Quizzes (best 2/3)
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Mid-term
30%
Final
50%
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Basic & Clinical Pharmacology, 11th Edition (Bertram G. Katzung, Susan B. Masters,
Anthony J. Trevor)
Principles of Pharmacology: The pathophysiologic Basis of Drug Therapy (David E.
Golan, Armen H. Tashjian. Ehrin J. Armstrong, April W. Armstrong). 3rd Edition I
Rang & Dale's Pharmacology, 6th Edition (H. P. Rang , M.M Dale, J. M. Rod, R. J.
Flower)
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'Goodman & Gilman's The Pharmacological Basis of
Therapeutics, Eleventh Edition( Laurence Brunton, John Lazo, Keith Parker)
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the study of substances (the effect and mechanism ) that interact with living
systems altering body processes%
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Antagonist
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Drug binds Ra>Ri
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Drug binds Ra=Ri
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to agonist will be
depressed
Partial agonist can act as an antagonist…how??
chemically
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substance,
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neutralizing
toxins
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effect of an
agonist
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receptors)
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Ligands must be lipid soluble, eg corticosteroids, …..why?
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