Applications in the Diels-Alder reactions
15:30-15:50
Xu Cheng (Nanjing University)
Enantioselective Construction of Chiral Carboniolamide
16:00-16:30
Closing Ceremony
(拱北楼四楼会议室 The 4th Floor Meeting Room, Gongbei
Building)
18:00-19:00
Buffet (重华堂 Chonghua Hall)
Hao Fang
生物有机化学分会场（会谈厅）
June 16
Section II Bioorganic Chemistry
(Monday)
(会谈厅 Meeting Hall)
13:30-13:50
Zhongwu Guo (Wayne State University)
Chairperson
Synthesis and Biological Studies of GPI Anchors and
GPI-Anchored Proteins
13:50-14:10
Yu Rao (Tsinghua University)
Developing Novel Chemical Probes for Early Drug Discovery
14:10-14:30
Xiangming
Guan
Zheng Yin (Nankai University)
Discovery of Enterovirus 71 3C Protease Inhibitors
14:30-14:50
Xiangming Guan (South Dakota State University)
A combined inhibition of lactate dehydrogenase and pyruvate
dehydrogenase kinase through the use of oxamate and
dichloroacetate, and their prodrugs as a novel approach for cancer
growth inhibition
14:50-15:10
Zhongwu Guo
Xichen Lin （GSK China）
Identification of S1P1 Agonists for the Treatment of Multiple
Sclerosis
15:10-15:30
15:30-15:50
Coffee Break
Yujun Zheng (The University of Georgia)
Bioorthogonal Chemical Probes of Protein Lysine
Acetyltransferases
15:50-16:10
Zongbao Zhao (Dalian Institute of Chemical Physics, Chinese
Academy of Sciences)
Protein methylation in yeast
16:10-16:30
Wenfang Xu
Qingsong Liu (High Magnetic Field Laboratory, Chinese Academy
of Sciences)
Discovery of a super potent BTK kinase inhibitor which induce
strong protein degradation
16:30-16:50
Li Niu (University at Albany, State University of New York)
Developing chemical inhibitors and RNA aptamers against AMPA
receptor channels
16:50-17:10
Peng Chen（Peking University）
Deprotection Chemistry-mediated Protein Activation in Living
Xinyong Liu
Cells
17:10-17:30
Yi Tang (University of California, Los Angeles)
Exciting New Enzymes from Fungal Biosynthetic Pathways
18:00-20:00
Welcome Dinner Reception (重华堂 Chonghua Hall)
Fengshan
Wang
June 17
Section II Bioorganic Chemistry
(Tuesday)
(会谈厅 Meeting Hall)
8:00-8:20
Bin Xu (Virginia Tech)
Chairperson
Molecular Mechanisms of Amylin as a Novel Contributor to
Alzheimer’s Disease and Natural Product Inhibitor Discovery
8:20-8:50
Haibing Zhou (Wuhan University)
Novel Selective Estrogen Receptor Modulators (SERMs):
Qian Wang
Protein-Ligand Interactions and the Dual Regulation Mechanism
Study
8:50-9:10
Luqing Shang (Nankai University)
Discovery of anti-HCV Agents
9:10-9:30
Qian Wang (University of South Carolina)
Probing reversible click reactions at the single-molecule level
9:30-9:50
Xiaohua Peng (University of Wisconsin Milwaukee)
Diwan S
Inducible DNA Cross-Linking Agents as Selective Anticancer
Drugs
9:50-10:10
Rawat
Wei Li (University of Tennessee Health Science Center)
Discovery of novel tubulin inhibitors for metastatic melanoma
10:10-10:30
Coffee Break
10:30-10:50
Diwan S Rawat (University of Delhi)
Identification of Lead Antimalarial Through Rational Drug Design
10:50-11:10
Bingui Wang (Institute of Oceanology, Chinese Academy of
Sciences)
In vitro and in vivo anticancer evaluation of norditerpenoids from
the marine alga-derived endophytic fungus Aspergillus wentii
11:10-11:30
Bin Xu
Dianqing Sun (University of Hawaii at Hilo)
Natural Product-Inspired Novel Antibacterial Agents
11:30-11:50
Bin He (Guiyang Medical University)
Development of Mechanism-based Inhibitors for Sirtuins
12:00-13:00
Buffet (重华堂 Chonghua Hall)
16:00-16:30
Closing Ceremony (拱北楼四楼会议室 The 4th Floor Meeting
Room, Gongbei Building)
18:00-19:00
Buffet (重华堂 Chonghua Hall)
Hao Fang
材料与应用化学分会场（第六会议室）
June 16
Section III Materials and Applied Chemistry
(Monday)
(第六会议室 No.6 Conference Room)
13:30-13:50
Wenfang Sun (North Dakota State University)
Chairperson
Heteroleptic cationic iridium complexes: Synthesis, photophysics
and nonlinear absorption
13:50-14:10
Yonghai Chai (Shanxi Normal University)
New type of aza-MBH reaction and its application to one-pot
Guijun Wang
efficient synthesis of highly substituted dihydropyrroles
14:10-14:30
Guangxi Zhai (Shandong University)
Hyaluronic acid-quercetin conjugate micelles: Synthesis,
characterization, in vitro and in vivo evaluation
14:30-14:50
Guijun Wang (Old Dominion University)
Design, synthesis, and characterization of a series of functional
glycoclusters
14:50-15:10
Jun Li (National University of Singapore)
Wenfang Sun
Smart Supramolecular Nano Drug/Gene Carriers
Self-Assembled from Functional Polymers
15:10-15:30
Coffee Break
15:30-15:50
Xiaogang Liu (National University of Singapore)
Upconversion Nanocrystals: A New Class of Luminescent
Bioprobes
15:50-16:10
Wei Zhang (University of Colorado Boulder)
Novel Shape-Persistent Organic Molecular Cages and Their
Liang Xue
Biological Activity
16:10-16:30
Yongsheng Zhao (Institute of Chemistry, Chinese Academy of
Sciences)
Organic Nanophotonic Materials and Devices
16:30-16:50
Liang Xue (University of the Pacific)
Targeting Telomeric G-quadruplex DNA with Phenanthroline
Based Metal Complexes
16:50-17:10
Jia Sheng (University at Albany, State University of New York)
Crystal Structure Studies of 2’-5’-linked RNA
17:10-17:30
Guodong Liu (North Dakota State University)
Xiaogang Liu
Nucleic Acid-Based Lateral Flow Biosensors for Biomedical and
Environmental Applications
17:30-17:50
Yaoqun Li (Xiamen University)
Hot-spot surface plasmon-coupled directional emission and its
biosensing applications
18:00-20:00
Welcome Dinner Reception (重华堂 Chonghua Hall)
Fengshan
Wang
June 17
Section III Materials and Applied Chemistry
Chairperson
(Tuesday)
(第六会议室 No.6 Conference Room)
8:00-8:20
Jian Liu (University of North Carolina)
Chemoenzymatic synthesis of low molecular weight heparins
8:20-8:50
Yongshu Xie (East China University of Science and Technology)
Ion probes based on linear and macrocyclic polypyrroles
8:50-9:10
Haoru Sun
Jiayu Zhou (Shimadzu China)
新型高效高纯度粉末化技术(C2P)用于化学合成物及天然产物
的纯化与干燥
9:10-9:30
Haoran Sun (University of South Dakota)
Fluorinated Materials for a Sustainable World: from Energy
Harvesting and Storage to Biomedical Applications
9:30-9:50
Hongzhi Cao (Shandong University)
Substrate engineering directed chemoenzymatic synthesis of
Lixin Zhang
sialosides
9:50-10:10
Chu Wang (Peking University)
A Chemoproteomic Platform to Quantitatively Map Targets of
Lipid-derived Electrophiles
10:10-10:30
Coffee Break
10:30-10:50
Lixin Zhang (Institute of Microbiology, Chinese Academy of
Sciences)
Bioprospecting Novel Marine Natural Products for Potential
Anti-infective Drugs
10:50-11:10
Xinjing Tang (Peking University)
Bioorthogonal SERS Nanoprobes for Tumor Targeting and
Spectroscopic Detection
11:10-11:30
Qianbin Li (Central South University)
Novel anti-NSCLC strategy: Dual inhibition of
RAF/MEK/ERK and PI3K/AKT/mTOR signaling pathways
with small molecules
11:30-11:50
Yawen Wang (Lanzhou University)
Jian Liu
Merging of Supramolecular Chemistry Approach and Specific
Reactions: Development of Several Fluorescent Chemosensors
and Chemodosimeters
12:00-13:00
Buffet (重华堂 Chonghua Hall)
16:00-16:30
Closing Ceremony (拱北楼四楼会议室 The 4th Floor Meeting
Room, Gongbei Building)
18:00-19:00
Buffet (重华堂 Chonghua Hall)
Hao Fang